相关参考文献
注意:仅列出部分参考文献,下载原文获取全部文献信息。Characterization of a novel non-steroidal glucocorticoid receptor antagonist
Qun-Yi Li et al.
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS (2010)
Glucocorticoid Dysregulations and Their Clinical Correlates From Receptors to Therapeutics
Andrea H. Marques et al.
GLUCOCORTICOIDS AND MOOD CLINICAL MANIFESTATIONS, RISK FACTORS, AND MOLECULAR MECHANISMS (2009)
Discovery of novel dihydro-9,10-ethano-anthracene carboxamides as glucocorticoid receptor modulators
Bingwei V. Yang et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2009)
Characterization of ZK 245186, a novel, selective glucocorticoid receptor agonist for the topical treatment of inflammatory skin diseases
H. Schaecke et al.
BRITISH JOURNAL OF PHARMACOLOGY (2009)
Glucocorticoids and the risk of osteoporosis
Liron Caplan et al.
EXPERT OPINION ON DRUG SAFETY (2009)
Modulation of glucocorticoid receptor induction properties by cofactors in peripheral blood mononuclear cells
Min Luo et al.
HUMAN IMMUNOLOGY (2009)
Ligand-selective transactivation and transrepression via the glucocorticoid receptor: Role of cofactor interaction
Katharina Ronacher et al.
MOLECULAR AND CELLULAR ENDOCRINOLOGY (2009)
Design and x-ray crystal structures of high-potency nonsteroidal glucocorticoid agonists exploiting a novel binding site on the receptor
Keith Biggadike et al.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2009)
The first X-ray crystal structure of the glucocorticoid receptor bound to a non-steroidal agonist
Kevin P. Madauss et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2008)
Recent developments in the discovery of selective glucocorticoid receptor modulators (SGRMs)
Andrew R. Hudson et al.
CURRENT TOPICS IN MEDICINAL CHEMISTRY (2008)
Recent progress in the discovery of novel glucocorticoid receptor modulators
Hidenori Takahashi et al.
CURRENT TOPICS IN MEDICINAL CHEMISTRY (2008)
Dissociated non-steroidal glucocorticoid receptor modulators: an update on new compounds
Heike Schacke et al.
EXPERT OPINION ON THERAPEUTIC PATENTS (2008)
Novel insights into mechanisms of glucocorticoid action and the development of new glucocorticoid receptor ligands
Mark Lowenberg et al.
STEROIDS (2008)
Genomic and nongenomic effects of glucocorticoids
Cindy Stahn et al.
NATURE CLINICAL PRACTICE RHEUMATOLOGY (2008)
Doubling the size of the glucocorticoid receptor ligand binding pocket by deacylcortivazol
Kelly Suino-Powell et al.
MOLECULAR AND CELLULAR BIOLOGY (2008)
Modulation of glucocorticoid action and the treatment of type-2 diabetes
Jeremy W. Tomlinson et al.
BEST PRACTICE & RESEARCH CLINICAL ENDOCRINOLOGY & METABOLISM (2007)
Glucocorticoids, metabolism and metabolic diseases
Alexandros Vegiopoulos et al.
MOLECULAR AND CELLULAR ENDOCRINOLOGY (2007)
Selective glucocorticoid receptor agonists (SEGRAs): Novel ligands with an improved therapeutic index
Heike Schaecke et al.
MOLECULAR AND CELLULAR ENDOCRINOLOGY (2007)
Effects of glucocorticoids on inflammation and arthritis
Eric F. Morand
CURRENT OPINION IN RHEUMATOLOGY (2007)
Liver-selective glucocorticoid receptor antagonism decreases glucose production and increases glucose disposal, ameliorating insulin resistance
Bradley Zinker et al.
METABOLISM-CLINICAL AND EXPERIMENTAL (2007)
Non-steroidal glucocorticoid receptor antagonists: the race to replace RU-486 for anti-glucocorticoid therapy
Michael L. Mohler et al.
EXPERT OPINION ON THERAPEUTIC PATENTS (2007)
Modelling the glucocorticoid receptor and producing therapeutic agents with anti-inflammatory effects but reduced side-effects
Andrew McMaster et al.
EXPERIMENTAL PHYSIOLOGY (2007)
Corticosteroid design for the treatment of asthma: Structural insights and the therapeutic potential of soft corticosteroids
Nicholas Bodor et al.
CURRENT PHARMACEUTICAL DESIGN (2006)
Controlling nuclear receptors: The circular logic of cofactor cycles
V Perissi et al.
NATURE REVIEWS MOLECULAR CELL BIOLOGY (2005)
Dissociation of transactivation from transrepression by a selective glucocorticoid receptor agonist leads to separation of therapeutic effects from side effects
H Schäcke et al.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2004)
A single amino acid change in the first zinc finger of the DNA binding domain of the glucocorticoid receptor regulates differential promoter selectivity
BM Necela et al.
JOURNAL OF BIOLOGICAL CHEMISTRY (2004)
Glucocorticoid-induced apoptosis and glucocorticoid resistance: molecular mechanisms and clinical relevance
S Schmidt et al.
CELL DEATH AND DIFFERENTIATION (2004)
Principles for modulation of the nuclear receptor superfamily
H Gronemeyer et al.
NATURE REVIEWS DRUG DISCOVERY (2004)
Mechanisms involved in the side effects of glucocorticoids
H Schäcke et al.
PHARMACOLOGY & THERAPEUTICS (2002)
Discovery of potent, nonsteroidal, and highly selective glucocorticoid receptor antagonists
BP Morgan et al.
JOURNAL OF MEDICINAL CHEMISTRY (2002)
Repression of inflammatory responses in the absence of DNA binding by the glucocorticoid receptor
HM Reichardt et al.
EMBO JOURNAL (2001)