4.4 Article

Differential inhibition of PDKs by phenylbutyrate and enhancement of pyruvate dehydrogenase complex activity by combination with dichloroacetate

相关参考文献

注意:仅列出部分参考文献,下载原文获取全部文献信息。
Article Oncology

Phase 1 trial of dichloroacetate (DCA) in adults with recurrent malignant brain tumors

E. M. Dunbar et al.

INVESTIGATIONAL NEW DRUGS (2014)

Article Multidisciplinary Sciences

Structure-based design and mechanisms of allosteric inhibitors for mitochondrial branched-chain α-ketoacid dehydrogenase kinase

Shih-Chia Tso et al.

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2013)

Article Cell Biology

Phenylbutyrate Therapy for Pyruvate Dehydrogenase Complex Deficiency and Lactic Acidosis

Rosa Ferriero et al.

SCIENCE TRANSLATIONAL MEDICINE (2013)

Article Pharmacology & Pharmacy

Clinical and Experimental Applications of Sodium Phenylbutyrate

Tommaso Iannitti et al.

Drugs in research & development (2013)

Editorial Material Oncology

Phenylbutyrate increases activity of pyruvate dehydrogenase complex.

Rosa Ferriero et al.

ONCOTARGET (2013)

Article Endocrinology & Metabolism

Spectrum of neurological and survival outcomes in pyruvate dehydrogenase complex (PDC) deficiency: Lack of correlation with genotype

Suzanne D. DeBrosse et al.

MOLECULAR GENETICS AND METABOLISM (2012)

Article Endocrinology & Metabolism

Urinary phenylacetylglutamine as dosing biomarker for patients with urea cycle disorders

M. Mokhtarani et al.

MOLECULAR GENETICS AND METABOLISM (2012)

Review Genetics & Heredity

Suggested guidelines for the diagnosis and management of urea cycle disorders

Johannes Haeberle et al.

ORPHANET JOURNAL OF RARE DISEASES (2012)

Article Biochemistry & Molecular Biology

Phenylbutyrate therapy for maple syrup urine disease

Nicola Brunetti-Pierri et al.

HUMAN MOLECULAR GENETICS (2011)

Article Cell Biology

Metabolic Modulation of Glioblastoma with Dichloroacetate

E. D. Michelakis et al.

SCIENCE TRANSLATIONAL MEDICINE (2010)

Review Oncology

Dichloroacetate (DCA) as a potential metabolic-targeting therapy for cancer

E. D. Michelakis et al.

BRITISH JOURNAL OF CANCER (2008)

Article Biochemistry & Molecular Biology

Pyruvate dehydrogenase kinase-4 structures reveal a metastable open conformation fostering robust core-free basal activity

R. Max Wynn et al.

JOURNAL OF BIOLOGICAL CHEMISTRY (2008)

Article Biochemistry & Molecular Biology

Pyruvate dehydrogenase complex activity controls metabolic and malignant phenotype in cancer cells

Thomas McFate et al.

JOURNAL OF BIOLOGICAL CHEMISTRY (2008)

Article Biochemistry & Molecular Biology

Induction of pyruvate dehydrogenase kinase-3 by hypoxia-inducible factor-1 promotes metabolic switch and drug resistance

Chun-Wun Lu et al.

JOURNAL OF BIOLOGICAL CHEMISTRY (2008)

Review Biochemistry & Molecular Biology

Pyruvate dehydrogenase kinase regulatory mechanisms and inhibition in treating diabetes, heart ischemia, and cancer

T. E. Roche et al.

CELLULAR AND MOLECULAR LIFE SCIENCES (2007)

Review Endocrinology & Metabolism

Recent advances in mechanisms regulating glucose oxidation at the level of the pyruvate dehydrogenase complex by PDKs

MC Sugden et al.

AMERICAN JOURNAL OF PHYSIOLOGY-ENDOCRINOLOGY AND METABOLISM (2003)

Article Multidisciplinary Sciences

The protein kinase complement of the human genome

G Manning et al.

SCIENCE (2002)

Article Multidisciplinary Sciences

Structure of rat BCKD kinase: Nucleotide-induced domain communication in a mitochondrial protein kinase

M Machius et al.

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2001)

Article Biochemistry & Molecular Biology

Probing the mechanism of inactivation of human pyruvate dehydrogenase by phosphorylation of three sites

LG Korotchkina et al.

JOURNAL OF BIOLOGICAL CHEMISTRY (2001)

Article Biochemistry & Molecular Biology

Marked differences between two isoforms of human pyruvate dehydrogenase kinase

JC Baker et al.

JOURNAL OF BIOLOGICAL CHEMISTRY (2000)

Review Biochemistry & Molecular Biology

GHKL, an emergent ATPase/kinase superfamily

R Dutta et al.

TRENDS IN BIOCHEMICAL SCIENCES (2000)

Article Biochemistry & Molecular Biology

Mechanistic and kinetic studies of inhibition of enzymes

CG Whiteley

CELL BIOCHEMISTRY AND BIOPHYSICS (2000)