4.5 Article

Synthesis and Biological Evaluation of Acridine Derivatives as Antimalarial Agents

相关参考文献

注意:仅列出部分参考文献,下载原文获取全部文献信息。
Article Chemistry, Medicinal

Synthesis and Evaluation of 7-Substituted 4-Aminoquinoline Analogues for Antimalarial Activity

Jong Yeon Hwang et al.

JOURNAL OF MEDICINAL CHEMISTRY (2011)

Article Biochemistry & Molecular Biology

Synthesis, antimalarial activity, and cellular toxicity of new arylpyrrolylaminoquinolines

Manolo Casagrande et al.

BIOORGANIC & MEDICINAL CHEMISTRY (2010)

Article Chemistry, Medicinal

Synthesis of new 4-aminoquinolines and quinoline-acridine hybrids as antimalarial agents

Ashok Kumar et al.

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2010)

Review Biochemistry & Molecular Biology

DNA Topoisomerases and Their Poisoning by Anticancer and Antibacterial Drugs

Yves Pommier et al.

CHEMISTRY & BIOLOGY (2010)

Correction Microbiology

Artemisinin resistance: current status and scenarios for containment (vol 8, pg 272, 2010)

Arjen M. Dondorp et al.

NATURE REVIEWS MICROBIOLOGY (2010)

Article Microbiology

Plasmodium falciparum Na+/H+ Exchanger 1 Transporter Is Involved in Reduced Susceptibility to Quinine

Maud Henry et al.

ANTIMICROBIAL AGENTS AND CHEMOTHERAPY (2009)

Article Microbiology

Atorvastatin Is a Promising Partner for Antimalarial Drugs in Treatment of Plasmodium falciparum Malaria

Veronique Parquet et al.

ANTIMICROBIAL AGENTS AND CHEMOTHERAPY (2009)

Article Biochemistry & Molecular Biology

Antimalarial acridines: Synthesis, in vitro activity against P. falciparum and interaction with hematin

Lucie Guetzoyan et al.

BIOORGANIC & MEDICINAL CHEMISTRY (2009)

Article Chemistry, Medicinal

Antitumour and antimalarial activity of artemisinin-acridine hybrids

Michael Jones et al.

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2009)

Article Chemistry, Medicinal

Identification of acridinyl hydrazides as potent aspartic protease inhibitors

M. Kamran Azim et al.

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2008)

Review Chemistry, Medicinal

Inhibition of efflux of quinolines as new therapeutic strategy in malaria

Maud Henry et al.

CURRENT TOPICS IN MEDICINAL CHEMISTRY (2008)

Article Chemistry, Medicinal

Identification of new functional inhibitors of acid sphingomyelinase using a structure-property-activity relation model

Johannes Kornhuber et al.

JOURNAL OF MEDICINAL CHEMISTRY (2008)

Review Multidisciplinary Sciences

Qinghaosu (Artemisinin): The price of success

N. J. White

SCIENCE (2008)

Article Chemistry, Medicinal

Amine-guanidine switch: A promising approach to improve DNA binding and antiproliferative activities

Keiichiro Ohara et al.

JOURNAL OF MEDICINAL CHEMISTRY (2007)

Review Biotechnology & Applied Microbiology

Genotoxicity of non-covalent interactions: DNA intercalators

Lynnette R. Ferguson et al.

MUTATION RESEARCH-FUNDAMENTAL AND MOLECULAR MECHANISMS OF MUTAGENESIS (2007)

Review Dermatology

New concepts in antimalarial use and mode of action in dermatology

Sunil Kalia et al.

DERMATOLOGIC THERAPY (2007)

Article Pharmacology & Pharmacy

Novel tetra-acridine derivatives as dual inhibitors of topoisomerase II and the human proteasome

S. Vispe et al.

BIOCHEMICAL PHARMACOLOGY (2007)

Article Biochemistry & Molecular Biology

In vitro efficiency of new acridyl derivatives against Plasmodium falciparum

Lucie Guetzoyan et al.

BIOORGANIC & MEDICINAL CHEMISTRY (2007)

Review Medicine, Research & Experimental

Antimalarial drugs inhibiting hemozoin (β-hematin) formation:: A mechanistic update

Sanjay Kumar et al.

LIFE SCIENCES (2007)

Article Biochemistry & Molecular Biology

Synthesis and evaluation of acridine- and acridone-based anti-herpes agents with topoisomerase activity

John R. Goodell et al.

BIOORGANIC & MEDICINAL CHEMISTRY (2006)

Review Pharmacology & Pharmacy

Chloroquine resistance reversal agents as promising antimalarial drugs

Maud Henry et al.

CURRENT DRUG TARGETS (2006)

Article Biochemistry & Molecular Biology

Parallel synthesis of 9-aminoacridines and their evaluation against chloroquine-resistant Plasmodium falciparum

MO Anderson et al.

BIOORGANIC & MEDICINAL CHEMISTRY (2006)

Article Respiratory System

Alternative widely available, inexpensive agents for pleurodesis

O Dikensoy et al.

CURRENT OPINION IN PULMONARY MEDICINE (2005)

Article Chemistry, Medicinal

Arylsulfonyl acridinyl derivatives acting on Plasmodium falciparum

C Santelli-Rouvier et al.

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2004)

Article Microbiology

Antimalarial 9-anilinoacridine compounds directed at hematin

S Auparakkitanon et al.

ANTIMICROBIAL AGENTS AND CHEMOTHERAPY (2003)

Article Obstetrics & Gynecology

Quinacrine sterilization: a retrospective

J Zipper et al.

INTERNATIONAL JOURNAL OF GYNECOLOGY & OBSTETRICS (2003)

Review Pharmacology & Pharmacy

Mode of action and mechanisms of resistance for antimalarial drugs

P Olliaro

PHARMACOLOGY & THERAPEUTICS (2001)