4.5 Article

Synthesis and Biological Evaluation of ortho-Aryl N-Hydroxycinnamides as Potent Histone Deacetylase (HDAC) 8 Isoform-Selective Inhibitors

相关参考文献

注意:仅列出部分参考文献,下载原文获取全部文献信息。
Article Chemistry, Medicinal

Discovery of histone deacetylase 8 selective inhibitors

Weiping Tang et al.

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2011)

Article Biochemistry & Molecular Biology

On the inhibition of histone deacetylase 8

Guillermina Estiu et al.

BIOORGANIC & MEDICINAL CHEMISTRY (2010)

Review Oncology

Isoform-specific histone deacetylase inhibitors: The next step?

Sriram Balasubramanian et al.

CANCER LETTERS (2009)

Article Chemistry, Medicinal

Azetidinones as Zinc-Binding Groups to Design Selective HDAC8 Inhibitors

Paola Galletti et al.

CHEMMEDCHEM (2009)

Review Pharmacology & Pharmacy

Targeting Histone Deacetylases in Neuroblastoma

O. Witt et al.

CURRENT PHARMACEUTICAL DESIGN (2009)

Review Pharmacology & Pharmacy

Targeting of HDAC8 and investigational inhibitors in neuroblastoma

Ina Oehme et al.

EXPERT OPINION ON INVESTIGATIONAL DRUGS (2009)

Article Biochemistry & Molecular Biology

Determination of the class and isoform selectivity of small-molecule histone deacetylase inhibitors

Nagma Khan et al.

BIOCHEMICAL JOURNAL (2008)

Review Chemistry, Medicinal

Histone deacetylase inhibitors: From bench to clinic

Marielle Paris et al.

JOURNAL OF MEDICINAL CHEMISTRY (2008)

Article Multidisciplinary Sciences

HDAC inhibitor PCI-24781 decreases RAD51 expression and inhibits homologous recombination

Shanthi Adimoolam et al.

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2007)

Article Chemistry, Medicinal

Design and evaluation of 'Linkerless' hydroxamic acids as selective HDAC8 inhibitors

Keris KrennHrubec et al.

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2007)

Article Biochemistry & Molecular Biology

Dissecting the biological functions of Drosophila histone deacetylases by RNA interference and transcriptional profiling

Cristiana Foglietti et al.

JOURNAL OF BIOLOGICAL CHEMISTRY (2006)

Article Biochemistry & Molecular Biology

Role of Class I and Class II histone deacetylases in carcinoma cells using siRNA

KB Glaser et al.

BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS (2003)

Article Pharmacology & Pharmacy

Identification of novel isoform-selective inhibitors within class I histone deacetylases

ED Hu et al.

JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS (2003)

Article Biochemistry & Molecular Biology

The inv(16) fusion protein associates with corepressors via a smooth muscle myosin heavy-chain domain

KL Durst et al.

MOLECULAR AND CELLULAR BIOLOGY (2003)

Article Biochemistry & Molecular Biology

A fluorogenic histone deacetylase assay well suited for high-throughput activity screening

D Wegener et al.

CHEMISTRY & BIOLOGY (2003)

Article Biochemistry & Molecular Biology

Cloning and functional characterization of HDAC11, a novel member of the human histone deacetylase family

L Gao et al.

JOURNAL OF BIOLOGICAL CHEMISTRY (2002)