期刊
CHEMISTRY-AN ASIAN JOURNAL
卷 9, 期 8, 页码 2113-2118出版社
WILEY-V C H VERLAG GMBH
DOI: 10.1002/asia.201402071
关键词
arylation; copper; homogeneous catalysis; indoles; synthesis design
资金
- National Natural Science Foundation of China [21025209, 21121062, 21272252, 21332009]
Copper-catalyzed C-2 arylation and vinylation of indole derivatives with iodonium salts have been realized. This method, featuring a simple operational procedure, mild reaction conditions, and a wide substrate scope, provided versatile indole derivatives with direct and selective functionalization at the C-2 position of the indole core. In the presence of excess amounts of iodonium salts, cascade C-2 arylation and dearomatization through the C-3 arylation reaction also proceeded smoothly.
作者
我是这篇论文的作者
点击您的名字以认领此论文并将其添加到您的个人资料中。
推荐
暂无数据