期刊
CHEMICAL COMMUNICATIONS
卷 50, 期 99, 页码 15714-15717出版社
ROYAL SOC CHEMISTRY
DOI: 10.1039/c4cc04508d
关键词
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资金
- National Natural Science Foundation of China [21432003, 81473095, 21272102]
- Key National S&T Program Major New Drug Development of the Ministry of Science and Technology of China [2012ZX09504001-003]
- Program for Changjiang Scholars and Innovative Research Team in University (PCSIRT) [IRT1137]
A direct oxidative cross-dehydrogenative coupling (CDC) of N-aryl tetrahydroisoquinolins with 5H-oxazol-4-ones catalyzed by CuBr using air as the only oxidant has been developed, which could also proceed smoothly under a metal-free oxidative system with PhI(OAc)(2) as the oxidant. A series of alkylated tetrahydroisoquinolin derivatives were obtained in good yields and excellent diastereoselectivities.
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