期刊
CHEMICAL COMMUNICATIONS
卷 47, 期 29, 页码 8355-8357出版社
ROYAL SOC CHEMISTRY
DOI: 10.1039/c1cc12619a
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资金
- National Natural Science Foundation of China [20872153, 21021063, 81025017]
The asymmetric synthesis of syn-beta-substituted tryptophan derivatives was carried out by the Michael addition of chiral equivalent of nucleophilic glycine with sulfonylindoles, and high diastereo- and enantioselectivities were achieved. The resulting adducts were readily converted to syn-beta-substituted tryptophans in 96% yield, indicating that the proposed method is a highly efficient route to chiral syn-beta-substituted tryptophans.
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