4.4 Article

A New i, i+3 Peptide Stapling System for α-Helix Stabilization

相关参考文献

注意:仅列出部分参考文献,下载原文获取全部文献信息。
Article Chemistry, Multidisciplinary

Structure of the Stapled p53 Peptide Bound to Mdm2

Sohee Baek et al.

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2012)

Article Chemistry, Multidisciplinary

Design and Structure of Stapled Peptides Binding to Estrogen Receptors

Chris Phillips et al.

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2011)

Article Biochemical Research Methods

Synthesis of all-hydrocarbon stapled α-helical peptides by ring-closing olefin metathesis

Young-Woo Kim et al.

NATURE PROTOCOLS (2011)

Article Biochemistry & Molecular Biology

The MCL-1 BH3 helix is an exclusive MCL-1 inhibitor and apoptosis sensitizer

Michelle L. Stewart et al.

NATURE CHEMICAL BIOLOGY (2010)

Article Chemistry, Medicinal

Stereochemical effects of all-hydrocarbon tethers in i,i+4 stapled peptides

Young-Woo Kim et al.

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2009)

Article Multidisciplinary Sciences

Direct inhibition of the NOTCH transcription factor complex

Raymond E. Moellering et al.

NATURE (2009)

Review Biochemistry & Molecular Biology

Contemporary strategies for the stabilization of peptides in the α-helical conformation

Laura K. Henchey et al.

CURRENT OPINION IN CHEMICAL BIOLOGY (2008)

Article Biochemistry & Molecular Biology

Solution structure of a hydrocarbon stapled peptide inhibitor in complex with monomeric C-terminal domain of HIV-1 capsid

Shibani Bhattacharya et al.

JOURNAL OF BIOLOGICAL CHEMISTRY (2008)

Article Biochemistry & Molecular Biology

A cell-penetrating helical peptide as a potential HIV-1 inhibitor

Hongtao Zhang et al.

JOURNAL OF MOLECULAR BIOLOGY (2008)

Article Multidisciplinary Sciences

BAX activation is initiated at a novel interaction site

Evripidis Gavathiotis et al.

NATURE (2008)

Article Biochemistry & Molecular Biology

Dual role of proapoptotic BAD in insulin secretion and beta cell survival

Nika N. Danial et al.

NATURE MEDICINE (2008)

Article Chemistry, Multidisciplinary

Facile and E-selective intramolecular ring-closing metathesis reactions in 310-helical peptides:: A 3D structural study

Amie K. Boal et al.

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2007)

Article Biochemistry & Molecular Biology

A stapled BID BH3 helix directly binds and activates BAX

Loren D. Walensky et al.

MOLECULAR CELL (2006)

Article Chemistry, Organic

Solid-phase synthesis of hydrogen-bond surrogate-derived α-helices

G Dimartino et al.

ORGANIC LETTERS (2005)

Article Multidisciplinary Sciences

Activation of apoptosis in vivo by a hydrocarbon-stapled BH3 helix

LD Walensky et al.

SCIENCE (2004)

Article Chemistry, Multidisciplinary

A highly stable short α-helix constrained by a main-chain hydrogen-bond surrogate

RN Chapman et al.

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2004)

Article Chemistry, Multidisciplinary

An all-hydrocarbon cross-linking system for enhancing the helicity and metabolic stability of peptides

CE Schafmeister et al.

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2000)