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BIOORGANIC & MEDICINAL CHEMISTRY (2007)
Carbonic anhydrase inhibitors:: The β-carbonic anhydrase from Helicobacter pylori is a new target for sulfonamide and sulfamate inhibitors
Isao Nishimori et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2007)
Phosph(on)ate as a zinc-binding group in metalloenzyme inhibitors: X-ray crystal structure of the antiviral drug foscarnet complexed to human carbonic anhydrase I
Claudia Temperini et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2007)
Carbonic anhydrase inhibitors: Inhibition of cytosolic/tumor-associated isoforms I, II, and IX with iminodiacetic carboxylates/hydroxamates also incorporating benzenesulfonamide moieties
M. Amelia Santos et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2007)
Carbonic anhydrase and matrix metalloproteinase inhibitors. Inhibition of human tumor-associated isozymes IX and cytosolic isozyme I and II with sulfonylated hydroxamates
Elisa Nuti et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2007)
Saccharin inhibits carbonic anhydrases: Possible explanation for its unpleasant metallic aftertaste
Karen Koehler et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2007)
The development of topically acting carbonic anhydrase inhibitors as antiglaucoma agents
Francesco Mincione et al.
CURRENT TOPICS IN MEDICINAL CHEMISTRY (2007)
Carbonic anhydrase activators. Activation of isozymes I, II, IV, VA, VII, and XIV with L- and D-histidine and crystallographic analysis of their adducts with isoform II: Engineering proton-transfer processes within the active site of an enzyme
Claudia Temperini et al.
CHEMISTRY-A EUROPEAN JOURNAL (2006)
Carbonic anhydrase inhibitors: X-ray and molecular modeling study for the interaction of a fluorescent antitumor sulfonamide with isozyme II and IX
Vincenzo Alterio et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2006)
Ultrahigh resolution crystal structures of human carbonic anhydrases I and II complexed with two-prong inhibitors reveal the molecular basis of high affinity
KM Jude et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2006)
Carbonic anhydrase inhibitors: Valdecoxib binds to a different active site region of the human isoform II as compared to the structurally related cyclooxygenase II 'selective' inhibitor celecoxib
A Di Fiore et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2006)
Carbonic anhydrase inhibitors: Novel sulfonamides incorporating 1,3,5-triazine moieties as inhibitors of the cytosolic and tumour-associated carbonic anhydrase isozymes I, II and IX
V Garaj et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2005)
Spacer-based selectivity in the binding of two-prong ligands to recombinant human carbonic anhydrase I
AL Banerjee et al.
BIOCHEMISTRY (2005)
Carbonic anhydrase inhibitors. Interaction of isozymes I, II, IV, V, and IX with carboxylates
A Innocenti et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2005)
Unexpected nanomolar inhibition of carbonic anhydrase by COX-2-selective celecoxib: New pharmacological opportunities due to related binding site recognition
A Weber et al.
JOURNAL OF MEDICINAL CHEMISTRY (2004)
Carbonic anhydrase inhibitors.: Inhibition of the prokariotic beta and gamma-class enzymes from Archaea with sulfonamides
S Zimmerman et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2004)
Carbonic anhydrase inhibitors. Interaction of isozymes I, II, IV, V, and IX with phosphates, carbamoyl phosphate, and the phosphonate antiviral drug foscarnet
S Rusconi et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2004)
Hypoxia activates the capacity of tumor-associated carbonic anhydrase IX to acidify extracellular pH
E Svastová et al.
FEBS LETTERS (2004)
Carbonic anhydrases: Current state of the art, therapeutic applications and future prospects
S Pastorekova et al.
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (2004)
Carbonic anhydrase inhibitors: synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with sulfonamides incorporating 1,2,4-triazine moieties
V Garaj et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2004)
Protease inhibitors: Synthesis of bacterial collagenase and matrix metalloproteinase inhibitors incorporating succinyl hydroxamate and iminodiacetic acid hydroxamate moieties
MA Santos et al.
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (2003)
Hydroxyurea is a carbonic anhydrase inhibitor
A Scozzafava et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2003)
Carbonic anhydrase inhibitors:: SAR and x-ray crystallographic study for the interaction of sugar sulfamates/sulfamides with Isozymes I, II and IV
A Casini et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2003)
Carbonic anhydrase inhibitors
CT Supuran et al.
MEDICINAL RESEARCH REVIEWS (2003)
Carbonic anhydrase inhibitors. A general approach for the preparation of water-soluble sulfonamides incorporating polyamino-polycarboxylate tails and of their metal complexes possessing long-lasting, topical intraocular pressure-lowering properties
A Scozzafava et al.
JOURNAL OF MEDICINAL CHEMISTRY (2002)
Carbonic anhydrase inhibitors: Water-soluble 4-sulfamoylphenylthioureas as topical intraocular pressure-lowering agents with long-lasting effects
A Casini et al.
JOURNAL OF MEDICINAL CHEMISTRY (2000)
Carbonic anhydrase and matrix metalloproteinase inhibitors:: Sulfonylated amino acid hydroxamates with MMP inhibitory properties act as efficient inhibitors of CA isozymes I, II, and IV, and N-hydroxysulfonamides inhibit both these zinc enzymes
A Scozzafava et al.
JOURNAL OF MEDICINAL CHEMISTRY (2000)
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