相关参考文献
注意:仅列出部分参考文献,下载原文获取全部文献信息。From cradle to twilight: The carboxyl terminus directs the fate of the A2A-adenosine receptor
Simon Keuerleber et al.
BIOCHIMICA ET BIOPHYSICA ACTA-BIOMEMBRANES (2011)
Real-time cellular impedance measurements detect Ca2+ channel-dependent oscillations of morphology in human H295R adrenoma cells
Athanasios Denelavas et al.
BIOCHIMICA ET BIOPHYSICA ACTA-MOLECULAR CELL RESEARCH (2011)
The Protease-activated Receptor-2-specific Agonists 2-Aminothiazol-4-yl-LIGRL-NH2 and 6-Aminonicotinyl-LIGRL-NH2 Stimulate Multiple Signaling Pathways to Induce Physiological Responses in Vitro and in Vivo
Andrea N. Flynn et al.
JOURNAL OF BIOLOGICAL CHEMISTRY (2011)
Agonist-bound adenosine A2A receptor structures reveal common features of GPCR activation
Guillaume Lebon et al.
NATURE (2011)
International Union of Basic and Clinical Pharmacology. LXXXI. Nomenclature and Classification of Adenosine Receptors-An Update
Bertil B. Fredholm et al.
PHARMACOLOGICAL REVIEWS (2011)
Functional selectivity of adenosine receptor ligands
Dennis Verzijl et al.
PURINERGIC SIGNALLING (2011)
Structure of an Agonist-Bound Human A2A Adenosine Receptor
Fei Xu et al.
SCIENCE (2011)
Long-lasting target binding and rebinding as mechanisms to prolong in vivo drug action
Georges Vauquelin et al.
BRITISH JOURNAL OF PHARMACOLOGY (2010)
Evaluation of Cannabinoid Receptor 2 and Metabotropic Glutamate Receptor 1 Functional Responses Using a Cell Impedance-Based Technology
Paola Scandroglio et al.
JOURNAL OF BIOMOLECULAR SCREENING (2010)
SAR of a series of inhaled A2A agonists and comparison of inhaled pharmacokinetics in a preclinical model with clinical pharmacokinetic data
Simon J. Mantell et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2009)
Exploring the Mechanism of Agonist Efficacy: A Relationship between Efficacy and Agonist Dissociation Rate at the Muscarinic M-3 Receptor
David A. Sykes et al.
MOLECULAR PHARMACOLOGY (2009)
Evaluating Cellular Impedance Assays for Detection of GPCR Pleiotropic Signaling and Functional Selectivity
Matthew F. Peters et al.
JOURNAL OF BIOMOLECULAR SCREENING (2009)
Residence time of receptor-ligand complexes and its effect on biological function
Peter J. Tummino et al.
BIOCHEMISTRY (2008)
Inhaled adenosine A2A receptor agonists for the treatment of chronic obstructive pulmonary disease
Simon J. Mantell et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2008)
The application of cell-based label-free technology in drug discovery
Biao Xi et al.
Biotechnology Journal (2008)
Partial agonism at the human α2A-autoreceptor:: role of binding duration
M. Hoeren et al.
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY (2008)
The 2.6 Angstrom Crystal Structure of a Human A2A Adenosine Receptor Bound to an Antagonist
Veli-Pekka Jaakola et al.
SCIENCE (2008)
Impedance-based cellular assay technologies: recent advances, future promise
Ryan McGuinness
CURRENT OPINION IN PHARMACOLOGY (2007)
Emerging adenosine receptor agonists
Zhan-Guo Gao et al.
EXPERT OPINION ON EMERGING DRUGS (2007)
Quantifying the association and dissociation rates of unlabelled antagonists at the muscarinic M3 receptor
Mark R. Dowling et al.
BRITISH JOURNAL OF PHARMACOLOGY (2006)
Opinion - Drug-target residence time and its implications for lead optimization
Robert A. Copeland et al.
NATURE REVIEWS DRUG DISCOVERY (2006)
Slow antagonist dissociation and long-lasting in vivo receptor protection
Georges Vauquelin et al.
TRENDS IN PHARMACOLOGICAL SCIENCES (2006)
Adenosine receptors as therapeutic targets
KA Jacobson et al.
NATURE REVIEWS DRUG DISCOVERY (2006)
Real-time monitoring of morphological changes in living cells by electronic cell sensor arrays: An approach to study G protein-coupled receptors
NC Yu et al.
ANALYTICAL CHEMISTRY (2006)
Biochemical mechanisms of drug action: what does it take for success?
DC Swinney
NATURE REVIEWS DRUG DISCOVERY (2004)
New, non-adenosine, high-potency agonists for the human adenosine A2B receptor with an improved selectivity profile compared to the reference agonist n-ethylcarboxamidoadenosine
MW Beukers et al.
JOURNAL OF MEDICINAL CHEMISTRY (2004)
Modeling the adenosine receptors:: Comparison of the binding domains of A2A agonists and antagonists
SK Kim et al.
JOURNAL OF MEDICINAL CHEMISTRY (2003)
The adenosine A2A receptor interacts with the actin-binding protein α-actinin
J Burgueño et al.
JOURNAL OF BIOLOGICAL CHEMISTRY (2003)
2,8-Disubstituted adenosine derivatives as partial agonists for the adenosine A2A receptor
EW van Tilburg et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2003)
2,5′-disubstituted adenosine derivatives:: Evaluation of selectivity and efficacy for the adenosine A1, A2A, and A3 receptor
EW van Tilburg et al.
JOURNAL OF MEDICINAL CHEMISTRY (2002)
Binding of [3H]MSX-2 (3-(3-hydroxypropyl)-7-methyl-8-(m-methoxystyryl)-1-propargylxanthine) to rat striatal membranes -: a new, selective antagonist radioligand for A2A adenosine receptors
CE Müller et al.
EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES (2000)