期刊
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
卷 15, 期 10, 页码 2533-2536出版社
PERGAMON-ELSEVIER SCIENCE LTD
DOI: 10.1016/j.bmcl.2005.03.055
关键词
DPP-IV
anti-Substituted beta-methylphenylalanine derived amides have been shown to be potent DPP-IV inhibitors exhibiting excellent selectivity over both DPP8 and DPP9. These are among the most potent compounds reported to date lacking an electrophilic trap. The most potent compound among these is 5-oxo-1,2,4-oxadiazole 44, which is a 3 nM DPP-IV inhibitor. (c) 2005 Elsevier Ltd. All rights reserved.
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