期刊
TETRAHEDRON LETTERS
卷 46, 期 34, 页码 5699-5702出版社
PERGAMON-ELSEVIER SCIENCE LTD
DOI: 10.1016/j.tetlet.2005.06.083
关键词
copper; coupling; heteroatom; nucleoside
The synthesis of a series of N-1-aryl inosine and guanosine derivatives is described. The procedure for chemoselective N-1-arylation involves the mild oxidative copper(II) mediated coupling with boronic acids. This approach provides access to substituted N-1-aryl purines with interesting structural characteristics and novel scaffolds for drug discovery. (c) 2005 Elsevier Ltd. All rights reserved.
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