4.8 Article

Multidimensional De Novo Design Reveals 5-HT2B Receptor-Selective Ligands

相关参考文献

注意:仅列出部分参考文献,下载原文获取全部文献信息。
Article Chemistry, Multidisciplinary

Combining On-Chip Synthesis of a Focused Combinatorial Library with Computational Target Prediction Reveals Imidazopyridine GPCR Ligands

Michael Reutlinger et al.

ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2014)

Review Chemistry, Multidisciplinary

Accessing New Chemical Entities through Microfluidic Systems

Tiago Rodrigues et al.

ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2014)

Article Chemistry, Multidisciplinary

Multi-Objective Molecular De Novo Design by Adaptive Fragment Prioritization

Michael Reutlinger et al.

ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2014)

Article Multidisciplinary Sciences

Identifying the macromolecular targets of de novo-designed chemical entities through self-organizing map consensus

Daniel Reker et al.

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2014)

Article Chemistry, Multidisciplinary

Drugs by Numbers: Reaction-Driven De Novo Design of Potent and Selective Anticancer Leads

Birgit Spaenkuch et al.

ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2013)

Article Chemistry, Multidisciplinary

Steering Target Selectivity and Potency by Fragment-Based De Novo Drug Design

Tiago Rodrigues et al.

ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2013)

Article Chemistry, Medicinal

Colloidal Aggregation Causes Inhibition of G Protein-Coupled Receptors

Maria F. Sassano et al.

JOURNAL OF MEDICINAL CHEMISTRY (2013)

Review Chemistry, Multidisciplinary

The past, present and potential for microfluidic reactor technology in chemical synthesis

Katherine S. Elvira et al.

NATURE CHEMISTRY (2013)

Article Biochemical Research Methods

A pharmacological organization of G protein-coupled receptors

Henry Lin et al.

NATURE METHODS (2013)

Article Chemistry, Multidisciplinary

De novo design and optimization of Aurora A kinase inhibitors

Tiago Rodrigues et al.

CHEMICAL SCIENCE (2013)

Article Multidisciplinary Sciences

Automated design of ligands to polypharmacological profiles

Jeremy Besnard et al.

NATURE (2012)

Article Biotechnology & Applied Microbiology

Reducing safety-related drug attrition: the use of in vitro pharmacological profiling

Joanne Bowes et al.

NATURE REVIEWS DRUG DISCOVERY (2012)

Article Biochemistry & Molecular Biology

ChEMBL: a large-scale bioactivity database for drug discovery

Anna Gaulton et al.

NUCLEIC ACIDS RESEARCH (2012)

Article Biochemical Research Methods

DOGS: Reaction-Driven de novo Design of Bioactive Compounds

Markus Hartenfeller et al.

PLOS COMPUTATIONAL BIOLOGY (2012)

Article Chemistry, Multidisciplinary

Neighborhood-Preserving Visualization of Adaptive Structure-Activity Landscapes: Application to Drug Discovery

Michael Reutlinger et al.

ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2011)

Article Pharmacology & Pharmacy

Special Issue: Guide to Receptors and Channels, 5th Edition Abstracts

Stephen P. H. Alexander et al.

BRITISH JOURNAL OF PHARMACOLOGY (2011)

Review Pharmacology & Pharmacy

Drug discovery in the next decade: innovation needed ASAP

Youssef L. Bennani

DRUG DISCOVERY TODAY (2011)

Article Chemistry, Multidisciplinary

An Integrated Synthesis-Purification System to Accelerate the Generation of Compounds in Pharmaceutical Discovery

Jill E. Hochlowski et al.

JOURNAL OF FLOW CHEMISTRY (2011)

Article Chemistry, Medicinal

N-Tetrahydrothiochromenoisoxazole-1-carboxamides as selective antagonists of cloned human 5-HT2B

Yoon Jin Kwon et al.

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2010)

Article Chemistry, Medicinal

Extended-Connectivity Fingerprints

David Rogers et al.

JOURNAL OF CHEMICAL INFORMATION AND MODELING (2010)

Review Medicine, Research & Experimental

The Expanded Biology of Serotonin

Miles Berger et al.

ANNUAL REVIEW OF MEDICINE (2009)

Article Chemistry, Medicinal

A new class of 5-HT2B antagonists possesses favorable potency, selectivity, and rat pharmacokinetic properties

Neil Moss et al.

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2009)

Article Pharmacology & Pharmacy

GPCR Theme Editorial

G. Milligan et al.

BRITISH JOURNAL OF PHARMACOLOGY (2009)

Review Chemistry, Medicinal

In vitro safety pharmacology profiling: what else beyond hERG?

Jacques Hamon et al.

FUTURE MEDICINAL CHEMISTRY (2009)

Article Biochemical Research Methods

FAF-Drugs2: Free ADME/tox filtering tool to assist drug discovery and chemical biology projects

David Lagorce et al.

BMC BIOINFORMATICS (2008)

Review Biochemistry & Molecular Biology

Network pharmacology: the next paradigm in drug discovery

Andrew L. Hopkins

NATURE CHEMICAL BIOLOGY (2008)

Article Biotechnology & Applied Microbiology

Relating protein pharmacology by ligand chemistry

Michael J. Keiser et al.

NATURE BIOTECHNOLOGY (2007)