4.8 Article

Probing the Bioactive Conformation of an Archetypal Natural Product HDAC Inhibitor with Conformationally Homogeneous Triazole-Modified Cyclic Tetrapeptides

期刊

ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
卷 48, 期 26, 页码 4718-4724

出版社

WILEY-V C H VERLAG GMBH
DOI: 10.1002/anie.200805900

关键词

cyclic peptides; drug design; enzyme inhibitors; structure-activity relationships; triazoles

资金

  1. National Science Foundation
  2. NASA Earth and Space Science [NNX07AR35H]
  3. Spanish Ministry for Science and Education
  4. Lundbeck Foundation
  5. Danish Research Council for Technology and Production Sciences [274-06-0317]
  6. National Institute of General Medical Sciences [GM52190]
  7. Skaggs Institute for Chemical Biology
  8. NATIONAL INSTITUTE OF GENERAL MEDICAL SCIENCES [R01GM052190] Funding Source: NIH RePORTER

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