相关参考文献
注意:仅列出部分参考文献,下载原文获取全部文献信息。The GPRC6A receptor displays constitutive internalization and sorting to the slow recycling pathway
Stine Engesgaard Jacobsen et al.
JOURNAL OF BIOLOGICAL CHEMISTRY (2017)
Dynamic monitoring of Gi/o-protein-mediated decreases of intracellular cAMP by FRET-based Epac sensors
Ursula Storch et al.
PFLUGERS ARCHIV-EUROPEAN JOURNAL OF PHYSIOLOGY (2017)
Neuroprotective properties of icariin in MPTP-induced mouse model of Parkinson's disease: Involvement of PI3K/Akt and MEK/ERK signaling pathways
Wen-Fang Chen et al.
PHYTOMEDICINE (2017)
Fluorescence- and bioluminescence-based approaches to study GPCR ligand binding
Leigh A. Stoddart et al.
BRITISH JOURNAL OF PHARMACOLOGY (2016)
Modulation of primary cilia length by melanin-concentrating hormone receptor 1
Akie Hamamoto et al.
CELLULAR SIGNALLING (2016)
ERK activated by Histamine H1 receptor is anti-proliferative through spatial restriction in the cytosol
Ruchi Jain et al.
EUROPEAN JOURNAL OF CELL BIOLOGY (2016)
Desensitization-resistant and -sensitive GPCR-mediated inhibition of GABA release occurs by Ca2+-dependent and -independent mechanisms at a hypothalamic synapse
Reagan L. Pennock et al.
JOURNAL OF NEUROPHYSIOLOGY (2016)
Kinetics of recruitment and allosteric activation of ARHGEF25 isoforms by the heterotrimeric G-protein Gαq
Jakobus van Unen et al.
SCIENTIFIC REPORTS (2016)
The Histamine H3 Receptor: Structure, Pharmacology, and Function
Gustavo Nieto-Alamilla et al.
MOLECULAR PHARMACOLOGY (2016)
Application of BRET to monitor ligand binding to GPCRs
Leigh A. Stoddart et al.
NATURE METHODS (2015)
Pyrosequencing Characterization of the Microbiota from Atlantic Intertidal Marine Sponges Reveals High Microbial Diversity and the Lack of Co-Occurrence Patterns
Anoop Alex et al.
PLOS ONE (2015)
A Perspective on Studying G-Protein-Coupled Receptor Signaling with Resonance Energy Transfer Biosensors in Living Organisms
Jakobus van Unen et al.
MOLECULAR PHARMACOLOGY (2015)
Uncovering Caffeine's Adenosine A(2A) Receptor Inverse Agonism in Experimental Parkinsonism
Victor Fernandez-Duenas et al.
ACS CHEMICAL BIOLOGY (2014)
Histamine H3 Receptor Activation Counteracts Adenosine A2A Receptor-Mediated Enhancement of Depolarization-Evoked [3H]-GABA Release from Rat Globus Pallidus Synaptosomes
Guadalupe-Elide Morales-Figueroa et al.
ACS CHEMICAL NEUROSCIENCE (2014)
Fluorescence-Based Force/Tension Sensors: A Novel Tool to Visualize Mechanical Forces in Structural Proteins in Live Cells
Jun Guo et al.
ANTIOXIDANTS & REDOX SIGNALING (2014)
The evolving small-molecule fluorescent-conjugate toolbox for Class A GPCRs
Andrea J. Vernall et al.
BRITISH JOURNAL OF PHARMACOLOGY (2014)
Engineering Genetically Encoded FRET Sensors
Laurens Lindenburg et al.
SENSORS (2014)
Identification and pharmacological characterization of the histamine H3 receptor in cultured rat astrocytes
Tina Mele et al.
EUROPEAN JOURNAL OF PHARMACOLOGY (2013)
Pitolisant versus placebo or modafinil in patients with narcolepsy: a double-blind, randomised trial
Yves Dauvilliers et al.
LANCET NEUROLOGY (2013)
The histaminergic network in the brain: basic organization and role in disease
Pertti Panula et al.
NATURE REVIEWS NEUROSCIENCE (2013)
Single-cycle kinetic analysis of ternary DNA complexes by surface plasmon resonance on a decaying surface
William Palau et al.
BIOCHIMIE (2012)
Restructuring G-Protein-Coupled Receptor Activation
Martin Audet et al.
CELL (2012)
Mechanical Stress Stimulates Conformational Changes in 5-Hydroxytryptamine Receptor 1B in Bone Cells
Jose Candelario et al.
CELLULAR AND MOLECULAR BIOENGINEERING (2012)
Intramolecular Fluorescence Resonance Energy Transfer (FRET) Sensors of the Orexin OX1 and OX2 Receptors Identify Slow Kinetics of Agonist Activation
Tian-Rui Xu et al.
JOURNAL OF BIOLOGICAL CHEMISTRY (2012)
FRET-Based Detection of M1 Muscarinic Acetylcholine Receptor Activation by Orthosteric and Allosteric Agonists
Danijela Markovic et al.
PLOS ONE (2012)
Identification and Characterization of ZEL-H16 as a Novel Agonist of the Histamine H3 Receptor
Ying Shi et al.
PLOS ONE (2012)
Fluorescence/Bioluminescence Resonance Energy Transfer Techniques to Study G-Protein-Coupled Receptor Activation and Signaling
Martin J. Lohse et al.
PHARMACOLOGICAL REVIEWS (2012)
FRET-based sensors for the human M1-, M3-, and M5-acetylcholine receptors
Nicole Ziegler et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2011)
Ligand-induced internalization of the orexin OX1 and cannabinoid CB1 receptors assessed via N-terminal SNAP and CLIP-tagging
Richard J. Ward et al.
BRITISH JOURNAL OF PHARMACOLOGY (2011)
Real Time FRET Based Detection of Mechanical Stress in Cytoskeletal and Extracellular Matrix Proteins
Fanjie Meng et al.
CELLULAR AND MOLECULAR BIOENGINEERING (2011)
The hydrophobic amino acids in putative helix 8 in carboxy-terminus of histamine H3 receptor are involved in receptor-G-protein coupling
Atsuo Kuramasu et al.
CELLULAR SIGNALLING (2011)
Heteromultimerization of Cannabinoid CB1 Receptor and Orexin OX1 Receptor Generates a Unique Complex in Which Both Protomers Are Regulated by Orexin A
Richard J. Ward et al.
JOURNAL OF BIOLOGICAL CHEMISTRY (2011)
Discovery of Histamine H-3 Antagonists for the Treatment of Cognitive Disorders and Alzheimer's Disease
Jorge D. Brioni et al.
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS (2011)
Developing Chemical Genetic Approaches to Explore G Protein-Coupled Receptor Function: Validation of the Use of a Receptor Activated Solely by Synthetic Ligand (RASSL)
Elisa Alvarez-Curto et al.
MOLECULAR PHARMACOLOGY (2011)
PRE-SYNAPTIC HISTAMINE H3 RECEPTORS MODULATE GLUTAMATERGIC TRANSMISSION IN RAT GLOBUS PALLIDUS
A. Osorio-Espinoza et al.
NEUROSCIENCE (2011)
Histamine H3 Antagonists for Treatment of Cognitive Deficits in CNS Diseases
Rita Raddatz et al.
CURRENT TOPICS IN MEDICINAL CHEMISTRY (2010)
A Fluorescence Resonance Energy Transfer-based M2 Muscarinic Receptor Sensor Reveals Rapid Kinetics of Allosteric Modulation
Monika Maier-Peuschel et al.
JOURNAL OF BIOLOGICAL CHEMISTRY (2010)
Beyond Desensitization: Physiological Relevance of Arrestin-Dependent Signaling
Louis M. Luttrell et al.
PHARMACOLOGICAL REVIEWS (2010)
A Fluorescent Ligand-Binding Alternative Using Tag-lite (R) Technology
Jurriaan M. Zwier et al.
JOURNAL OF BIOMOLECULAR SCREENING (2010)
Fluorescence changes reveal kinetic steps of muscarinic receptor-mediated modulation of phosphoinositides and Kv7.2/7.3 K+ channels
Jill B. Jensen et al.
JOURNAL OF GENERAL PHYSIOLOGY (2009)
A fluorescence energy transfer-based mechanical stress sensor for specific proteins in situ
Fanjie Meng et al.
FEBS JOURNAL (2008)
Histamine in the nervous system
Helmut L. Haas et al.
PHYSIOLOGICAL REVIEWS (2008)
GSK189254, a novel H3 receptor antagonist that binds to histamine H3 receptors in Alzheimer's disease brain and improves cognitive performance in preclinical models
Andrew D. Medhurst et al.
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS (2007)
Real-time analysis of agonist-induced activation of protease-activated receptor 1/Gαi1 protein complex measured by bioluminescence resonance energy transfer in living cells
Mohammed A. Ayoub et al.
MOLECULAR PHARMACOLOGY (2007)
The brain H3-receptor as a novel therapeutic target for vigilance and sleep-wake disorders
R. Parmentier et al.
BIOCHEMICAL PHARMACOLOGY (2007)
Molecular aspects of the histamine H3 receptor
Gerold Bongers et al.
BIOCHEMICAL PHARMACOLOGY (2007)
Fluorescent protein pair emit intracellular FRET signal suitable for FACS screening
Daniel X. Johansson et al.
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS (2007)
G protein coupled receptor structure and activation
Brian K. Kobilka
BIOCHIMICA ET BIOPHYSICA ACTA-BIOMEMBRANES (2007)
A FlAsH-based FRET approach to determine G protein -: coupled receptor activation in living cells
C Hoffmann et al.
NATURE METHODS (2005)
The histamine H3 receptor:: From gene cloning to H3 receptor drugs
R Leurs et al.
NATURE REVIEWS DRUG DISCOVERY (2005)
Characterisation of the binding of [H-3]-SB-674042, a novel nonpeptide antagonist, to the human orexin-1 receptor
CJ Langmead et al.
BRITISH JOURNAL OF PHARMACOLOGY (2004)
Synthesis and structure-activity relationships of conformationally constrained histamine H3 receptor agonists
R Kitbunnadaj et al.
JOURNAL OF MEDICINAL CHEMISTRY (2003)
Two novel and selective nonimidazole histamine H3 receptor antagonists A-304121 and A-317920:: I.: In vitro pharmacological effects
TA Esbenshade et al.
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS (2003)
FRET imaging
EA Jares-Erijman et al.
NATURE BIOTECHNOLOGY (2003)
Characteristics of recombinantly expressed rat and human histamine H3 receptors
BS Wulff et al.
EUROPEAN JOURNAL OF PHARMACOLOGY (2002)
Histamine H3 receptor activation inhibits glutamate release from rat striatal synaptosomes
A Molina-Hernández et al.
NEUROPHARMACOLOGY (2001)
Imaging protein-protein interactions using fluorescence resonance energy transfer microscopy
AK Kenworthy
METHODS (2001)
Discovery of a novel member of the histamine receptor family
T Nguyen et al.
MOLECULAR PHARMACOLOGY (2001)
Cloning and pharmacological characterization of a fourth histamine receptor (H4) expressed in bone marrow
CL Liu et al.
MOLECULAR PHARMACOLOGY (2001)