相关参考文献
注意:仅列出部分参考文献,下载原文获取全部文献信息。Systematic Tuning of Fluoro-galectin-3 Interactions Provides Thiodigalactoside Derivatives with Single-Digit nM Affinity and High Selectivity
Kristoffer Peterson et al.
JOURNAL OF MEDICINAL CHEMISTRY (2018)
Insights into Thiol-Aromatic Interactions: A Stereoelectronic Basis for S-H/π Interactions
Christina R. Forbes et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2017)
Galectins: emerging regulatory checkpoints linking tumor immunity and angiogenesis
Santiago P. Mendez-Huergo et al.
CURRENT OPINION IN IMMUNOLOGY (2017)
Galectin-3-Binding Glycomimetics that Strongly Reduce Bleomycin-Induced Lung Fibrosis and Modulate Intracellular Glycan Recognition
Tamara Delaine et al.
CHEMBIOCHEM (2016)
The Halogen Bond
Gabriella Cavallo et al.
CHEMICAL REVIEWS (2016)
Recent Developments of C-Aryl Glucoside SGLT2 Inhibitors
Yang Zhang et al.
CURRENT MEDICINAL CHEMISTRY (2016)
FimH Antagonists: Phosphate Prodrugs Improve Oral Bioavailability
Simon Kleeb et al.
JOURNAL OF MEDICINAL CHEMISTRY (2016)
Recent Developments in Synthetic Carbohydrate-Based Diagnostics, Vaccines, and Therapeutics
Alberto Fernandez-Tejada et al.
CHEMISTRY-A EUROPEAN JOURNAL (2015)
A Survey of the Role of Noncovalent Sulfur Interactions in Drug Design
Brett R. Beno et al.
JOURNAL OF MEDICINAL CHEMISTRY (2015)
FimH Antagonists: Bioisosteres To Improve the in Vitro and in Vivo PK/PD Profile
Simon Kleeb et al.
JOURNAL OF MEDICINAL CHEMISTRY (2015)
Discovery of Multifold Modified Sialosides as Human CD22/Siglec-2 Ligands with Nanomolar Activity on B-Cells
Horst Prescher et al.
ACS CHEMICAL BIOLOGY (2014)
Synthesis and evaluation of iminocoumaryl and coumaryl derivatized glycosides as galectin antagonists
Vishal Kumar Rajput et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2014)
Glycotherapy: New Advances Inspire a Reemergence of Glycans in Medicine
Jason E. Hudak et al.
CHEMISTRY & BIOLOGY (2014)
Nanomolar E-Selectin Antagonists with Prolonged Half-Lives by a Fragment-Based Approach
Jonas Egger et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2013)
When Galectins Recognize Glycans: From Biochemistry to Physiology and Back Again
Santiago Di Lella et al.
BIOCHEMISTRY (2011)
1H-1,2,3-Triazol-1-yl thiodigalactoside derivatives as high affinity galectin-3 inhibitors
Bader A. Salameh et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2010)
Lactose Binding to Galectin-1 Modulates Structural Dynamics, Increases Conformational Entropy, and Occurs with Apparent Negative Cooperativity
Irina V. Nesmelova et al.
JOURNAL OF MOLECULAR BIOLOGY (2010)
Protein Flexibility and Conformational Entropy in Ligand Design Targeting the Carbohydrate Recognition Domain of Galectin-3
Carl Diehl et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2010)
From carbohydrate leads to glycomimetic drugs
Beat Ernst et al.
NATURE REVIEWS DRUG DISCOVERY (2009)
Double affinity amplification of galectin-ligand interactions through arginine-arene interactions: Synthetic, thermodynamic, and computational studies with aromatic diamido thiodigalactosides
Ian Cumpstey et al.
CHEMISTRY-A EUROPEAN JOURNAL (2008)
Galectin-Inhibitory Thiodigalactoside Ester Derivatives Have Antimigratory Effects in Cultured Lung and Prostate Cancer Cells
Tamara Delaine et al.
JOURNAL OF MEDICINAL CHEMISTRY (2008)
Studies of arginine-arene interactions through synthesis and evaluation of a series of galectin-binding aromatic lactose esters
Ian Cumpstey et al.
CHEMBIOCHEM (2007)
Global changes in local protein dynamics reduce the entropic cost of carbohydrate binding in the arabinose-binding protein
Christopher A. MacRaild et al.
JOURNAL OF MOLECULAR BIOLOGY (2007)
Antiviral agents active against influenza A viruses
Erik De Clercq
NATURE REVIEWS DRUG DISCOVERY (2006)
Structural and thermodynamic studies on cation -: II: interactions in lectin-ligand complexes:: High-affinity galectin-3 inhibitors through fine-tuning of an arginine-arene interaction
P Sörme et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2005)
Synthesis of a phenyl thio-beta-D-galactopyranoside library from 1,5-difluoro-2,4-dinitrobenzene: discovery of effcient and selective monosaccharide inhibitors of galectin-7
I Cumpstey et al.
ORGANIC & BIOMOLECULAR CHEMISTRY (2005)
C-2-symmetrical thiodigalactoside bis-benzamido derivatives as high-affinity inhibitors of galectin-3: efficient lectin inhibition through double arginine-arene interactions
I Cumpstey et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2005)
A synthetic antithrombin III binding pentasaccharide is now a drug! What comes next?
M Petitou et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2004)
The ligand-binding domain of CD22 is needed for inhibition of the B cell receptor signal, as demonstrated by a novel human CD22-specific inhibitor compound
S Kelm et al.
JOURNAL OF EXPERIMENTAL MEDICINE (2002)