4.8 Article

High-Throughput Kinetic Analysis for Target-Directed Covalent Ligand Discovery

相关参考文献

注意:仅列出部分参考文献,下载原文获取全部文献信息。
Article Biochemistry & Molecular Biology

Chemical Proteomics Identifies Druggable Vulnerabilities in a Genetically Defined Cancer

Liron Bar-Peled et al.

Editorial Material Chemistry, Medicinal

Hope and Disappointment: Covalent Inhibitors to Overcome Drug Resistance in Non-Small Cell Lung Cancer

Julian Engel et al.

ACS MEDICINAL CHEMISTRY LETTERS (2016)

Article Multidisciplinary Sciences

Proteome-wide covalent ligand discovery in native biological systems

Keriann M. Backus et al.

NATURE (2016)

Article Chemistry, Multidisciplinary

A Small Molecule That Switches a Ubiquitin Ligase From a Processive to a Distributive Enzymatic Mechanism

Stefan G. Kathman et al.

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2015)

Review Biotechnology & Applied Microbiology

The history and future of targeting cyclin-dependent kinases in cancer therapy

Uzma Asghar et al.

NATURE REVIEWS DRUG DISCOVERY (2015)

Article Chemistry, Medicinal

A Fragment-Based Method to Discover Irreversible Covalent Inhibitors of Cysteine Proteases

Stefan G. Kathman et al.

JOURNAL OF MEDICINAL CHEMISTRY (2014)

Article Chemistry, Multidisciplinary

Design of Reversible, Cysteine-Targeted Michael Acceptors Guided by Kinetic and Computational Analysis

Shyam Krishnan et al.

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2014)

Article Biochemical Research Methods

Comparative studies of thiol-sensitive fluorogenic probes for HAT assays

Tielong Gao et al.

ANALYTICAL AND BIOANALYTICAL CHEMISTRY (2013)

Review Pharmacology & Pharmacy

αC helix displacement as a general approach for allosteric modulation of protein kinases

Lorenzo Palmieri et al.

DRUG DISCOVERY TODAY (2013)

Article Biochemistry & Molecular Biology

Fragment-Based Approaches in Drug Discovery and Chemical Biology

Duncan E. Scott et al.

BIOCHEMISTRY (2012)

Review Biochemistry & Molecular Biology

Structural Biology and Drug Discovery of Difficult Targets: The Limits of Ligandability

Sachin Surade et al.

CHEMISTRY & BIOLOGY (2012)

Article Chemistry, Medicinal

Kinetic Template-Guided Tethering of Fragments

Rebecca H. Nonoo et al.

CHEMMEDCHEM (2012)

Article Biochemistry & Molecular Biology

Discovery of a Potential Allosteric Ligand Binding Site in CDK2

Stephane Betzi et al.

ACS CHEMICAL BIOLOGY (2011)

Article Biochemistry & Molecular Biology

A miniaturized technique for assessing protein thermodynamics and function using fast determination of quantitative cysteine reactivity

Daniel G. Isom et al.

PROTEINS-STRUCTURE FUNCTION AND BIOINFORMATICS (2011)

Review Chemistry, Multidisciplinary

Copper-catalyzed azide-alkyne cycloaddition (CuAAC) and beyond: new reactivity of copper(I) acetylides

Jason E. Hein et al.

CHEMICAL SOCIETY REVIEWS (2010)

Review Chemistry, Multidisciplinary

Fluorescent and colorimetric probes for detection of thiols

Xiaoqiang Chen et al.

CHEMICAL SOCIETY REVIEWS (2010)

Article Chemistry, Multidisciplinary

Sensitized detection of inhibitory fragments and iterative development of non-peptidic protease inhibitors by dynamic Ligation screening

Marco Florian Schmidt et al.

ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2008)

Article Chemistry, Multidisciplinary

Oxidation of thiol compounds by molecular oxygen in aqueous solutions

GA Bagiyan et al.

RUSSIAN CHEMICAL BULLETIN (2003)

Article Biochemical Research Methods

A competitive fluorescence assay to measure the reactivity of compounds

DE Epps et al.

ANALYTICAL BIOCHEMISTRY (2001)