期刊
ORGANIC & BIOMOLECULAR CHEMISTRY
卷 15, 期 28, 页码 6033-6041出版社
ROYAL SOC CHEMISTRY
DOI: 10.1039/c7ob01149k
关键词
-
资金
- National Natural Science Foundation of China [21572200]
- Fundamental Research Funds for the Central Universities [2017QNA3013]
A highly enantioselective aza-Friedel-Crafts reaction of N-sulfonyl cyclic ketimines with indoles catalyzed by chiral phosphoric acids has been developed. This methodology provides an efficient and facile route to indole-containing chiral cyclic alpha-amino acid derivatives bearing a quaternary stereocenter in high yields and up to 98% enantioselectivity.
作者
我是这篇论文的作者
点击您的名字以认领此论文并将其添加到您的个人资料中。
推荐
暂无数据