期刊
ORGANIC & BIOMOLECULAR CHEMISTRY
卷 18, 期 2, 页码 305-315出版社
ROYAL SOC CHEMISTRY
DOI: 10.1039/c9ob02445j
关键词
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资金
- Academia Sinica [AS-SUMMIT-108]
- Ministry of Science and Technology [MOST 108-3114Y-001-002]
This study describes an efficient protocol for the preparation of substituted 2,4-diaryl-3-sulfonylquinolines from functionalized 2-aminobenzophenones and aromatic beta-ketosulfones by using p-toluenesulfonic acid monohydrate under microwave irradiation. In this atom-economical synthetic route, a series of pharmaceutically active 3-arylsulfonylquinolines with good functional group tolerance are prepared in good to excellent yields. Some structures are confirmed by single-crystal X-ray diffraction analysis.
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