期刊
ORGANIC CHEMISTRY FRONTIERS
卷 7, 期 16, 页码 2278-2283出版社
ROYAL SOC CHEMISTRY
DOI: 10.1039/d0qo00507j
关键词
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资金
- National Natural Science Foundation of China [21702013]
- Fundamental Research Funds for the Central Universities at BUCT [XK1802-6, buctrc201721]
- Beijing Key Laboratory of Flavor Chemistry, Beijing Technology and Business University (BTBU), Beijing, China [SPFW2019YB06]
A platform approach for the direct synthesis of 3-substituted 2H-indazole derivatives has been developed using a Ag(i)/Na(2)S(2)O(8)system. This regioselective alkylation/acylation protocol operates under mild conditions, tolerates a wide range of structural moieties and delivers versatile 2H-indazole derivatives with high efficiency. The gram-scale reaction and the application to the synthesis of bioactive molecules further demonstrate the utility of our protocol.
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