期刊
CHINESE JOURNAL OF ORGANIC CHEMISTRY
卷 40, 期 8, 页码 2476-2482出版社
SCIENCE PRESS
DOI: 10.6023/cjoc202002042
关键词
benzothiazole; arylation; diaryliodonium salt; cross coupling; C-H activation
资金
- National Natural Science Foundation of China [21262028, 21762039, 21762040]
Diaryliodonium salts have low toxicity and good stability, and their mediated reactions often have advantages of mild reaction conditions and high selectivity. They have received extensive attention and have been widely used as arylating agents in organic synthesis. A simple and efficient method for the synthesis of 2-arylbenzothiazole derivatives via copper-catalyzed C-H direct arylation of benzothiazoles with diaryliodonium salts as electrophilic arylating reagents was developed. This method shows wide range of substrates, good group tolerance, simple operation and high product yields.
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