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N,N-Dimethyl-S-difluoromethyl-S-phenylsulfoximinium tetrafluoroborate: A versatile electrophilic difluoromethylating reagent
G. K. Surya Prakash et al.
JOURNAL OF FLUORINE CHEMISTRY (2011)
Synthesis and Biological Evaluation of Novel Analogues of the Pan Class I Phosphatidylinositol 3-Kinase (PI3K) Inhibitor 2-(Difluoromethyl)-1-[4,6-di(4-morpholinyl)-1,3,5-triazin-2-yl]-1H-benzimidazole (ZSTK474)
Gordon W. Rewcastle et al.
JOURNAL OF MEDICINAL CHEMISTRY (2011)
Efficient and Direct Nucleophilic Difluoromethylation of Carbonyl Compounds and Imines with Me3SiCF2H at Ambient or Low Temperature
Yanchuan Zhao et al.
ORGANIC LETTERS (2011)
A New Method for Aromatic Difluoromethylation: Copper-Catalyzed Cross-Coupling and Decarboxylation Sequence from Aryl Iodides
Kenichi Fujikawa et al.
ORGANIC LETTERS (2011)
Transition-Metal-Catalyzed Trifluoromethylation of Aryl Halides
Rylan J. Lundgren et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2010)
Discovery of 4-tert-Butyl-2,6-dimethylphenylsulfur Trifluoride as a Deoxofluorinating Agent with High Thermal Stability as Well as Unusual Resistance to Aqueous Hydrolysis, and Its Diverse Fluorination Capabilities Including Deoxofluoro-Arylsulfinylation with High Stereoselectivity
Teruo Umemoto et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2010)
Transition-Metal-Mediated Reactions for Csp2-F Bond Construction: The State of Play
John M. Brown et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2009)
Aminodifluorosulfinium Tetrafluoroborate Salts as Stable and Crystalline Deoxofluorinating Reagents
Francis Beaulieu et al.
ORGANIC LETTERS (2009)
N-Tosyl-S-difluoromethyl-S-phenylsulfoximine: A New Difluoromethylation Reagent for S-, N-, and C-Nucleophiles
Wei Zhang et al.
ORGANIC LETTERS (2009)
Diethyl bromodifluoromethylphosphonate: a highly efficient and environmentally benign difluorocarbene precursor
Yossi Zafrani et al.
TETRAHEDRON (2009)
Understanding organofluorine chemistry. An introduction to the C-F bond
David O'Hagan
CHEMICAL SOCIETY REVIEWS (2008)
Fluorine in medicinal chemistry
Sophie Purser et al.
CHEMICAL SOCIETY REVIEWS (2008)
The preparation of HCF2CdX and HCF2ZnX via direct insertion into the carbon halogen bond of CF2HY (Y = Br, I)
Donald J. Burton et al.
JOURNAL OF FLUORINE CHEMISTRY (2007)
Fluorine in pharmaceuticals:: Looking beyond intuition
Klaus Mueller et al.
SCIENCE (2007)
Chlorodifluoromethyl phenyl sulfone: a novel non-ozone-depleting substance-based difluorocarbene reagent for O- and N-difluoromethylations
Ji Zheng et al.
CHEMICAL COMMUNICATIONS (2007)
2-chloro-2,2-difluoroacetophenone: A non-ODS-based difluorocarbene precursor and its use in the difluoromethylation of phenol derivatives
Laijun Zhang et al.
JOURNAL OF ORGANIC CHEMISTRY (2006)
Facile Ar-CF3 bond formation at Pd.: Strikingly different outcomes of reductive elimination from [(Ph3P)2Pd(CF3)Ph] and [(Xantphos)Pd(CF3)Ph]
Vladimir V. Grushin et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2006)
Facile one-pot synthesis of N-difluoromethyl-2-pyridone derivatives
Makoto Ando et al.
ORGANIC LETTERS (2006)
NMR method for the determination of solute hydrogen bond acidity
MH Abraham et al.
JOURNAL OF ORGANIC CHEMISTRY (2006)
Unexpected H2O-induced Ar-X activation with trifluoromethylpalladium(II) aryls
VV Grushin et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2006)
Reactions of aliphatic fluoro-alcohols with CHClF2 at atmospheric pressure
J Mizukado et al.
JOURNAL OF FLUORINE CHEMISTRY (2006)
Recent changes in the production and global atmospheric emissions of chlorodifluoromethane (HCFC-22)
A McCulloch et al.
ATMOSPHERIC ENVIRONMENT (2006)
Insertion reactions of difluorocarbene generated by pyrolysis of hexafluoropropene oxide to O-H bond
J Mizukado et al.
JOURNAL OF FLUORINE CHEMISTRY (2005)
Carbon-carbon bond-forming reductive elimination from arylpalladium complexes containing functionalized alkyl groups. Influence of ligand steric and electronic properties on structure, stability, and reactivity
DA Culkin et al.
ORGANOMETALLICS (2004)
Difluoromethylation of sulfonamides
KI Petko et al.
RUSSIAN JOURNAL OF ORGANIC CHEMISTRY (2002)
Novel fluorination reagent:: IF5/Et3N-3HF
N Yoneda et al.
CHEMISTRY LETTERS (2001)
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