4.6 Article

Structure-activity relationship, in vitro and in vivo evaluation of novel dienyl sulphonyl fluorides as selective BuChE inhibitors for the treatment of Alzheimer's disease

相关参考文献

注意:仅列出部分参考文献,下载原文获取全部文献信息。
Review Clinical Neurology

Aging and Alzheimer's disease pathology

Renpei Sengoku

NEUROPATHOLOGY (2020)

Article Chemistry, Applied

An Easy, General and Practical Method for the Construction of Alkyl Sulfonyl Fluorides

Xu Zhang et al.

ADVANCED SYNTHESIS & CATALYSIS (2020)

Article Chemistry, Medicinal

New deferiprone derivatives as multi-functional cholinesterase inhibitors: design, synthesis and in vitro evaluation

Martina Bortolami et al.

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2020)

Article Biochemistry & Molecular Biology

Developing Covalent Protein Drugs via Proximity-Enabled Reactive Therapeutics

Qingke Li et al.

Article Chemistry, Medicinal

Discovery and Biological Evaluation of a Novel Highly Potent Selective Butyrylcholinsterase Inhibitor

Qi Li et al.

JOURNAL OF MEDICINAL CHEMISTRY (2020)

Review Neurosciences

Synergy between amyloid-β and tau in Alzheimer's disease

Marc Aurel Busche et al.

NATURE NEUROSCIENCE (2020)

Article Chemistry, Medicinal

The structure-based optimization of δ-sultone-fused pyrazoles as selective BuChE inhibitors

Ziwen Zhang et al.

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2020)

Article Chemistry, Organic

Protocol for Stereoselective Construction of Highly Functionalized Dienyl Sulfonyl Fluoride Warheads

Zai-Wei Zhang et al.

JOURNAL OF ORGANIC CHEMISTRY (2020)

Article Clinical Neurology

2020 Alzheimer's disease facts and figures

[Anonymous]

ALZHEIMERS & DEMENTIA (2020)

Article Biochemistry & Molecular Biology

Piperine attenuates cognitive impairment in an experimental mouse model of sporadic Alzheimer's disease

Che Wang et al.

JOURNAL OF NUTRITIONAL BIOCHEMISTRY (2019)

Review Chemistry, Multidisciplinary

The growing applications of SuFEx click chemistry

A. S. Barrow et al.

CHEMICAL SOCIETY REVIEWS (2019)

Article Chemistry, Medicinal

BACE-1 Inhibitors: From Recent Single-Target Molecules to Multitarget Compounds for Alzheimer's Disease

Federica Prati et al.

JOURNAL OF MEDICINAL CHEMISTRY (2018)

Review Chemistry, Medicinal

Donepezil-based multi-functional cholinesterase inhibitors for treatment of Alzheimer's disease

Qi Li et al.

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2018)

Article Biochemistry & Molecular Biology

Ethenesulfonyl fluoride derivatives as telomerase inhibitors: structure-based design, SAR, and anticancer evaluation in vitro

Xing Chen et al.

JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (2018)

Article Biochemistry & Molecular Biology

Design, synthesis and biological evaluation of tricyclic pyrazolo[1,5-c][1,3]benzoxazin-5(5H)-one scaffolds as selective BuChE inhibitors

Guo-Liang Qiu et al.

JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (2018)

Article Biochemistry & Molecular Biology

Synthesis and bioevaluation of new tacrine-cinnamic acid hybrids as cholinesterase inhibitors against Alzheimer's disease

Yao Chen et al.

JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (2017)

Article Behavioral Sciences

Learning performances and vulnerability to amyloid toxicity in the butyrylcholinesterase knockout mouse

Tangui Maurice et al.

BEHAVIOURAL BRAIN RESEARCH (2016)

Article Biochemistry & Molecular Biology

Proteasome inhibition by new dual warhead containing peptido vinyl sulfonyl fluorides

Arwin J. Brouwer et al.

BIOORGANIC & MEDICINAL CHEMISTRY (2016)

Article Neurosciences

Alzheimer's Disease: Targeting the Cholinergic System

Talita H. Ferreira-Vieira et al.

CURRENT NEUROPHARMACOLOGY (2016)

Article Chemistry, Medicinal

Versatility of the Curcumin Scaffold: Discovery of Potent and Balanced Dual BACE-1 and GSK-3β Inhibitors

Rita Maria Concetta Di Martino et al.

JOURNAL OF MEDICINAL CHEMISTRY (2016)

Review Medicine, General & Internal

Alzheimer's disease

Philip Scheltens et al.

LANCET (2016)

Review Chemistry, Multidisciplinary

Sulfur(VI) Fluoride Exchange (SuFEx): Another Good Reaction for Click Chemistry

Jiajia Dong et al.

ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2014)

Review Chemistry, Multidisciplinary

BACE1 (beta-secretase) inhibitors for the treatment of Alzheimer's disease

Arun K. Ghosh et al.

CHEMICAL SOCIETY REVIEWS (2014)

Article Chemistry, Medicinal

Oxidative Stress in Alzheimer's Disease: Are We Connecting the Dots?

Michela Rosini et al.

JOURNAL OF MEDICINAL CHEMISTRY (2014)

Article Chemistry, Medicinal

De novo tyrosinase inhibitor: 4-(6,7-Dihydro-5H-indeno[5,6-d]thiazol-2-yl) benzene-1,3-diol (MHY1556)

June Whan Park et al.

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2013)

Review Behavioral Sciences

The history of the cholinergic hypothesis

Antonio Contestabile

BEHAVIOURAL BRAIN RESEARCH (2011)

Article Behavioral Sciences

Butyrylcholinesterase inhibitors ameliorate cognitive dysfunction induced by amyloid-β peptide in mice

Yoko Furukawa-Hibi et al.

BEHAVIOURAL BRAIN RESEARCH (2011)

Article Biochemical Research Methods

Morris water maze: procedures for assessing spatial and related forms of learning and memory

Charles V. Vorhees et al.

NATURE PROTOCOLS (2006)

Article Multidisciplinary Sciences

Selective butyrylcholinesterase inhibition elevates brain acetylcholine, augments learning and lowers Alzheimer β-amyloid peptide in rodent

NH Greig et al.

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2005)

Article Chemistry, Medicinal

High throughput artificial membrane permeability assay for blood-brain barrier

L Di et al.

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2003)