相关参考文献
注意：仅列出部分参考文献，下载原文获取全部文献信息。Novel 2-indolinone thiazole hybrids as sunitinib analogues: Design, synthesis, and potent VEGFR-2 inhibition with potential anti-renal cancer activity
Huda K. Mahmoud et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2020)
Synthesis of indole-tethered [1,3,4]thiadiazolo and [1,3,4]oxadiazolo[3,2-a] pyrimidin-5-one hybrids as anti-pancreatic cancer agents
Lalitha Gummidi et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2020)
New NSAID-Pt(IV) prodrugs to suppress metastasis and invasion of tumor cells and enhance anti-tumor effect in vitro and in vivo
Xue-Qing Song et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2019)
Synthesis of Thymoquinone-Artemisinin Hybrids: New Potent Antileukemia, Antiviral, and Antimalarial Agents
Tony Froehlich et al.
ACS MEDICINAL CHEMISTRY LETTERS (2018)
A novel penicillin derivative induces antitumor effect in melanoma cells
Viviana Blank et al.
ANTI-CANCER DRUGS (2018)
Structure-based design, synthesis, and evaluation of structurally rigid donepezil analogues as dual AChE and BACE-1 inhibitors
Moustafa T. Gabr et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2018)
Discovery of Novel 2-Amino-5-(Substituted)-1,3,4-Thiadiazole Derivatives: New Utilities for Colon Cancer Treatment
Vinit Raj et al.
ANTI-CANCER AGENTS IN MEDICINAL CHEMISTRY (2018)
Synthesis and biological evaluation of a library of hybrid derivatives as inhibitors of influenza virus PA-PB1 interaction
Ilaria D'Agostino et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2018)
Recent advances (2015-2016) in anticancer hybrids
Nagaraju Kerru et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2017)
Carbon Tetrabromide/Triphenylphosphine-Activated Beckmann Rearrangement of Ketoximes for Synthesis of Amides
Peng Gao et al.
CHINESE JOURNAL OF CHEMISTRY (2017)
Cancer Immunotherapy: Selected Targets and Small-Molecule Modulators
Hilmar Weinmann
CHEMMEDCHEM (2016)
Synthesis and Biological Evaluation of 2-methoxy-N-phenyl-6-(5-phenyl-1,3,4-oxadiazol-2-yl) pyridin-3-amine Derivatives as Antimicrobial Agents
Vasu Namani et al.
LETTERS IN ORGANIC CHEMISTRY (2016)
Synthesis and Biological Activities of Oxadiazole Derivatives: A Review
Ankur Vaidya et al.
MINI-REVIEWS IN MEDICINAL CHEMISTRY (2016)
5-Hydroxy-7-azaindolin-2-one, a novel hybrid of pyridinol and sunitinib: design, synthesis and cytotoxicity against cancer cells
Sajita Shah et al.
ORGANIC & BIOMOLECULAR CHEMISTRY (2016)
Synthesis and Biological Evaluation of Novel Series of 3-Substituted 2-Methoxy-6-(5-phenyl-[1,3,4]oxadiazol-2-yl)pyridine Derivatives as Antimicrobial Agents
Vasu Namani et al.
ASIAN JOURNAL OF CHEMISTRY (2015)
Synthesis, molecular modeling, and biological evaluation of quinazoline derivatives containing the 1,3,4-oxadiazole scaffold as novel inhibitors of VEGFR2
Fang Qiao et al.
RSC ADVANCES (2015)
Synthesis of 1,3,4-oxadiazole derivatives from α-amino acid and acyl hydrazides under thermal heating or microwave irradiation conditions
Luciano Dornelles et al.
ARKIVOC (2015)
Discovery and characterization of AZD9272 and AZD6538-Two novel mGluR5 negative allosteric modulators selected for clinical development
Patrick Raboisson et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2012)
Diversity-oriented synthesis: producing chemical tools for dissecting biology
Cornelius J. O'Connor et al.
CHEMICAL SOCIETY REVIEWS (2012)
Oxadiazoles in Medicinal Chemistry
Jonas Bostrom et al.
JOURNAL OF MEDICINAL CHEMISTRY (2012)
Chemoselective Schmidt Reaction Mediated by Triflic Acid: Selective Synthesis of Nitriles from Aldehydes
Balaji V. Rokade et al.
JOURNAL OF ORGANIC CHEMISTRY (2012)
Synthetic Approaches and Pharmacological Activity of 1,3,4-Oxadiazoles: A Review of the Literature from 2000-2012
Cledualdo Soares de Oliveira et al.
MOLECULES (2012)
Chemical genetics
Cornelius J. O' Connor et al.
CHEMICAL SOCIETY REVIEWS (2011)
Diversity-oriented synthesis as a tool for the discovery of novel biologically active small molecules
Warren R. J. D. Galloway et al.
NATURE COMMUNICATIONS (2010)
The design of potent and selective inhibitors of DPP-4: Optimization of ADME properties by amide replacements
Sonja Nordhoff et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2009)
Emerging Treatments in Cystic Fibrosis
Andrew M. Jones et al.
DRUGS (2009)
Oxadiazolylindazole Sodium Channel Modulators are Neuroprotective toward Hippocampal Neurones
Lisa A. Clutterbuck et al.
JOURNAL OF MEDICINAL CHEMISTRY (2009)
The preparation of optically active α-amino 4H-[1,2,4]oxadiazol-5-ones from optically active α-amino acids
John E. Mangette et al.
TETRAHEDRON (2009)
Structures of PD-1 with its ligands: Sideways and dancing cheek to cheek
Gordon J. Freeman
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2008)
Discovery of potent 3,5-diphenyl-1,2,4-oxadiazole sphingosine-1-phosphate-1 (S1P1) receptor agonists with exceptional selectivity against S1P2 and S1P3
Z Li et al.
JOURNAL OF MEDICINAL CHEMISTRY (2005)
A facile and efficient one-pot synthesis of nitriles from carboxylic acids
K Mlinaric-Majerski et al.
SYNLETT (2005)
Discovery and structure-activity relationship of 3-aryl-5-aryl-1,2,4-oxadiazoles as a new series of apoptosis inducers and potential anticancer agents
HZ Zhang et al.
JOURNAL OF MEDICINAL CHEMISTRY (2005)
Novel semicarbazide-derived inhibitors of human dipeptidyl peptidase I (hDPPI)
J Bondebjerg et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2005)
Design and synthesis of new 2-substituted-5-(2-benzylthiophenyl)1,3,4-oxadiazoles as benzodiazepine receptor agonists
A Zarghi et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2005)
Synthesis and anticonvulsant activity of new 2-substituted-5-(2-benzyloxyphenyl)-1,3,4-oxadiazoles
A Zarghi et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2005)
O-alkoxyamidine prodrugs of furamidine:: In vitro transport and microsomal metabolism as indicators of in vivo efficacy in a mouse model of Trypanosoma brucei rhodesiense infection
JH Ansede et al.
JOURNAL OF MEDICINAL CHEMISTRY (2004)
Synthesis of New 1,2,4-oxadiazoles carrying (1'S,2'S)-t-butyloxycarbonyl-1-amino-2methyl-1-butyl and (1'S)-t-butyloxycarbonyl-1'-amino-1'-ethyl groups at C-5
VML Braga et al.
JOURNAL OF THE BRAZILIAN CHEMICAL SOCIETY (2004)
Parallel synthesis of 1,2,4-oxadiazoles from carboxylic acids using an improved, uronium-based, activation
RF Poulain et al.
TETRAHEDRON LETTERS (2001)
Apoptotic cell death in mammary adenocarcinoma cells is prevented by soluble factors present in the target organ of metastasis
V Ladeda et al.
BREAST CANCER RESEARCH AND TREATMENT (2001)
分享论文
