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Naturally occurring polyphenolic inhibitors of amyloid beta aggregation
Quentin I. Churches et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2014)
Aurones as histone deacetylase inhibitors: Identification of key features
Vincent Zwick et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2014)
Investigation of Binding-Site Homology between Mushroom and Bacterial Tyrosinases by Using Aurones as Effectors
Romain Haudecoeur et al.
CHEMBIOCHEM (2014)
Stereoselective synthesis of epsilon-lactones or spiro-heterocycles through NHC-catalyzed annulation: divergent reactivity by catalyst control
Min Wang et al.
CHEMICAL COMMUNICATIONS (2014)
Flavonoids from Garcinia paucinervis and their Biological Activities
Qiufen Hu et al.
CHEMISTRY OF NATURAL COMPOUNDS (2014)
Making Fast Photoswitches Faster-Using Hammett Analysis to Understand the Limit of Donor-Acceptor Approaches for Faster Hemithioindigo Photoswitches
Benjamin Maerz et al.
CHEMISTRY-A EUROPEAN JOURNAL (2014)
Recent developments in tubulin polymerization inhibitors: An overview
Ramandeep Kaur et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2014)
Probing the aurone scaffold against Plasmodium falciparum: Design, synthesis and antimalarial activity
Marta P. Carrasco et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2014)
Design, synthesis and structure-activity relationship of novel semi-synthetic flavonoids as antiproliferative agents
F. A. Ragab et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2014)
Discovery of indanone derivatives as multi-target-directed ligands against Alzheimer's disease
Ling Huang et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2014)
B-ring modified aurones as promising allosteric inhibitors of hepatitis C virus RNA-dependent RNA polymerase
Amel Meguellati et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2014)
Biological Activity and Molecular Docking Studies of Curcumin-Related α,β-Unsaturated Carbonyl-Based Synthetic Compounds as Anticancer Agents and Mushroom Tyrosinase Inhibitors
Syed Nasir Abbas Bukhari et al.
JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY (2014)
Identification of specific reversal agents for Leishmania ABCI4-mediated antimony resistance by flavonoid and trolox derivative screening
Jose Ignacio Manzano et al.
JOURNAL OF ANTIMICROBIAL CHEMOTHERAPY (2014)
Discovery of Entamoeba histolytica hexokinase 1 inhibitors through homology modeling and virtual screening
Maria Leticia Saucedo-Mendiola et al.
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (2014)
Discovery and Structure-Activity Relationship of Novel 2,3-Dihydrobenzofuran-7-carboxamide and 2,3-Dihydrobenzofuran-3(2H)-one-7-carboxamide Derivatives as Poly(ADP-ribose)polymerase-1 Inhibitors
Maulik R. Patel et al.
JOURNAL OF MEDICINAL CHEMISTRY (2014)
Photopharmacology: Beyond Proof of Principle
Willem A. Velema et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2014)
Sulfuretin inhibits 6-hydroxydopamine-induced neuronal cell death via reactive oxygen species-dependent mechanisms in human neuroblastoma SH-SY5Y cells
Seung-Hwan Kwon et al.
NEUROCHEMISTRY INTERNATIONAL (2014)
Pharmacophore and QSAR modeling of some structurally diverse azaaurones derivatives as anti-malarial activity
Mukesh C. Sharma et al.
MEDICINAL CHEMISTRY RESEARCH (2014)
Schistosomicidal and Antioxidant Flavonoids from Astragalus englerianus
Chao-Jiang Xiao et al.
PLANTA MEDICA (2014)
Synthesis of Some New 3-Coumaranone and Coumarin Derivatives as Dual Inhibitors of Acetyl- and Butyrylcholinesterase
Masoumeh Alipour et al.
ARCHIV DER PHARMAZIE (2013)
Potential neuroprotective flavonoid-based inhibitors of CDK5/p25 from Rhus parviflora
Sabina Shrestha et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2013)
Adamantyl Arotinoids That Inhibit IB Kinase and IB Kinase
Paula Lorenzo et al.
CHEMMEDCHEM (2013)
Flavonoids from the fruits of Nepalese sumac (Rhus parviflora) attenuate glutamate-induced neurotoxicity in HT22 cells
Sabina Shrestha et al.
FOOD SCIENCE AND BIOTECHNOLOGY (2013)
AURONES AND ISOAURONES FROM THE FLOWERS OF ROSA DAMASCENA AND THEIR BIOLOGICAL ACTIVITIES
Xue-Mei Gao et al.
HETEROCYCLES (2013)
Synthesis, docking studies and antioxidant activity of some chalcone and aurone derivatives
Tamanna Narsinghani et al.
MEDICINAL CHEMISTRY RESEARCH (2013)
5,6-Dimethoxybenzofuran-3-one derivatives: a novel series of dual Acetylcholinesterase/Butyrylcholinesterase inhibitors bearing benzyl pyridinium moiety
Hamid Nadri et al.
DARU-JOURNAL OF PHARMACEUTICAL SCIENCES (2013)
Influence of the skeleton on the cytotoxicity of flavonoids
Guy Lewin et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2012)
Synthesis and anticancer activity of 2-benzylidene indanones through inhibiting tubulin polymerization
A. P. Prakasham et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2012)
Synthesis and biological evaluation of novel oxindole derivatives for imaging neurofibrillary tangles in Alzheimer's disease
Hiroyuki Watanabe et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2012)
Structure-based virtual screening approach to the discovery of novel PTPMT1 phosphatase inhibitors
Hwangseo Park et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2012)
A scaffold hopping approach to identify novel monoamine oxidase B inhibitors
Werner J. Geldenhuys et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2012)
Design, synthesis, and evaluation of indanone derivatives as acetylcholinesterase inhibitors and metal-chelating agents
Fan-Chao Meng et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2012)
Ethylenediamine diacetate (EDDA) mediated synthesis of aurones under ultrasound: Their evaluation as inhibitors of SIRT1
Khanapur Manjulatha et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2012)
Versatile Effects of Aurone Structure on Mushroom Tyrosinase Activity
Carole Dubois et al.
CHEMBIOCHEM (2012)
Novel Indanone Derivatives as Potential Imaging Probes for ß-Amyloid Plaques in the Brain
Jin-Ping Qiao et al.
CHEMBIOCHEM (2012)
Recent Advances in the Medicinal Chemistry of Aurones
R. Haudecoeur et al.
CURRENT MEDICINAL CHEMISTRY (2012)
In vitro inhibitory properties of ferrocene-substituted chalcones and aurones on bacterial and human cell cultures
Keshri Nath Tiwari et al.
DALTON TRANSACTIONS (2012)
Synthesis of 1-Indanones from Benzoic Acids
Yun-Sheng Huang et al.
INDUSTRIAL & ENGINEERING CHEMISTRY RESEARCH (2012)
Rational Evolution of a Novel Type of Potent and Selective Proviral Integration Site in Moloney Murine Leukemia Virus Kinase 1 (PIM1) Inhibitor from a Screening-Hit Compound
Hirofumi Nakano et al.
JOURNAL OF MEDICINAL CHEMISTRY (2012)
Multitarget-Directed Benzylideneindanone Derivatives: Anti-β-Amyloid (Aβ) Aggregation, Antioxidant, Metal Chelation, and Monoamine Oxidase B (MAO-B) Inhibition Properties against Alzheimer's Disease
Ling Huang et al.
JOURNAL OF MEDICINAL CHEMISTRY (2012)
Antiviral Activities of Flavonoids Isolated from the Bark of Rhus verniciflua Stokes against Fish Pathogenic Viruses In Vitro
So Young Kang et al.
JOURNAL OF MICROBIOLOGY (2012)
A Novel Pim-1 Kinase Inhibitor Targeting Residues That Bind the Substrate Peptide
Keiko Tsuganezawa et al.
JOURNAL OF MOLECULAR BIOLOGY (2012)
Light-Switchable Hemithioindigo-Hemistilbene-Containing Peptides: Ultrafast Spectroscopy of the Z → E Isomerization of the Chromophore and the Structural Dynamics of the Peptide Moiety
N. Regner et al.
JOURNAL OF PHYSICAL CHEMISTRY B (2012)
Sulfuretin, a major flavonoid isolated from Rhus verniciflua, ameliorates experimental arthritis in mice
Young-Rae Lee et al.
LIFE SCIENCES (2012)
High throughput screening of a library based on kinase inhibitor scaffolds against Mycobacterium tuberculosis H37Rv
Robert C. Reynolds et al.
TUBERCULOSIS (2012)
Aurones: A Promising Heterocyclic Scaffold for the Development of Potent Antileishmanial Agents
Marina Roussaki et al.
INTERNATIONAL JOURNAL OF MEDICINAL CHEMISTRY (2012)
Aurones: Small Molecule Visible Range Fluorescent Probes Suitable for Biomacromolecules
Natasha Shanker et al.
JOURNAL OF FLUORESCENCE (2011)
Discovery of Naturally Occurring Aurones That Are Potent Allosteric Inhibitors of Hepatitis C Virus RNA-Dependent RNA Polymerase
Romain Haudecoeur et al.
JOURNAL OF MEDICINAL CHEMISTRY (2011)
Functionalized aurones as inducers of NAD(P)H:quinone oxidoreductase 1 that activate AhR/XRE and Nrf2/ARE signaling pathways: Synthesis, evaluation and SAR
Chong-Yew Lee et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2010)
Divergent Approach to Flavones and Aurones via Dihaloacrylic Acids. Unexpected Dependence on the Halogen Atom
George A. Kraus et al.
ORGANIC LETTERS (2010)
Design, synthesis and AChE inhibitory activity of indanone and aurone derivatives
Rong Sheng et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2009)
Molecular Mechanism of the Z/E-Photoisomerization of Hemithioindigo Hemistilbene
J. Ploetner et al.
JOURNAL OF PHYSICAL CHEMISTRY A (2009)
Versatile and expeditious synthesis of aurones via AuI-catalyzed cyclization
Hassina Harkat et al.
JOURNAL OF ORGANIC CHEMISTRY (2008)
Chemistry and folding of photomodulable peptides - stilbene and thioaurone-type candidates for conformational switches
Mate Erdelyi et al.
ORGANIC & BIOMOLECULAR CHEMISTRY (2008)
RAR and RXR modulation in cancer and metabolic disease
Lucia Altucci et al.
NATURE REVIEWS DRUG DISCOVERY (2007)
An antagonist of dishevelled protein-protein interaction suppresses β-catenin-dependent tumor cell growth
Naoaki Fujii et al.
CANCER RESEARCH (2007)
Hemithioindigo-based photoswitches as ultrafast light trigger in chromopeptides
T. Cordes et al.
CHEMICAL PHYSICS LETTERS (2006)
Photoactivation of an inhibitor of the 12/15-lipoxygenase pathway
Stephan Herre et al.
CHEMBIOCHEM (2006)
Discovery of benzylidenebenzofuran-3(2H)-one (aurones) as inhibitors of tyrosinase derived from human melanocytes
S Okombi et al.
JOURNAL OF MEDICINAL CHEMISTRY (2006)
Synthesis of 1-indanones by intramolecular Friedel-Crafts reaction of 3-arylpropionic acids catalyzed by Tb(OTf)3
DM Cui et al.
TETRAHEDRON LETTERS (2004)
Indanocine, a microtubule-binding indanone and a selective inducer of apoptosis in multidrug-resistant cancer cells
LM Leoni et al.
JNCI-JOURNAL OF THE NATIONAL CANCER INSTITUTE (2000)
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