4.4 Article

A Facile One-Pot Solvent-Free Synthesis, in Vitro and in Silico Studies of a Series of Tetrahydropyridine Derivatives as Breast Cancer Inhibitors

相关参考文献

注意:仅列出部分参考文献,下载原文获取全部文献信息。
Article Biochemistry & Molecular Biology

Design, synthesis and molecular docking studies of some 1-(5-(2-fluoro-5-(trifluoromethoxy)phenyl)-1,2,4-oxadiazol-3-yl)piperazine derivatives as potential anti-inflammatory agents

B. Kulkarni et al.

Summary: A series of 3,5-substituted-1,2,4-oxadiazole derivatives were synthesized in good to excellent yields, showing promising anti-inflammatory potential compared to the standard drug diclofenac sodium. Molecular docking and SAR studies were conducted to gain further insights into the activity profile of the synthesized molecules.

MOLECULAR DIVERSITY (2022)

Article Chemistry, Physical

Synthesis, stereochemical, single crystal X-ray structural and antimicrobial studies of some isobutyl-1,2,6-triaryl-4-(arylamino)-1,2,5,6-tetrahydropyridine-3-carboxylates: Exploring RAHB with S(6) graph set

Poyyamozhi Surendar Anand et al.

Summary: A new set of compounds with intra-molecular hydrogen bonding has been synthesized and analyzed, with a focus on Resonance Assisted Hydrogen Bonding (RAHB). The structures of the compounds were determined using analytical and spectral data, with confirmation from single crystal X-ray diffraction analysis. The study also includes antimicrobial testing against various bacterial and fungal strains, with results summarized.

JOURNAL OF MOLECULAR STRUCTURE (2021)

Article Tropical Medicine

Leishmaniasis en Bolivia, revisión y estado actual en Tarija, frontera con Argentina

Juan Sergio Mollinedo et al.

Biomedica (2020)

Article Chemistry, Medicinal

4-Aryl-1,4-Dihydropyridines as Potential Enoyl-Acyl Carrier Protein Reductase Inhibitors: Antitubercular Activity and Molecular Docking Study

Katharigatta N. Venugopala et al.

CURRENT TOPICS IN MEDICINAL CHEMISTRY (2020)

Article Biochemistry & Molecular Biology

Synthesis and characterization of a novel series of 1,4-dihydropyridine analogues for larvicidal activity against Anopheles arabiensis

Bhaskara D. Dharma Rao et al.

CHEMICAL BIOLOGY & DRUG DESIGN (2017)

Article

Antimicrobial and antioxidant activities of piperidine derivatives

Naicker Leeantha et al.

African Journal of Pharmacy and Pharmacology (2016)

Article Chemistry, Multidisciplinary

Multicomponent synthesis and antimicrobial activity of alkyl 4-arylamino-1,2,6-triaryl-1,2,5,6-tetrahydropyridine-3-carboxylates

A. N. Yankin et al.

RUSSIAN JOURNAL OF GENERAL CHEMISTRY (2015)

Article Chemistry, Multidisciplinary

Crystal structure refinement with SHELXL

George M. Sheldrick

ACTA CRYSTALLOGRAPHICA SECTION C-STRUCTURAL CHEMISTRY (2015)

Review Pharmacology & Pharmacy

Advances in Drug Development for Parkinson's Disease: Present Status

Dibbanti Harikrishna Reddy et al.

PHARMACOLOGY (2014)

Article Chemistry, Organic

La(NO3)3.6H2O Catalyzed One-pot Highly Diastereoselective Synthesis of Functionalized Piperidines

Mir Rasul Mousavi et al.

LETTERS IN ORGANIC CHEMISTRY (2013)

Article Crystallography

Methyl 2,6-diphenyl-1-p-tolyl-4-(p-tolylamino)-1,2,5,6-tetrahydropyridine-3-carboxylate

K. N. Venugopala et al.

ACTA CRYSTALLOGRAPHICA SECTION E-STRUCTURE REPORTS ONLINE (2012)

Article Chemistry, Multidisciplinary

Nickel (II) chloride hexahydrate as an efficient catalyst for the preparation of highly functionalised piperidine derivatives

Mohammad Reza Mohammad Shafiee et al.

JOURNAL OF CHEMICAL RESEARCH (2012)

Article Chemistry, Organic

Iodine-Catalyzed, Efficient, One-Pot Protocol for the Conversion of Araldehydes into 5-Aryl-1H-tetrazoles

M. B. Madhusudana Reddy et al.

SYNTHETIC COMMUNICATIONS (2011)

Review Chemistry, Analytical

Analysis of anticancer drugs: A review

Susanne Nussbaumer et al.

TALANTA (2011)

Article Chemistry, Medicinal

Synthesis, antimicrobial evaluation and QSAR studies of novel piperidin-4-yl-5-spiro-thiadiazoline derivatives

Seeman Umamatheswari et al.

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2010)

Article Biochemistry & Molecular Biology

Organocatalyzed highly atom economic one pot synthesis of tetrahydropyridines as antimalarials

Mridul Misra et al.

BIOORGANIC & MEDICINAL CHEMISTRY (2009)

Article Chemistry, Medicinal

Benzophenone-N-ethyl piperidine ether analogues-Synthesis and efficacy as anti-inflammatory agent

Shaukath A. Khanum et al.

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2009)

Article Chemistry, Medicinal

First stereoselective total synthesis and anticancer activity of new amide alkaloids of roots of pepper

Ch. Srinivas et al.

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2009)

Article Biochemical Research Methods

Molecular modeling of ligand-receptor interactions in GABAC receptor

Dmitry I. Osolodkin et al.

JOURNAL OF MOLECULAR GRAPHICS & MODELLING (2009)

Article Biochemistry & Molecular Biology

Antimycobacterial and H1-antihistaminic activity of 2-substituted piperidine derivatives

Robert Weis et al.

BIOORGANIC & MEDICINAL CHEMISTRY (2008)

Article Chemistry, Medicinal

Synthesis and antibacterial activity of novel fluoroquinolones containing substituted piperidines

Zhao Dang et al.

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2007)

Article Biochemistry & Molecular Biology

CCR5 antagonists as anti-HIV-1 agents. Part 3: Synthesis and biological evaluation of piperidine-4-carboxamide derivatives

S Imamura et al.

BIOORGANIC & MEDICINAL CHEMISTRY (2005)

Article Biochemistry & Molecular Biology

Dihydropyridine neuropeptide YY1 receptor antagonists 2:: bioisosteric urea replacements

GS Poindexter et al.

BIOORGANIC & MEDICINAL CHEMISTRY (2004)

Review Pharmacology & Pharmacy

Dietary agents in cancer prevention: flavonoids and isoflavonoids

DF Birt et al.

PHARMACOLOGY & THERAPEUTICS (2001)