相关参考文献
注意:仅列出部分参考文献,下载原文获取全部文献信息。Photochemical Fluorination Reactions - A Promising Research Field for Continuous-Flow Synthesis
Thomas H. Rehm
CHEMICAL ENGINEERING & TECHNOLOGY (2016)
A Fluorination/Aryl Migration/Cyclization Cascade for the Metal-Free Synthesis of Fluoro-Benzoxazepines
Anna Ulmer et al.
CHEMISTRY-A EUROPEAN JOURNAL (2016)
Small-Molecule Therapeutics for Ebola Virus (EBOV) Disease Treatment
Kunisuke Izawa et al.
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY (2016)
Fluorinated betulinic acid derivatives and evaluation of their anti-HIV activity
Jizhen Li et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2016)
Catalytic C-F bond activation of geminal difluorocyclopropanes by nickel(I) complexes via a radical mechanism
Jan Wenz et al.
CHEMICAL COMMUNICATIONS (2016)
Next Generation of Fluorine-Containing Pharmaceuticals, Compounds Currently in Phase II-III Clinical Trials of Major Pharmaceutical Companies: New Structural Trends and Therapeutic Areas
Yu Zhou et al.
CHEMICAL REVIEWS (2016)
18F-Labeling of Arenes and Heteroarenes for Applications in Positron Emission Tomography
Sean Preshlock et al.
CHEMICAL REVIEWS (2016)
[18F]-Group 13 fluoride derivatives as radiotracers for positron emission tomography
Kantapat Chansaenpak et al.
CHEMICAL SOCIETY REVIEWS (2016)
The medicinal chemist's toolbox for late stage functionalization of drug-like molecules
Tim Cernak et al.
CHEMICAL SOCIETY REVIEWS (2016)
Mono- and Difluorination of Benzylic Carbon Atoms
Ana Koperniku et al.
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY (2016)
Methyl NFSI: atom-economical alternative to NFSI shows higher fluorination reactivity under Lewis acid-catalysis and non-catalysis
Kazunobu Fukushi et al.
GREEN CHEMISTRY (2016)
Sustainable synthesis of enantiopure fluorolactam derivatives by a selective direct fluorination - amidase strategy
Nicky J. Willis et al.
GREEN CHEMISTRY (2016)
Regioselective Electrophilic Fluorination of Rationally Designed Imidazole Derivatives
Klaus Albertshofer et al.
JOURNAL OF ORGANIC CHEMISTRY (2016)
Enantioselective aldol reactions with masked fluoroacetates
Jakub Saadi et al.
NATURE CHEMISTRY (2016)
The total synthesis of calcium atorvastatin
Luiz C. Dias et al.
ORGANIC & BIOMOLECULAR CHEMISTRY (2016)
Pd(II)-Catalyzed Aminofluorination of Alkenes in Total Synthesis 6-(R)-Fluoroswainsonine and 5-(R)-Fluorofebrifugine
Liang Wu et al.
ORGANIC LETTERS (2016)
Diastereoselective Synthesis and Conformational Analysis of (2R)- and (2S)-Fluorostatines: An Approach Based on Organocatalytic Fluorination of a Chiral Aldehyde
Xiang-Guo Hu et al.
ORGANIC LETTERS (2016)
Aminofluorination: transition-metal-free N-F bond insertion into diazocarbonyl compounds
Gui Chen et al.
CHEMICAL SCIENCE (2016)
Asymmetric 18F-fluorination for applications in positron emission tomography
Faye Buckingham et al.
CHEMICAL SCIENCE (2016)
Fluorine-18 patents (2009-2015). Part 1: novel radiotracers
Allen F. Brooks et al.
PHARMACEUTICAL PATENT ANALYST (2016)
Organomediated Enantioselective 18FFluorination for PET Applications
Faye Buckingham et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2015)
18F-Labeling of Aryl-SCF3, -OCF3 and -OCHF2 with [18F]Fluoride
Tanatorn Khotavivattana et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2015)
Triazole: A Promising Antitubercular Agent
Rangappa S. Keri et al.
CHEMICAL BIOLOGY & DRUG DESIGN (2015)
Direct photocatalytic fluorination of benzylic C-H bonds with N-fluorobenzenesulfonimide
Matthew B. Nodwell et al.
CHEMICAL COMMUNICATIONS (2015)
Introduction: Fluorine Chemistry
Veronique Gouverneur et al.
CHEMICAL REVIEWS (2015)
Monofluorination of Organic Compounds: 10 Years of Innovation
Pier Alexandre Champagne et al.
CHEMICAL REVIEWS (2015)
Organocatalytic Asymmetric Fluorination of 4-Substituted Isoxazolinones
Huanrui Zhang et al.
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY (2015)
Advancements in Aminofluorination of Alkenes and Alkynes: Convenient Access to β-Fluoroamines
Pinhong Chen et al.
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY (2015)
Synthesis of 5-Fluorotriazoles by Silver-Mediated Fluorination of 5-Iodotriazoles
Damin Wang et al.
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY (2015)
Organofluorine chemistry: applications, sources and sustainability
Antal Harsanyi et al.
GREEN CHEMISTRY (2015)
Synthesis of fluorinated oxygen- and sulfur-containing heteroaromatics
Eileen M. O'Leary et al.
JOURNAL OF FLUORINE CHEMISTRY (2015)
Oxidative fluorination of N-arylsulfonamides
Faye Buckingham et al.
JOURNAL OF FLUORINE CHEMISTRY (2015)
Fluorination Patterning: A Study of Structural Motifs That Impact Physicochemical Properties of Relevance to Drug Discovery
Quentin A. Huchet et al.
JOURNAL OF MEDICINAL CHEMISTRY (2015)
Applications of Fluorine in Medicinal Chemistry
Eric P. Gillis et al.
JOURNAL OF MEDICINAL CHEMISTRY (2015)
Investigation and Conformational Analysis of Fluorinated Nucleoside Antibiotics Targeting Siderophore Biosynthesis
Surendra Dawadi et al.
JOURNAL OF ORGANIC CHEMISTRY (2015)
Transition-Metal-Free Oxyfluorination of Olefinic Amides for the Synthesis of Fluorinated Heterocycles
Jing-Feng Zhao et al.
JOURNAL OF ORGANIC CHEMISTRY (2015)
Anhydrous Tetramethylammonium Fluoride for Room-Temperature SNAr Fluorination
Sydonie D. Schimler et al.
JOURNAL OF ORGANIC CHEMISTRY (2015)
Regioselective Fluorination of Imidazo[1,2-a]pyridines with Selectfluor in Aqueous Condition
Ping Liu et al.
JOURNAL OF ORGANIC CHEMISTRY (2015)
A Fluorinated Ligand Enables Room-Temperature and Regioselective Pd-Catalyzed Fluorination of Aryl Triflates and Bromides
Aaron C. Sather et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2015)
PyFluor: A Low-Cost, Stable, and Selective Deoxyfluorination Reagent
Matthew K. Nielsen et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2015)
Fluorination of 2-substituted benzo[b]furans with Selectfluor™
Mingliang Wang et al.
ORGANIC & BIOMOLECULAR CHEMISTRY (2015)
Efficient Palladium-Catalyzed C-H Fluorination of C(sp3)-H Bonds: Synthesis of β-Fluorinated Carboxylic Acids
Qihua Zhu et al.
ORGANIC LETTERS (2015)
Development of a Direct Photocatalytic C-H Fluorination for the Preparative Synthesis of Odanacatib
Shira D. Halperin et al.
ORGANIC LETTERS (2015)
Asymmetric Fluorination Approach to the Scalable Synthesis of a SYK Inhibitor
Neil R. Curtis et al.
ORGANIC PROCESS RESEARCH & DEVELOPMENT (2015)
Selective C-H Bond Fluorination of Phenols with a Removable Directing Group: Late-Stage Fluorination of 2-Phenoxyl Nicotinate Derivatives
Shao-Jie Lou et al.
ACS CATALYSIS (2015)
Transition-metal free oxidative aliphatic C-H fluorination
Xiaofei Zhang et al.
Organic Chemistry Frontiers (2015)
Modern Carbon-Fluorine Bond Forming Reactions for Aryl Fluoride Synthesis
Michael G. Campbell et al.
CHEMICAL REVIEWS (2015)
Advances in Catalytic Enantioselective Fluorination, Mono-, Di-, and Trifluoromethylation, and Trifluoromethylthiolation Reactions
Xiaoyu Yang et al.
CHEMICAL REVIEWS (2015)
Preparation of iodonium ylides: probing the fluorination of 1,3-dicarbonyl compounds with a fluoroiodane
Gemma C. Geary et al.
RSC ADVANCES (2015)
Asymmetric Fluorocyclizations of Alkenes
Jamie R. Wolstenhulme et al.
ACCOUNTS OF CHEMICAL RESEARCH (2014)
Inside Cover: Thiophene-Based, Radial π-Conjugation: Synthesis, Structure, and Photophysical Properties of Cyclo-1,4-phenylene-2′,5′-thienylenes (Angew. Chem. Int. Ed. 1/2015)
Hideto Ito et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2014)
A General Copper-Mediated Nucleophilic 18F Fluorination of Arenes
Matthew Tredwell et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2014)
The synthesis of gemcitabine
Kylie Brown et al.
CARBOHYDRATE RESEARCH (2014)
Silver-catalyzed one-pot cyclization/fluorination of 2-alkynylanilines: highly efficient synthesis of structurally diverse fluorinated indole derivatives
Lei Yang et al.
CHEMICAL COMMUNICATIONS (2014)
Fluorine in Pharmaceutical Industry: Fluorine-Containing Drugs Introduced to the Market in the Last Decade (2001-2011)
Jiang Wang et al.
CHEMICAL REVIEWS (2014)
Divergent Reaction Mechanisms in the Aminofluorination of Alkenes
Wangqing Kong et al.
CHIMIA (2014)
Palladium-Catalyzed Oxidative Olefination of Phenols Bearing Removable Directing Groups under Molecular Oxygen
Bin Liu et al.
JOURNAL OF ORGANIC CHEMISTRY (2014)
Direct C-F Bond Formation Using Photoredox Catalysis
Montserrat Rueda-Becerril et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2014)
How Cinchona Alkaloid-Derived Primary Amines Control Asymmetric Electrophilic Fluorination of Cyclic Ketones
Yu-hong Lam et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2014)
A General and Enantioselective Approach to Pentoses: A Rapid Synthesis of PSI-6130, the Nucleoside Core of Sofosbuvir
Manuel Peifer et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2014)
Double Annulative Cascade of Tryptophan-Containing Peptides Triggered by Selectfluor
Bret Treguier et al.
ORGANIC LETTERS (2014)
Metal-Free, Efficient Oxyfluorination of Olefins for the Synthesis of α-Fluoroketones
Qiang Yang et al.
ORGANIC LETTERS (2014)
Late-Stage Fluorination: From Fundamentals to Application
Michael G. Campbell et al.
ORGANIC PROCESS RESEARCH & DEVELOPMENT (2014)
PhenoFluor: Practical Synthesis, New Formulation, and Deoxyfluorination of Heteroaromatics
Teppei Fujimoto et al.
ORGANIC PROCESS RESEARCH & DEVELOPMENT (2014)
Discovery of a Novel Class of Imidazo[1,2-a]Pyridines with Potent PDGFR Activity and Oral Bioavailability
Erik J. Hicken et al.
ACS MEDICINAL CHEMISTRY LETTERS (2014)
On the role of fluoro-substituted nucleosides in DNA radiosensitization for tumor radiation therapy
J. Kopyra et al.
RSC ADVANCES (2014)
Palladium-Catalyzed Decarboxylative Coupling of α- Oxocarboxylic Acids with C(sp2)-H of 2-Aryloxypyridines
Jinzhong Yao et al.
ADVANCED SYNTHESIS & CATALYSIS (2013)
Stereoselectively fluorinated N-heterocycles: a brief survey
Xiang-Guo Hu et al.
BEILSTEIN JOURNAL OF ORGANIC CHEMISTRY (2013)
Electrophilic fluorination using a hypervalent iodine reagent derived from fluoride
Gemma C. Geary et al.
CHEMICAL COMMUNICATIONS (2013)
Ruthenium(II)-Catalyzed C-H Alkenylations of Phenols with Removable Directing Groups
Wenbo Ma et al.
CHEMISTRY-A EUROPEAN JOURNAL (2013)
A Two-Step Sequence to Ethyl α-Fluorocyclopropanecarboxylates Through MIRC Reaction of Ethyl Dichloroacetate and Highly Regioselective Fluorination
Min Zhang et al.
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY (2013)
5-alkyl-1,3-oxazole derivatives of 6-amino-nicotinic acids as alkyl ester bioisosteres are antagonists of the P2Y12 receptor
Peter Bach et al.
FUTURE MEDICINAL CHEMISTRY (2013)
Non-Nucleoside Inhibitors of BasE, an Adenylating Enzyme in the Siderophore Biosynthetic Pathway of the Opportunistic Pathogen Acinetobacter baumannii
Joao Neres et al.
JOURNAL OF MEDICINAL CHEMISTRY (2013)
Enantioselective Synthesis of cis-3-Fluoropiperidin-4-ol, a Building Block for Medicinal Chemistry
Simon J. Shaw et al.
JOURNAL OF ORGANIC CHEMISTRY (2013)
Late-Stage Deoxyfluorination of Alcohols with PhenoFluor
Filippo Sladojevich et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2013)
Mild Copper-Mediated Fluorination of Aryl Stannanes and Aryl Trifluoroborates
Yingda Ye et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2013)
Silver-Catalyzed Radical Phosphonofluorination of Unactivated Alkenes
Chengwei Zhang et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2013)
Copper-Mediated Fluorination of Arylboronate Esters. Identification of a Copper(III) Fluoride Complex
Patrick S. Fier et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2013)
Oxidative aliphatic C-H fluorination with manganese catalysts and fluoride ion
Wei Liu et al.
NATURE PROTOCOLS (2013)
One-Pot Gold-Catalyzed Aminofluorination of Unprotected 2-Alkynylanilines
Antonio Arcadi et al.
ORGANIC LETTERS (2013)
Selective C-H Fluorination of Pyridines and Diazines Inspired by a Classic Amination Reaction
Patrick S. Fier et al.
SCIENCE (2013)
Cover Picture: Champagne and Fireworks:Angewandte ChemieCelebrates Its Birthday (Angew. Chem. Int. Ed. 1/2013)
Peter Gölitz
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2012)
Synthesis, evaluation of anti-HIV-1 and anti-HCV activity of novel 2′,3′-dideoxy-2′,2′-difluoro-4′-azanucleosides
Saul Martinez-Montero et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2012)
Transition metal catalysis and nucleophilic fluorination
Charlotte Hollingworth et al.
CHEMICAL COMMUNICATIONS (2012)
Synthesis and biological evaluation of novel flavonols as potential anti-prostate cancer agents
Robert G. Britton et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2012)
Zolpidem for insomnia
David J. Greenblatt et al.
EXPERT OPINION ON PHARMACOTHERAPY (2012)
Synthesis and applications of fluorinated nucleoside analogues
Hanna Wojtowicz-Rajchel
JOURNAL OF FLUORINE CHEMISTRY (2012)
Fluorine Transfer to Alkyl Radicals
Montserrat Rueda-Becerril et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2012)
Fe(III)/NaBH4-Mediated Free Radical Hydrofluorination of Unactivated Alkenes
Timothy J. Barker et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2012)
Copper-Mediated Fluorination of Aryl Iodides
Patrick S. Fier et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2012)
Silver-Catalyzed Decarboxylative Fluorination of Aliphatic Carboxylic Acids in Aqueous Solution
Feng Yin et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2012)
Ag(I)-Catalyzed Aminofluorination of Alkynes: Efficient Synthesis of 4-Fluoroisoquinolines and 4-Fluoropyrrolo[α]isoquinolines
Tao Xu et al.
ORGANIC LETTERS (2012)
Metal-Free Ortho C-H Borylation of 2-Phenoxypyridines under Mild Conditions
Liting Niu et al.
ORGANIC LETTERS (2012)
Ruthenium-Catalyzed C-H Bond Arylations of Arenes Bearing Removable Directing Groups via Six-Membered Ruthenacycles
Lutz Ackermann et al.
ORGANIC LETTERS (2012)
Development of Two Complementary Syntheses for a Privileged CGRP Receptor Antagonist Substructure
David K. Leahy et al.
ORGANIC PROCESS RESEARCH & DEVELOPMENT (2012)
Oxidative Aliphatic C-H Fluorination with Fluoride Ion Catalyzed by a Manganese Porphyrin
Wei Liu et al.
SCIENCE (2012)
Synthesis and PET imaging studies of [18F]2-fluoroquinolin-8-ol ([18F]CABS13) in transgenic mouse models of Alzheimer's disease
Neil Vasdev et al.
MEDCHEMCOMM (2012)
Ir-catalysed formation of C-F bonds. From allylic alcohols to alpha-fluoroketones
Nanna Ahlsten et al.
CHEMICAL COMMUNICATIONS (2011)
Iminosugars as therapeutic agents: recent advances and promising trends
Robert J. Nash et al.
FUTURE MEDICINAL CHEMISTRY (2011)
Pseudomonas stutzeri lipase: a useful biocatalyst for aminolysis reactions
S. van Pelt et al.
GREEN CHEMISTRY (2011)
Deoxyfluorination of Phenols
Pingping Tang et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2011)
Enantioselective Organocatalytic α-Fluorination of Cyclic Ketones
Piotr Kwiatkowski et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2011)
The flow synthesis of heterocycles for natural product and medicinal chemistry applications
Marcus Baumann et al.
MOLECULAR DIVERSITY (2011)
Catalysis for fluorination and trifluoromethylation
Takeru Furuya et al.
NATURE (2011)
An Efficient Difluorohydroxylation of Indoles Using Selectfluor as a Fluorinating Reagent
Riyuan Lin et al.
ORGANIC LETTERS (2011)
A Fluoride-Derived Electrophilic Late-Stage Fluorination Reagent for PET Imaging
Eunsung Lee et al.
SCIENCE (2011)
Silver-mediated fluorination of aryl silanes
Pingping Tang et al.
TETRAHEDRON (2011)
The Organometallic Fluorine Chemistry of Palladium and Rhodium: Studies toward Aromatic Fluorination
Vladimir V. Grushin
ACCOUNTS OF CHEMICAL RESEARCH (2010)
Convenient Electrophilic Fluorination of Functionalized Aryl and Heteroaryl Magnesium Reagents
Shigeyuki Yamada et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2010)
Fluorine-Enabled Cationic Gold Catalysis: Functionalized Hydration of Alkynes
Weibo Wang et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2010)
Amplification of the Inhibitory Activity and Reversal of the Selectivity of Miglitol by C(2′)-Monofluorination
Erik Prell et al.
ARCHIV DER PHARMAZIE (2010)
Fluorine in health care Organofluorine containing blockbuster drugs
David O'Hagan
JOURNAL OF FLUORINE CHEMISTRY (2010)
Aminodifluorosulfinium Salts: Selective Fluorination Reagents with Enhanced Thermal Stability and Ease of Handling
Alexandre L'Heureux et al.
JOURNAL OF ORGANIC CHEMISTRY (2010)
Silver-Catalyzed Late-Stage Fluorination
Pingping Tang et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2010)
New Synthesis of Fluorinated Pyrazoles
Riccardo Surmont et al.
ORGANIC LETTERS (2010)
Palladium(II)-Catalyzed Ortho Arylation of 2-Phenoxypyridines with Potassium Aryltrifluoroborates via C-H Functionalization
Jean-Ho Chu et al.
ORGANOMETALLICS (2010)
Fluorine in medicinal chemistry: a century of progress and a 60-year retrospective of selected highlights
Robert Filler et al.
FUTURE MEDICINAL CHEMISTRY (2009)
Semisynthesis, Biological Activity, and Molecular Modeling Studies of C-Ring-Modified Camptothecins
Cristian Samori et al.
JOURNAL OF MEDICINAL CHEMISTRY (2009)
Silver-Mediated Fluorination of Functionalized Aryl Stannanes
Takeru Furuya et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2009)
Tankyrase inhibition stabilizes axin and antagonizes Wnt signalling
Shih-Min A. Huang et al.
NATURE (2009)
Palladium-Catalyzed Acylation of sp2 C-H bond: Direct Access to Ketones from Aldehydes
Xiaofei Jia et al.
ORGANIC LETTERS (2009)
Fluorination of Boronic Acids Mediated by Silver(I) Triflate
Takeru Furuya et al.
ORGANIC LETTERS (2009)
Formation of ArF from LPdAr(F): Catalytic Conversion of Aryl Triflates to Aryl Fluorides
Donald A. Watson et al.
SCIENCE (2009)
Nitrogen-Containing Organofluorine Derivatives: An Overview
Santos Fustero et al.
SYNLETT (2009)
Micellar-System-Mediated Direct Fluorination of Ketones in Water
Gaj Stavber et al.
SYNLETT (2009)
Microwave-assisted aliphatic fluorine-chlorine exchange using triethylamine trihydrofluoride (TREAT-HF)
Jennifer A. Kremsner et al.
TETRAHEDRON LETTERS (2009)
Palladium-mediated fluorination of arylboronic acids
Takeru Furuya et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2008)
Fluorine in medicinal chemistry
Sophie Purser et al.
CHEMICAL SOCIETY REVIEWS (2008)
The many roles for fluorine in medicinal chemistry
William K. Hagmann
JOURNAL OF MEDICINAL CHEMISTRY (2008)
Highly Regioselective Fluorination and Iodination of Alkynyl Enolates
Han Yang et al.
ORGANIC LETTERS (2008)
Fluorination in medicinal chemistry: Methods, strategies, and recent developments
Kenneth L. Kirk
ORGANIC PROCESS RESEARCH & DEVELOPMENT (2008)
Direct synthesis of 8-Fluoro purine Nucleosides via metalation-fluorination
Arun K. Ghosh et al.
JOURNAL OF ORGANIC CHEMISTRY (2007)
Fluorine in pharmaceuticals:: Looking beyond intuition
Klaus Mueller et al.
SCIENCE (2007)
Predicting properties and tuning physicochemical in lead optimization:: Amine basicities
Martin Morgenthaler et al.
CHEMMEDCHEM (2007)
New approaches to enantioselective fluorination: Cinchona alkaloids combinations and chiral ligands/metal complexes
Norio Shibata et al.
JOURNAL OF FLUORINE CHEMISTRY (2007)
Discovery and development of clofarabine: a nucleoside analogue for treating cancer
Peter L. Bonate et al.
NATURE REVIEWS DRUG DISCOVERY (2006)
Recent advances (1995-2005) in fluorinated pharmaceuticals based on natural products
Jean-Pierre Begue et al.
JOURNAL OF FLUORINE CHEMISTRY (2006)
Fluorine in medicinal chemistry: Recent therapeutic applications of fluorinated small molecules
Kenneth L. Kirk
JOURNAL OF FLUORINE CHEMISTRY (2006)
Palladium-catalyzed fluorination of carbon-hydrogen bonds
Kami L. Hull et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2006)
Efficacy of etifoxine compared to lorazepam monotherapy in the treatment of patients with adjustment disorders with anxiety: a double-blind controlled study in general practice
N Nguyen et al.
HUMAN PSYCHOPHARMACOLOGY-CLINICAL AND EXPERIMENTAL (2006)
Fluorine in medicinal chemistry: A review of anti-cancer agents
C Isanbor et al.
JOURNAL OF FLUORINE CHEMISTRY (2006)
Prostanoids in the therapy of glaucoma
Naruhiro Ishida et al.
CARDIOVASCULAR DRUG REVIEWS (2006)
The role of clofarabine in hematologic and solid mal ignancies - Development of a next-generation nucleoside analog
S Faderl et al.
CANCER (2005)
Tetrabutylammonium salt induced denitration of nitropyridines: Synthesis of fluoro-, hydroxy-, and methoxypyridines
SD Kuduk et al.
ORGANIC LETTERS (2005)
Modern synthetic methods for fluorine-substituted target molecules
M Shimizu et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2005)
Selectfluor: Mechanistic insight and applications
PT Nyffeler et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2005)
Synthesis of the highly potent prostanoid FP receptor agonist, AFP-168:: a novel 15-deoxy-15,15-difluoroprostaglandin F2α derivative
Y Matsumura et al.
TETRAHEDRON LETTERS (2004)
Synthesis, structure-activity relationships, and drug resistance of β-D-3′-fluoro-2′,3′-unsaturated nucleosides as anti-HIV agents
W Zhou et al.
JOURNAL OF MEDICINAL CHEMISTRY (2004)
The polar hydrophobicity of fluorinated compounds
JC Biffinger et al.
CHEMBIOCHEM (2004)
Fluorine in medicinal chemistry
HJ Böhm et al.
CHEMBIOCHEM (2004)
Recent highlights in electrophilic fluorination with 1-chloromethyl-4-fluoro-1,4-diazoniabicyclo[2.2.2]octane bis(tetrafluoroborate)
RP Singh et al.
ACCOUNTS OF CHEMICAL RESEARCH (2004)
L-2′,3′-Didehydro-2′,3′-dideoxy-3′-fluoronucleosides:: Synthesis, anti-HIV activity, chemical and enzymatic stability, and mechanism of resistance
Y Chong et al.
JOURNAL OF MEDICINAL CHEMISTRY (2003)
Effect of minodronic acid (ONO-5920) on bone mineral density and arthritis in adult rats with collagen-induced arthritis
I Yamane et al.
ARTHRITIS AND RHEUMATISM (2003)
Aspartic proteinases in disease: A structural perspective
JB Cooper
CURRENT DRUG TARGETS (2002)
Structure-activity relationships of 2′-fluoro-2′,3′-unsaturated D-nucleosides as anti-HIV-1 agents
K Lee et al.
JOURNAL OF MEDICINAL CHEMISTRY (2002)
A new chelation-assistance mode for a ruthenium-catalyzed silylation at the C-H bond in aromatic ring with hydrosilanes
F Kakiuchi et al.
CHEMISTRY LETTERS (2002)
Synthesis and biological evaluation of imidazol-2-one and 2-cyanoiminoimidazole derivatives:: Novel series of PDE4 inhibitors
JI Andrés et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2002)
2,2-difluoro-1,3-dimethylimidazolidine (DFI). A new fluorinating agent
H Hayashi et al.
CHEMICAL COMMUNICATIONS (2002)
Enantioselective fluorination mediated by cinchona alkaloid derivatives/selectfluor combinations:: Reaction scope and structural information for N-fluorocinchona alkaloids
N Shibata et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2001)
3-(4-fluoropiperidin-3-yl)-2-phenylindoles as high affinity, selective, and orally bioavailable h5-HT2A receptor antagonist
M Rowley et al.
JOURNAL OF MEDICINAL CHEMISTRY (2001)