4.5 Article

In vitro multitarget activity of sulfadiazine substituted triazenes as antimicrobial, cytotoxic, and larvicidal agents

相关参考文献

注意:仅列出部分参考文献,下载原文获取全部文献信息。
Review Chemistry, Medicinal

Natural Products as Sources of Multitarget Compounds: Advances in the Development of Ferulic Acid as Multitarget Therapeutic

Rajwinder Kaur et al.

Summary: Nature provides therapeutic substances, and many valuable medications are derived from plants. Multitarget drugs are essential in treating various disorders. Ferulic acid, with low toxicity and minimal side effects, shows potential therapeutic actions by modulating various signal transduction pathways.

CURRENT TOPICS IN MEDICINAL CHEMISTRY (2022)

Article Biotechnology & Applied Microbiology

Antifungal activity of 2-chloro-N-phenylacetamide, docking and molecular dynamics studies against clinical isolates of Candida tropicalis and Candida parapsilosis

Shellygton Lima Silva et al.

Summary: This study evaluated the antifungal and antibiofilm activity of 2-chloro-N-phenylacetamide against Candida tropicalis and Candida parapsilosis isolates. The results showed that A1Cl has fungicide activity and can attenuate the expression of virulence factors, inhibit biofilm formation, and reduce mature biofilm biomass.

JOURNAL OF APPLIED MICROBIOLOGY (2022)

Article Biotechnology & Applied Microbiology

Anti-microbial efficacy, mechanisms and druggability evaluation of the natural flavonoids

Hongyan Lin et al.

Summary: Glabridin from Glycyrrhiza glabra L. exhibited potent antibacterial activity against Staph. aureus by acting as a DNA gyrase inhibitor, representing a promising natural antimicrobial agent.

JOURNAL OF APPLIED MICROBIOLOGY (2022)

Article Chemistry, Multidisciplinary

Synthesis, Characterization, and Biological Evaluation of Novel Cyclohexenone Derivatives Incorporating Azo, Triazene, and Tetraazene Moieties

Ebrahim Abdel-Galil et al.

Summary: New cyclohexenone derivatives were synthesized and evaluated for their antioxidant and antimicrobial activities. Compounds 8 and 15 exhibited the highest antioxidant activity, while compound 10 showed potent antibacterial activity against Staphylococcus aureus and Escherichia coli. Compounds 10, 12, and 14 demonstrated the best activities against Candida albicans.

RUSSIAN JOURNAL OF GENERAL CHEMISTRY (2022)

Article Chemistry, Physical

Crystal structure, mosquito larvicidal & antifungal activity of 3-tert-butyl-7-(2,3,4-trimethoxyphenyl)-4H-[1,3,4]thiadiazolo[2,3-c][1,2,4]triazin-4-one

V. J. Chandraprabha et al.

Summary: The title compound was synthesized and characterized using various methods, revealing its crystal structure, hydrogen bonding patterns, and thermal decomposition temperature. Additionally, its larvicidal and antifungal activities were evaluated.

JOURNAL OF MOLECULAR STRUCTURE (2021)

Article Toxicology

Investigation of the protective effect of acetazolamide and SLC-0111 on carbon tetrachloride-induced toxicity in fruit fly

Eda Gunes et al.

Summary: The study revealed that AAZ and SLC-0111 can protect fruit flies from the toxicity of carbon tetrachloride, positively affecting their survival and development, and influencing certain biochemical parameters.

TOXICOLOGY REPORTS (2021)

Article Chemistry, Multidisciplinary

Antidiabetic, antioxidant, DFT and molecular docking studies of a triazene derivative and its transition metal complexes

Surya Philip et al.

RESEARCH ON CHEMICAL INTERMEDIATES (2020)

Review Biochemistry & Molecular Biology

Mechanisms of Multidrug Resistance in Cancer Chemotherapy

Karol Bukowski et al.

INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES (2020)

Article Biochemistry & Molecular Biology

Synthesis and cytotoxic activities of novel copper and silver complexes of 1,3-diaryltriazene-substituted sulfonamides

Dilek Canakci et al.

JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (2019)

Review Pharmacology & Pharmacy

Drug discovery and computational strategies in the multitarget drugs era

Jessika de Oliveira Viana et al.

BRAZILIAN JOURNAL OF PHARMACEUTICAL SCIENCES (2018)

Article Biochemistry & Molecular Biology

Discovery of novel 1,3-diaryltriazene sulfonamides as carbonic anhydrase I, II, VII, and IX inhibitors

Suleyman Akocak et al.

JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (2018)

Article Entomology

A new method for the production of sterile colonies of Lucilia sericata

N. E. Gasz et al.

MEDICAL AND VETERINARY ENTOMOLOGY (2017)

Article Biochemistry & Molecular Biology

Sulfadiazine Salicylaldehyde-Based Schiff Bases: Synthesis, Antimicrobial Activity and Cytotoxicity

Martin Kratky et al.

MOLECULES (2017)

Article Chemistry, Medicinal

Anti-mycobacterial activity of 1,3-diaryltriazenes

Davie Cappoen et al.

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2014)

Article Chemistry, Medicinal

Synthesis of novel thiadiazolotriazin-4-ones and study of their mosquito-larvicidal and antibacterial properties

Prakash Anil Castelino et al.

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2014)

Review Oncology

Temozolomide and unusual indications: Review of literature

Zuzana Tatar et al.

CANCER TREATMENT REVIEWS (2013)

Article Chemistry, Multidisciplinary

In Vitro Evaluation of Triazenes: DNA Cleavage, Antibacterial Activity and Cytotoxicity against Acute Myeloid Leukemia Cells

Vanessa O. Domingues et al.

JOURNAL OF THE BRAZILIAN CHEMICAL SOCIETY (2010)

Article Biochemistry & Molecular Biology

Antiviral and cytotoxic activities of aminoarylazo compounds and aryltriazene derivatives

Michele Tonelli et al.

BIOORGANIC & MEDICINAL CHEMISTRY (2009)

Article Dermatology

Rearing larvae of Lucilia sericata for chronic ulcer treatment -: an improved method

H Wolff et al.

ACTA DERMATO-VENEREOLOGICA (2005)

Article Chemistry, Applied

Solid-phase synthesis of urea and amide libraries using the T2 triazene linker

S Bräse et al.

JOURNAL OF COMBINATORIAL CHEMISTRY (2000)

Article Biochemistry & Molecular Biology

Triazene drug metabolites. Part 17: Synthesis and plasma hydrolysis of acyloxymethyl carbamate derivatives of antitumour triazenes

E Carvalho et al.

BIOORGANIC & MEDICINAL CHEMISTRY (2000)