4.7 Article

Synthesis of the Key Intermediate of SM-406 (Xevinapant) and Its Analogues

相关参考文献

注意:仅列出部分参考文献,下载原文获取全部文献信息。
Review Biochemistry & Molecular Biology

Fukuyama reduction, Fukuyama coupling and Fukuyama-Mitsunobu alkylation: recent developments and synthetic applications

Sana Sikandar et al.

Summary: The Fukuyama reaction is an important method for the synthesis of multifunctional aldehydes, secondary amines, and ketones due to its mild reaction conditions. The use of thioesters in this reaction is attractive for organic chemists as they are easily accessible from corresponding carboxylic acids. The Fukuyama-Mitsunobu reaction utilizes 2-nitrobenzenesulfonyl (Ns) for the protection/activation/deprotection of primary amines to afford secondary amines in good yields and high enantioselectivities.

MOLECULAR DIVERSITY (2022)

Article Chemistry, Medicinal

Structure-Based Discovery of SD-36 as a Potent, Selective, and Efficacious PROTAC Degrader of STAT3 Protein

Haibin Zhou et al.

JOURNAL OF MEDICINAL CHEMISTRY (2019)

Review Chemistry, Organic

Design, synthesis, conformational analysis and application of indolizidin-2-one dipeptide mimics

Arkady Khashper et al.

ORGANIC & BIOMOLECULAR CHEMISTRY (2014)

Article Chemistry, Medicinal

Structure-Based Design of Conformationally Constrained, Cell-Permeable STAT3 Inhibitors

Jianyong Chen et al.

ACS MEDICINAL CHEMISTRY LETTERS (2010)

Review Chemistry, Multidisciplinary

Design of Small-Molecule Peptidic and Nonpeptidic Smac Mimetics

Haiying Sun et al.

ACCOUNTS OF CHEMICAL RESEARCH (2008)

Article Chemistry, Organic

Synthesis of 5/7-, 5/8- and 5/9-bicyclic lactam templates as constraints for external β-turns

HME Duggan et al.

ORGANIC & BIOMOLECULAR CHEMISTRY (2005)

Article Chemistry, Organic

Functionalized azabicycloalkane amino acids by nitrone 1,3-dipolar intramolecular cycloaddition

L Manzoni et al.

JOURNAL OF ORGANIC CHEMISTRY (2005)

Article Chemistry, Multidisciplinary

Structure-based design of potent, conformationally constrained Smac mimetics

HY Sun et al.

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2004)

Article Chemistry, Applied

A solid phase library synthesis of hydroxyindoline-derived tricyclic derivatives by Mitsunobu approach

P Arya et al.

JOURNAL OF COMBINATORIAL CHEMISTRY (2004)