4.4 Article

Catalytic Enantioselective Synthesis of 4-Amino-5-aryltetrahydro-1H-benzo[c]azepines by an Aminoarylation Reaction

相关参考文献

注意:仅列出部分参考文献,下载原文获取全部文献信息。
Article Chemistry, Organic

Asymmetric aminoarylation for the synthesis of trans-3-amino-4-aryltetrahydroquinolines: An access to aza-analogue of dihydrexidine

Sk Md Samim Akhtar et al.

Summary: A proficient stereoselective aminoarylation reaction of N-cinnamylanilines was developed based on a two-step protocol involving catalytic enantioselective aziridination and subsequent 6-endo-tet Friedel-Crafts cyclization. The reaction showed excellent diastereo- and enantioselectivity in the synthesis of trans-3-amino-4-aryltetrahydroquinolines, with the potential for concise synthesis of bioactive compounds.

TETRAHEDRON (2022)

Review Chemistry, Multidisciplinary

Domino-Ring Opening-Cyclization (DROC) of Donor-Acceptor (DA) Cyclopropanes

Ranadeep Talukdar et al.

ISRAEL JOURNAL OF CHEMISTRY (2016)

Article Chemistry, Organic

Asymmetric synthesis of 3-substituted tetrahydro-2-benzazepines

Matthias P. Quick et al.

ORGANIC & BIOMOLECULAR CHEMISTRY (2015)

Article Chemistry, Inorganic & Nuclear

7-endo cyclization of 2,3-epoxyamides and 2,3-aziridine carboxamides by intramolecular Friedel-Crafts reaction

Angel Palillero-Cisneros et al.

TETRAHEDRON-ASYMMETRY (2015)

Article Chemistry, Organic

Concise Synthesis of 2-Benzazepine Derivatives and Their Biological Activity

Masahiro So et al.

JOURNAL OF ORGANIC CHEMISTRY (2012)

Article Chemistry, Inorganic & Nuclear

Catalytic enantioselective synthesis of the dopamine D1 antagonist ecopipam

Saumen Hajra et al.

TETRAHEDRON-ASYMMETRY (2012)

Article Chemistry, Multidisciplinary

Catalytic enantioselective synthesis of A-86929, a dopamine D1 agonist

Saumen Hajra et al.

CHEMICAL COMMUNICATIONS (2011)

Article Chemistry, Inorganic & Nuclear

Asymmetric synthesis of the dopamine D1 agonist, dihydrexidine

Saumen Hajra et al.

TETRAHEDRON-ASYMMETRY (2011)

Article Chemistry, Medicinal

Rigid Analogues of Antimitotic Indolobenzazepinones: New Insights into Tubulin Binding via Molecular Modeling

Valerie Pons et al.

ACS MEDICINAL CHEMISTRY LETTERS (2011)

Article Chemistry, Inorganic & Nuclear

First asymmetric synthesis of (un)substituted bridged tetrahydro-2-benzazepines

David Dumoulin et al.

TETRAHEDRON-ASYMMETRY (2010)

Article Chemistry, Applied

A Catalytic and Enantioselective Synthesis of trans-2-Amino-1-aryltetralins

Saumen Hajra et al.

ADVANCED SYNTHESIS & CATALYSIS (2009)

Article Chemistry, Medicinal

11-Phenyl-[b,e]-dibenzazepine compounds: Novel antitumor agents

Raed A. Al-Qawasmeh et al.

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2009)

Article Biochemistry & Molecular Biology

SAR studies of capsazepinoid bronchodilators. Part 2: Chlorination and catechol replacement in the A-ring

Magnus Berglund et al.

BIOORGANIC & MEDICINAL CHEMISTRY (2008)

Article Biochemistry & Molecular Biology

SAR studies of capsazepinoid bronchodilators.: Part 1:: The importance of the catechol moiety and aspects of the B-ring structure

Maria F. Dalence-Guzman et al.

BIOORGANIC & MEDICINAL CHEMISTRY (2008)

Article Chemistry, Organic

Synthesis of 5-hydroxy-2,3,4,5-tetrahydro-[1H]-2-benzazepin-4-ones: selective antagonists of muscarinic (M-3) receptors

Benjamin Bradshaw et al.

ORGANIC & BIOMOLECULAR CHEMISTRY (2008)

Review Chemistry, Organic

Nucleophilic ring opening of aziridines

XE Hu

TETRAHEDRON (2004)

Article Chemistry, Organic

Convenient switching of 7-endo/6-exo radical cyclization

A Kamimura et al.

TETRAHEDRON LETTERS (2004)

Article Chemistry, Medicinal

Synthesis of N,N′-disubstituted 3-aminobenzo[c] and [d]azepin-2-ones as potent and specific farnesyl transferase inhibitors

T Le Diguarher et al.

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2004)

Article Pharmacology & Pharmacy

Chronic vasopeptidase inhibition normalizes diabetic endothelial dysfunction

S Schäfer et al.

EUROPEAN JOURNAL OF PHARMACOLOGY (2004)

Article Chemistry, Applied

Solid-supported solution-phase synthesis of 4-amino-1,2,4,5-tetrahydro-2-benzazepine-3-ones

I Van den Eynde et al.

JOURNAL OF COMBINATORIAL CHEMISTRY (2004)

Review Pharmacology & Pharmacy

Novel angiotensin II inhibitors in cardiovascular medicine

M Burnier

EXPERT OPINION ON INVESTIGATIONAL DRUGS (2001)

Article Chemistry, Organic

Asymmetric synthesis of 1-aryl 2,3,4,5-tetrahydro-2-benz[c]azepines

R Gamez-Montano et al.

TETRAHEDRON LETTERS (2001)

Review Pharmacology & Pharmacy

Galantamine - A review of its use in Alzheimer's disease

LJ Scott et al.

Article Multidisciplinary Sciences

Tumor selective G2/M cell cycle arrest and apoptosis of epithelial and hematological malignancies by BBL22, a benzazepine

WL Xia et al.

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2000)