相关参考文献
注意:仅列出部分参考文献,下载原文获取全部文献信息。An appraisal on synthetic and pharmaceutical perspectives of pyrazolo[4,3-d]pyrimidine scaffold
Srinivasulu Cherukupalli et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2018)
Synthesis, characterization and cytotoxicity studies of 1,2,3-triazoles and 1,2,4-triazolo [1,5-a] pyrimidines in human breast cancer cells
Maryam Gilandoust et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2018)
Design, synthesis and evaluation of photoactivatable derivatives of microtubule (MT)-active [1,2,4]triazolo[1,5-a]pyrimidines
Killian Oukoloff et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2018)
Synthesis of New [1,2,4]Triazolo[1,5-a]pyrimidine Derivatives: Reactivity of 3-Amino[1,2,4]triazole towards Enaminonitriles and Enaminones
Abdulaziz Alnajjar et al.
JOURNAL OF HETEROCYCLIC CHEMISTRY (2018)
Pd-catalyzed Suzuki/Sonogashira cross-coupling reaction and the direct sp3 arylation of 7-chloro-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidine
Mohammed Loubidi et al.
TETRAHEDRON LETTERS (2018)
Synthesis of novel 1, 2, 4-triazolopyrimidines and their evaluation as antimicrobial agents
Ameen A. Abu-Hashem et al.
MEDICINAL CHEMISTRY RESEARCH (2017)
Design, synthesis and biological evaluation of [1,2,4]triazolo[1,5-a]pyrimidines as potent lysine specific demethylase 1 (LSD1/KDM1A) inhibitors
Shuai Wang et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2017)
An insight on synthetic and medicinal aspects of pyrazolo[1,5-a] pyrimidine scaffold
Srinivasulu Cherukupalli et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2017)
A new synthesis of 2-(aminoalkyl)-1,2,4-triazolo[1,5-a]pyrimidines
Mikhail A. Prezent et al.
MENDELEEV COMMUNICATIONS (2017)
Efficient and regioselective one-step synthesis of 7-aryl-5-methyl- and 5-aryl-7-methyl-2-amino[1,2,4] triazolo[1,5-a] pyrimidine derivatives
Serena Massari et al.
ORGANIC & BIOMOLECULAR CHEMISTRY (2017)
A synthesis of 6-functionalized 4,7-dihydro[1,2,4]triazolo[1,5-a]pyrimidines
Maksim A. Kolosov et al.
TETRAHEDRON LETTERS (2017)
Synthesis and structure activity relationship investigation of triazolo[1,5-a]pyrimidines as CB2 cannabinoid receptor inverse agonists
Mojgan Aghazadeh Tabrizi et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2016)
Multicomponent facile synthesis of highly substituted [1,2,4]triazolo[1,5-a] pyrimidines
Belgheis Adrom et al.
JOURNAL OF CHEMICAL RESEARCH (2016)
Microwave-assisted synthesis and evaluation of antibacterial activity of novel 6-fluoroaryl-[1,2,4]triazolo[1,5-a]pyrimidines
Egor V. Verbitskiy et al.
ARKIVOC (2016)
Pyrazole clubbed triazolo[1,5-a]pyrimidine hybrids as an anti-tubercular agents: Synthesis, in vitro screening and molecular docking study
Jaimin D. Bhatt et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2015)
Asymmetric synthesis of pyrazoles and pyrazolones employing the reactivity of pyrazolin-5-one derivatives
Pankaj Chauhan et al.
CHEMICAL COMMUNICATIONS (2015)
Fused heterocycles bearing bridgehead nitrogen as potent HIV-1 NNRTIs. Part 3: Optimization of [1,2,4]triazolo[1,5-a]pyrimidine core via structure-based and physicochemical property-driven approaches
Boshi Huang et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2015)
Synthesis and Evaluation of 1,2,4-Triazolo[1,5-a]pyrimidines as Antibacterial Agents Against Enterococcus faecium
Huan Wang et al.
JOURNAL OF MEDICINAL CHEMISTRY (2015)
Base-catalyzed one-step synthesis of 5,7-disubstituted-1,2,4-triazolo[1,5-a]pyrimidines
Xinhua He et al.
TETRAHEDRON LETTERS (2015)
Fused heterocycles bearing bridgehead nitrogen as potent HIV-1 NNRTIs. Part 2: Discovery of novel [1,2,4]Triazolo[1,5-a]pyrimidines using a structure-guided core-refining approach
Liu Wang et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2014)
Ultrasound irradiation promotes the synthesis of new 1,2,4-triazolo [1,5-a]pyrimidine
Clarissa P. Frizzo et al.
ULTRASONICS SONOCHEMISTRY (2014)
Medicinal attributes of pyrazolo[3,4-d]pyrimidines: A review
Monika Chauhan et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2013)
Synthesis and antimicrobical evaluation of a novel class of 1,3,4-thiadiazole: Derivatives bearing 1,2,4-triazolo[1,5-a] pyrimidine moiety
Yin Luo et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2013)
Thiamine hydrochloride (VB1): an efficient promoter for the one-pot synthesis of benzo[4,5]imidazo[1,2-a]pyrimidine and [1,2,4]triazolo[1,5-a] pyrimidine derivatives in water medium
Junhua Liu et al.
GREEN CHEMISTRY (2012)
Synthesis and biological evaluation of novel steroidal[17,16-d][1,2,4]triazolo [1,5-a]pyrimidines
Li-Hua Huang et al.
STEROIDS (2012)
A dinuclear silver compound with 5,6,7-trimethyl-[1,2,4]triazolo[1,5-a]pyrimidine with a short Ag-Ag bond. Synthesis, characterization, single-crystal structure analysis and cytostatic activity
Koen Bavelaar et al.
INORGANICA CHIMICA ACTA (2011)
General Principles of Antimicrobial Therapy
Surbhi Leekha et al.
MAYO CLINIC PROCEEDINGS (2011)
Fluorinated 1,2,4-Triazolo[1,5-a]pyrimidine-6-carboxylic Acid Derivatives as Antimycobacterial Agents
Hamdy M. Abdel-Rahman et al.
ARCHIV DER PHARMAZIE (2009)
Synthesis and Fungicidal Activities of New 1,2,4-Triazolo[1,5-a]pyrimidines
Qiong Chen et al.
CHEMISTRY & BIODIVERSITY (2009)
Synthesis and antimicrobial activity of certain new 1,2,4-Triaz-olo[1,5-a]pyrimidine derivatives
Yaser A. -H. Mostafa et al.
ARCHIVES OF PHARMACAL RESEARCH (2008)
Synthesis and cytotoxicity studies of novel [1,2,4]triazolo[1,5-a]pyrimidine-7-amines
Xin Zhai et al.
CHEMICAL & PHARMACEUTICAL BULLETIN (2008)
Synthesis, antifungal activity and CoMFA analysis of novel l,2,4-triazolo[1,5-a]pyrimidine derivatives
Qiong Chen et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2008)
Synthesis of some novel pyrazolo[1,5-a]pyrimidine, 1,2,4-triazolo[1,5-a]pyrimidine, pyrido[2,3-d]pyrimidine, pyrazolo[5,1-c]-1,2,4-triazine and 1,2,4-triazolo[5,1-c]-1,2,4-triazine derivatives incorporating a thiazolo[3,2-a]benzimidazole moiety
Hatem A. Abdel-Aziz et al.
JOURNAL OF HETEROCYCLIC CHEMISTRY (2008)
Synthesis and anti-tumor activities of novel [1,2,4]triazolo[1,5-a]pyrimidines
Xiang-Lin Zhao et al.
MOLECULES (2007)
Synthesis and SAR of [1,2,4]Triazolo[1,5-a]pyrimidines, a class of anticancer agents with a unique mechanism of tubulin inhibition
Nan Zhang et al.
JOURNAL OF MEDICINAL CHEMISTRY (2007)
Microwave-assisted three-component synthesis of 7-aryl-2-alkylthio-4,7-dihydro-1,2,4-triazolo[1,5-a]-pyrimidine-6-carboxamides and their selective reduction
VA Chebanov et al.
JOURNAL OF COMBINATORIAL CHEMISTRY (2006)
Effect of trapidil, an antiplatelet and vasodilator agent on gentamicin-induced nephrotoxicity in rats
K Büyükafsar et al.
PHARMACOLOGICAL RESEARCH (2001)