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PSYCHIATRY RESEARCH-NEUROIMAGING (2008)
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A. D. Gee et al.
CURRENT RADIOPHARMACEUTICALS (2008)
Synthesis and biological evaluation in rat and cat of [18F]12ST05 as a potential 5-HT6 PET radioligand
Sandrine Tang et al.
NUCLEAR MEDICINE AND BIOLOGY (2007)
Elevated serotonin transporter binding in major depressive disorder assessed using positron emission tomography and [11C]DASB;: Comparison with bipolar disorder
Dara M. Cannon et al.
BIOLOGICAL PSYCHIATRY (2007)
Anorexia induced by activation of serotonin 5-HT4 receptors is mediated by increases in CART in the nucleus accumbens
Alexandra Jean et al.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2007)
Serotonin4 (5-HT4) receptor Agonists are putative antidepressants with a rapid onset of action
Guillaume Lucas et al.
NEURON (2007)
Differences of cortical 5-HT2A receptor binding index with SPECT in subtypes of anorexia nervosa:: Relationship with personality traits?
Ingeborg Goethals et al.
JOURNAL OF PSYCHIATRIC RESEARCH (2007)
Disulfiram inhibits defluorination of 18F-FCWAY, reduces bone radioactivity, and enhances visualization of radioligand binding to serotonin 5-HT1A receptors in human brain
Yong Hoon Ryu et al.
JOURNAL OF NUCLEAR MEDICINE (2007)
Synthesis and in vivo evaluation of a novel 5-HT1A receptor agonist radioligand [O-methyl-11C]2-(4-(4-(2-methoxyphenyl) piperazin-1-yl)butyl)-4-methyl-1,2,4-triazine-3, 5(2H,4H)dione in nonhuman primates
J. S. Dileep Kumar et al.
EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING (2007)
PET [11C]DASB imaging of serotonin transporters in patients with alcoholism
Amira K. Brown et al.
ALCOHOLISM-CLINICAL AND EXPERIMENTAL RESEARCH (2007)
[F-18]MPPF as a tool fot the in vivo imaging of 5-HT1A receptors in animal and human brain
Nicolas Aznavour et al.
NEUROPHARMACOLOGY (2007)
The 5-HT3 receptor as a therapeutic target
Andrew J. Thompson et al.
EXPERT OPINION ON THERAPEUTIC TARGETS (2007)
Serotonin transporter occupancy induced by paroxetine in patients with major depression disorder:: a 123I-ADAM SPECT study
Ana M. Catafau et al.
PSYCHOPHARMACOLOGY (2006)
Serotonin transporters - Structure and function
Gary Rudnick
JOURNAL OF MEMBRANE BIOLOGY (2006)
Measurement of serotonin transporter binding with PET and [11C]MADAM:: A test-retest reproducibility study
Johan Lundberg et al.
SYNAPSE (2006)
Radiochemical synthesis and tissue distribution of p-[18F]DMPPF, a new 5-HT1A ligand for PET, in rats
Caroline Defraiteur et al.
NUCLEAR MEDICINE AND BIOLOGY (2006)
Presynaptic serotonergic modulation of 5-HT and acetylcholine release in the hippocampus and the cortex of 5-HT1B-receptor knockout mice
Susanne Rutz et al.
BRAIN RESEARCH BULLETIN (2006)
Imaging of serotonin transporters and its blockade by citalopram in patients with major depression using a novel SPECT ligand [123I]-ADAM
N Herold et al.
JOURNAL OF NEURAL TRANSMISSION (2006)
Serotonin 1A receptors in the living brain of Alzheimer's disease patients
V Kepe et al.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2006)
Synthesis and in vivo validation of [O-methyl-11C]2-{4-[4-(7-methoxynaphthalen-1-yl)piperazin-yl]butyl}-4-methy1-2H-[1,2,4]triazine-3,5-dione:: A novel 5-HT1A receptor agonist positron emission tomography ligand
JSD Kumar et al.
JOURNAL OF MEDICINAL CHEMISTRY (2006)
5-HT1B receptors and aggression:: A review
B Olivier et al.
EUROPEAN JOURNAL OF PHARMACOLOGY (2005)
[11C]MADAM, a new serotonin transporter radioligand characterized in the monkey brain by PET
C Halldin et al.
SYNAPSE (2005)
4-(2-Aminoethoxy)-N-(phenylsulfonyl)indoles as novel 5-HT6 receptor ligands
P Zhou et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2005)
No change in serotonin type 1A receptor binding in patients with posttraumatic stress disorder
O Bonne et al.
AMERICAN JOURNAL OF PSYCHIATRY (2005)
5-HT1A receptor binding and intracerebral activity in temporal lobe epilepsy:: an [18F]MPPF-PET study
I Merlet et al.
BRAIN (2004)
A database of [18F]-altanserin binding to 5-HT2A receptors in normal volunteers:: normative data and relationship to physiological and demographic variables
KH Adams et al.
NEUROIMAGE (2004)
Decreased hippocampal 5-HT2A receptor binding in major depressive disorder:: In vivo measurement with [18F]Altanserin positron emission tomography
MA Mintun et al.
BIOLOGICAL PSYCHIATRY (2004)
Reduced serotonin type 1A receptor binding in panic disorder
A Neumeister et al.
JOURNAL OF NEUROSCIENCE (2004)
Distribution of 5-HT7 receptors in the human brain:: a preliminary autoradiographic study using [3H]SB-269970
K Varnäs et al.
NEUROSCIENCE LETTERS (2004)
In vivo quantification by SPECT of [123I] ADAM bound to serotonin transporters in the brains of rabbits
XX Ye et al.
NUCLEAR MEDICINE AND BIOLOGY (2004)
Biodistribution and radiation dosimetry of [11C]DASB in baboons
MJ Bélanger et al.
NUCLEAR MEDICINE AND BIOLOGY (2004)
The pyridinyl-6 position of WAY-100635 as a site for radiofluorination-effect on 5-HT1A receptor radioligand behavior in vivo
JA McCarron et al.
MOLECULAR IMAGING AND BIOLOGY (2004)
PET brain imaging with [11C](+)McN5652 shows increased serotonin transporter availability in major depression
M Reivich et al.
JOURNAL OF AFFECTIVE DISORDERS (2004)
Serotonin1B receptors:: from protein to physiological function and behavior
Y Sari
NEUROSCIENCE AND BIOBEHAVIORAL REVIEWS (2004)
Serotonin transporters in obsessive-compulsive disorder:: A positron emission tomography study with [11C]McN 5652
HB Simpson et al.
BIOLOGICAL PSYCHIATRY (2003)
In vivo measurement of the serotonin transporter with (S)-([18F]fluoromethyl)-(+)-McN5652
P Brust et al.
NEUROPSYCHOPHARMACOLOGY (2003)
Distribution of 5-HT4 receptors in the postmortem human brain -: an autoradiographic study using [125I]SB 207710
K Varnäs et al.
EUROPEAN NEUROPSYCHOPHARMACOLOGY (2003)
Synthesis of a [6-pyridinyl-18F]-labelled fluoro derivative of WAY-100635 as a candidate radioligand for brain 5-HT1A receptor imaging with PET
M Karramkam et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2003)
Imaging of the 5-HT2A system:: age-, gender-, and Alzheimer's disease-related findings
J Versijpt et al.
NEUROBIOLOGY OF AGING (2003)
Prefrontal 5-HT2a receptor binding index, hopelessness and personality characteristics in attempted suicide
C van Heeringen et al.
JOURNAL OF AFFECTIVE DISORDERS (2003)
PET imaging of 5-HT1A receptor binding in patients with temporal lobe epilepsy
MT Toczek et al.
NEUROLOGY (2003)
Positron emission tomography imaging of the serotonin transporter in the pig brain using [11C](+)-McN5652 and S-([18F]fluoromethyl)-(+)-McN5652
P Brust et al.
SYNAPSE (2003)
[11C]-DASB, a tool for in vivo measurement of SSRI-induced occupancy of the serotonin transporter:: PET characterization and evaluation in cats
N Ginovart et al.
SYNAPSE (2003)
Biodistribution and radiation dosimetry of [I-123]ADAM in healthy human subjects: preliminary results
TA Kauppinen et al.
EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING (2003)
Radioiodinated SB 207710 as a radioligand in vivo: imaging of brain 5-HT(4) receptors with SPET
VW Pike et al.
EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING (2003)
S-[F-18]fluoromethyl-(+)-McN5652, a PET tracer for the serotonin transporter: Evaluation in rats
P Marjamaki et al.
SYNAPSE (2003)
Opioid hyperalgesia and tolerance versus 5-HT1A receptor-mediated inverse tolerance
XJ Xu et al.
TRENDS IN PHARMACOLOGICAL SCIENCES (2003)
Reduced 5-HT2A receptor binding after recovery from anorexia nervosa
GK Frank et al.
BIOLOGICAL PSYCHIATRY (2002)
Synthesis and preliminary PET study of the 5-HT7 receptor antagonist [11C]DR4446
MR Zhang et al.
JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS (2002)
5-HT6 receptor binding sites in schizophrenia and following antipsychotic drug administration:: Autoradiographic studies with [125I]SB-258585
SZ East et al.
SYNAPSE (2002)
Biodistribution study of [123I] ADAM in mice:: correlation with whole body autoradiography
KH Lin et al.
NUCLEAR MEDICINE AND BIOLOGY (2002)
Pharmacokinetics and brain distribution in non human primate of R(-)[123I]DOI, A 5HT2A/2C serotonin agonist
Y Zea-Ponce et al.
NUCLEAR MEDICINE AND BIOLOGY (2002)
In vitro and in vivo characterisation of [11C]-DASB:: a probe for in vivo measurements of the serotonin transporter by positron emission tomography
AA Wilson et al.
NUCLEAR MEDICINE AND BIOLOGY (2002)
Serotonin transporter binding in patients with mood disorders:: a PET study with [11C](+)McN5652
T Ichimiya et al.
BIOLOGICAL PSYCHIATRY (2002)
The distribution of 5-HT6 receptors in rat brain:: an autoradiographic binding study using the radiolabelled 5-HT6 receptor antagonist [125I]SB-258585
JC Roberts et al.
BRAIN RESEARCH (2002)
A database of [C-11]WAY-100635 binding to 5-HT1A receptors in normal male volunteers: Normative data and relationship to methodological, demographic, physiological, and behavioral variables
EA Rabiner et al.
NEUROIMAGE (2002)
Carbon-11 labelling of MADAM in two different positions: a highly selective PET radioligand for the serotonin transporter
J Tarkiainen et al.
JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS (2001)
Occupancy of serotonin transporters by paroxetine and citalopram during treatment of depression:: A [11C]DASB PET imaging study
JH Meyer et al.
AMERICAN JOURNAL OF PSYCHIATRY (2001)
Analyses of [18F]altanserin bolus injection PET data.: I:: Consideration of radiolabeled metabolites in baboons
JC Price et al.
SYNAPSE (2001)
Reproducibility of in vivo brain measures of 5-HT2A receptors with PET and [18F]deuteroaltanserin
JC Soares et al.
PSYCHIATRY RESEARCH-NEUROIMAGING (2001)
Comparison of [18F]altanserin and [18F]deuteroaltanserin for PET imaging of serotonin2A receptors in baboon brain:: pharmacological studies
JK Staley et al.
NUCLEAR MEDICINE AND BIOLOGY (2001)
New halogenated [11C]WAY analogues, [11C]6FPWAY and [11C]6BPWAY -: Radiosynthesis and assessment as radioligands for the study of brain 5-HT1A receptors in living monkey
J Sandell et al.
NUCLEAR MEDICINE AND BIOLOGY (2001)
Decreased frontal serotonin 5-HT2a receptor binding index in deliberate self-harm patients
K Audenaert et al.
EUROPEAN JOURNAL OF NUCLEAR MEDICINE (2001)
Equilibrium modeling of 5-HT2A receptors with [18F]deuteroaltanserin and PET:: Feasibility of a constant infusion paradigm
CH van Dyck et al.
NUCLEAR MEDICINE AND BIOLOGY (2000)
Imaging the serotonin transporter with positron emission tomography:: initial human studies with [11C]DAPP and [11C]DASB
S Houle et al.
EUROPEAN JOURNAL OF NUCLEAR MEDICINE (2000)
Novel radiotracers for imaging the serotonin transporter by positron emission tomography:: Synthesis, radiosynthesis, and in vitro and ex vivo evaluation of 11C-labeled 2-(phenylthio)araalkylamines
AA Wilson et al.
JOURNAL OF MEDICINAL CHEMISTRY (2000)
Characterization of [125I]-SB-258585 binding to human recombinant and native 5-HT6 receptors in rat, pig and human brain tissue
WD Hirst et al.
BRITISH JOURNAL OF PHARMACOLOGY (2000)
[18F]p-MPPF:: A radiolabeled antagonist for the study of 5-HT1A receptors with PET
A Plenevaux et al.
NUCLEAR MEDICINE AND BIOLOGY (2000)
2-((2-((Dimethylamino)methyl)phenyl)thio-5-iodophenylamine (ADAM): An improved serotonin transporter ligand
S Oya et al.
NUCLEAR MEDICINE AND BIOLOGY (2000)
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