相关参考文献
注意:仅列出部分参考文献,下载原文获取全部文献信息。Molecular probes for the human adenosine receptors
Xue Yang et al.
PURINERGIC SIGNALLING (2021)
Pharmacological characterization of DPTN and other selective A3 adenosine receptor antagonists
Zhan-Guo Gao et al.
PURINERGIC SIGNALLING (2021)
Substituted 4-phenylthiazoles: Development of potent and selective A1, A3 and dual A1/A3 adenosine receptor antagonists
Aliaa Abdelrahman et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2020)
Direct Comparison of (N)-Methanocarba and Ribose-Containing 2-Arylalkynyladenosine Derivatives as A3 Receptor Agonists
Dilip K. Tosh et al.
ACS MEDICINAL CHEMISTRY LETTERS (2020)
Truncated (N)-Methanocarba Nucleosides as Partial Agonists at Mouse and Human A3 Adenosine Receptors: Affinity Enhancement by N6-(2-Phenylethyl) Substitution
Dilip K. Tosh et al.
JOURNAL OF MEDICINAL CHEMISTRY (2020)
The Anti-Inflammatory and Pain-Relieving Effects of AR170, an Adenosine A3Receptor Agonist, in a Rat Model of Colitis
Luca Antonioli et al.
CELLS (2020)
Pharmacological characterisation of novel adenosine A3 receptor antagonists
Kerry Barkan et al.
SCIENTIFIC REPORTS (2020)
Nucleotide P2Y1 receptor agonists are in vitro and in vivo prodrugs of A1/A3 adenosine receptor agonists: implications for roles of P2Y1 and A1/A3 receptors in physiology and pathology
Theodore E. Liston et al.
PURINERGIC SIGNALLING (2020)
撤稿声明: CNS Physicochemical Property Space Shaped by a Diverse Set of Molecules with Experimentally Determined Exposure in the Mouse Brain (Retraction of Vol 60, Pg 5943, 2017)
Zoran Rankovic
JOURNAL OF MEDICINAL CHEMISTRY (2019)
The A3 adenosine receptor agonist, namodenoson, ameliorates non-alcoholic steatohepatitis in mice
Pnina Fishman et al.
INTERNATIONAL JOURNAL OF MOLECULAR MEDICINE (2019)
A(3) Adenosine Receptors as Modulators of Inflammation: From Medicinal Chemistry to Therapy
Kenneth A. Jacobson et al.
MEDICINAL RESEARCH REVIEWS (2018)
GPCRdb in 2018: adding GPCR structure models and ligands
Gaspar Pandy-Szekeres et al.
NUCLEIC ACIDS RESEARCH (2018)
Preclinical In Vitro and In Vivo Evaluation of [F-18]FE@SUPPY for Cancer PET Imaging: Limitations of a Xenograft Model for Colorectal Cancer
T. Balber et al.
CONTRAST MEDIA & MOLECULAR IMAGING (2018)
Structure-Affinity Relationships and Structure-Kinetics Relationships of Pyrido[2,1-f]purine-2,4-dione Derivatives as Human Adenosine A3 Receptor Antagonists
Lizi Xia et al.
JOURNAL OF MEDICINAL CHEMISTRY (2017)
Human Adenosine A2A Receptor: Molecular Mechanism of Ligand Binding and Activation
Byron Carpenter et al.
FRONTIERS IN PHARMACOLOGY (2017)
Structure of the Adenosine A1 Receptor Reveals the Basis for Subtype Selectivity
Alisa Glukhova et al.
CELL (2017)
BDDCS, the Rule of 5 and drugability
Leslie Z. Benet et al.
ADVANCED DRUG DELIVERY REVIEWS (2016)
The A3 adenosine receptor (A3AR): therapeutic target and predictive biological marker in rheumatoid arthritis
Pnina Fishman et al.
CLINICAL RHEUMATOLOGY (2016)
Novel thiazole-thiophene conjugates as adenosine receptor antagonists: Synthesis, biological evaluation and docking studies
Dhaivat H. Pandya et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2015)
A Survey of the Role of Noncovalent Sulfur Interactions in Drug Design
Brett R. Beno et al.
JOURNAL OF MEDICINAL CHEMISTRY (2015)
Selectivity is species-dependent: Characterization of standard agonists and antagonists at human, rat, and mouse adenosine receptors
Mohamad Wessam Alnouri et al.
PURINERGIC SIGNALLING (2015)
Endogenous adenosine A(3) receptor activation selectively alleviates persistent pain states
Joshua W. Little et al.
BRAIN (2015)
The role of activated adenosine receptors in degranulation of human LAD2 mast cells
Chi Ting Leung et al.
PURINERGIC SIGNALLING (2014)
The stimulation of A3 adenosine receptors reduces bone-residing breast cancer in a rat preclinical model
Katia Varani et al.
EUROPEAN JOURNAL OF CANCER (2013)
New insight into adenosine receptors selectivity derived from a novel series of [5-substituted-4-phenyl-1,3-thiazol-2-yl] benzamides and furamides
Gajanan S. Inamdar et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2013)
Automated design of ligands to polypharmacological profiles
Jeremy Besnard et al.
NATURE (2012)
CF102 an A3 Adenosine Receptor Agonist Mediates Anti-Tumor and Anti-Inflammatory Effects in the Liver
S. Cohen et al.
JOURNAL OF CELLULAR PHYSIOLOGY (2011)
Pyrimidine Derivatives as Potent and Selective A3 Adenosine Receptor Antagonists
Vicente Yaziji et al.
JOURNAL OF MEDICINAL CHEMISTRY (2011)
Moving beyond Rules: The Development of a Central Nervous System Multiparameter Optimization (CNS MPO) Approach To Enable Alignment of Druglike Properties
Travis T. Wager et al.
ACS CHEMICAL NEUROSCIENCE (2010)
Adenosine A(3) receptors regulate heart rate, motor activity and body temperature
J. N. Yang et al.
ACTA PHYSIOLOGICA (2010)
Synthesis and pharmacological characterization of [125I]MRS1898, a high-affinity, selective radioligand for the rat A3 adenosine receptor
Zhan-Guo Gao et al.
PURINERGIC SIGNALLING (2009)
Design of (N)-methanocarba adenosine 5′-uronamides as species-independent A3 receptor-selective agonists
Artem Melman et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2008)
Synthesis and biological activities of 4-phenyl-5-pyridyl-1,3-thiazole derivatives as selective adenosine A3 antagonists
Seiji Miwatashi et al.
CHEMICAL & PHARMACEUTICAL BULLETIN (2008)
CGH2466, a combined adenosine receptor antagonist, p38 mitogen-activated protein kinase and phosphodiesterase type 4 inhibitor with potent in vitro and in vivo anti-inflammatory activities
A Trifilieff et al.
BRITISH JOURNAL OF PHARMACOLOGY (2005)
Structure-activity relationships of thiazole and thiadiazole derivatives as potent and selective human adenosine A3 receptor antagonists
KY Jung et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2004)
New highly potent and selective adenosine A(3) receptor antagonists
NJ Press et al.
CURRENT TOPICS IN MEDICINAL CHEMISTRY (2004)
N6-substituted adenosine derivatives:: selectivity, efficacy, and species differences at A3 adenosine receptors
ZG Gao et al.
BIOCHEMICAL PHARMACOLOGY (2003)
Thiazole and thiadiazole analogues as a novel class of adenosine receptor antagonists
JE van Muijlwijk-Koezen et al.
JOURNAL OF MEDICINAL CHEMISTRY (2001)
The utilization of a unified pharmacophore query in the discovery of new antagonists of the adenosine receptor family
TR Webb et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2000)