4.3 Article

Synthesis of 4-(1,2,3-triazol-1-yl)-L-phenylalanines

相关参考文献

注意:仅列出部分参考文献,下载原文获取全部文献信息。
Article Chemistry, Medicinal

Modified histidine containing amphipathic ultrashort antifungal peptide, His[2-p-(n-butyl)phenyl]-Trp-Arg-OMe exhibits potent anticryptococcal activity

Krishna K. Sharma et al.

Summary: A new structural class of ultrashort peptide-based antifungal, His(2-aryl)-Trp-Arg, was reported in this study. Structural changes on the His-Trp-Arg scaffold showed the impact of charge and lipophilic character on biological activity. Peptide 14f exhibited potent anticryptococcal activity and showed no cytotoxic effects, acting through nuclear fragmentation, membrane permeabilization, and pore formations in microbial cells.

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2021)

Review Chemistry, Medicinal

Comprehensive review on the anti-bacterial activity of 1,2,3-triazole hybrids

Bo Zhang

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2019)

Article Biochemistry & Molecular Biology

Site-selective installation of an electrophilic handle on proteins for bioconjugation

Bernadette Lee et al.

BIOORGANIC & MEDICINAL CHEMISTRY (2018)

Article Chemistry, Medicinal

New N-phenylpyrrolamide DNA gyrase B inhibitors: Optimization of efficacy and antibacterial activity

Martina Durcik et al.

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2018)

Article Chemistry, Multidisciplinary

Puromycin Analogues Capable of Multiplexed Imaging and Profiling of Protein Synthesis and Dynamics in Live Cells and Neurons

Jingyan Ge et al.

ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2016)

Article Chemistry, Physical

Isonitrile as an Ultrasensitive Infrared Reporter of Hydrogen-Bonding Structure and Dynamics

Michal Maj et al.

JOURNAL OF PHYSICAL CHEMISTRY B (2016)

Article Chemistry, Organic

Room temperature N-arylation of amino acids and peptides using copper(I) and β-diketone

Krishna K. Sharma et al.

ORGANIC & BIOMOLECULAR CHEMISTRY (2015)

Review Chemistry, Multidisciplinary

Beyond click chemistry - supramolecular interactions of 1,2,3-triazoles

Benjamin Schulze et al.

CHEMICAL SOCIETY REVIEWS (2014)

Article Chemistry, Organic

Regiocontrolled palladium-catalyzed and copper-mediated C-H bond functionalization of protected L-histidine

Amit Mahindra et al.

ORGANIC & BIOMOLECULAR CHEMISTRY (2014)

Article Chemistry, Medicinal

Discovery of Short Peptides Exhibiting High Potency against Cryptococcus neoformans

Amit Mahindra et al.

ACS MEDICINAL CHEMISTRY LETTERS (2014)

Review Pharmacology & Pharmacy

The impact of click chemistry in medicinal chemistry

Jingli Hou et al.

EXPERT OPINION ON DRUG DISCOVERY (2012)

Article Biochemical Research Methods

Amino acids: Chemistry, functionality and selected non-enzymatic post-translational modifications

Rainer Bischoff et al.

JOURNAL OF PROTEOMICS (2012)

Article Chemistry, Organic

Rapid microwave-assisted solution-phase peptide synthesis

Amit Mahindra et al.

TETRAHEDRON LETTERS (2012)

Review Chemistry, Multidisciplinary

Click to Join Peptides/Proteins Together

Xuechen Li

CHEMISTRY-AN ASIAN JOURNAL (2011)

Review Chemistry, Multidisciplinary

Click Chemistry: 1,2,3-Triazoles as Pharmacophores

Sandip G. Agalave et al.

CHEMISTRY-AN ASIAN JOURNAL (2011)

Review Pharmacology & Pharmacy

Triazole Antifungal Agents in Invasive Fungal Infections A Comparative Review

Cornelia Lass-Floerl

Review Microbiology

Cationic Amphiphiles, a New Generation of Antimicrobials Inspired by the Natural Antimicrobial Peptide Scaffold

Brandon Findlay et al.

ANTIMICROBIAL AGENTS AND CHEMOTHERAPY (2010)

Article Chemistry, Multidisciplinary

Nitrene addition to exfoliated graphene: a one-step route to highly functionalized graphene

T. Amanda Strom et al.

CHEMICAL COMMUNICATIONS (2010)

Review Biochemistry & Molecular Biology

Protein Chemical Modification on Endogenous Amino Acids

Emmanuel Basle et al.

CHEMISTRY & BIOLOGY (2010)

Article Chemistry, Organic

Click Chemistry to Fluorescent Amino Esters: Synthesis and Spectroscopic Studies

Chun Li et al.

EUROPEAN JOURNAL OF ORGANIC CHEMISTRY (2010)

Article Oncology

Growing Applications of Click Chemistry for Bioconjugation in Contemporary Biomedical Research

Kido Nwe et al.

CANCER BIOTHERAPY AND RADIOPHARMACEUTICALS (2009)

Review Chemistry, Multidisciplinary

Postsynthetic DNA Modification through the Copper-Catalyzed Azide-Alkyne Cycloaddition Reaction

Philipp M. E. Gramlich et al.

ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2008)

Article Chemistry, Medicinal

Phenylglycine and phenylalanine derivatives as potent and selective (H)under-barDAC(1)over-cap (i)under-barnhibitors (SHI-1)

Kevin J. Wilson et al.

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2008)

Review Biotechnology & Applied Microbiology

Peptides and metallic nanoparticles for biomedical applications

Marcelo J. Kogan et al.

NANOMEDICINE (2007)

Article Chemistry, Medicinal

Application of the Suzuki-Miyaura cross-coupling to increase antimicrobial potency generates promising novel antibacterials

Bengt Erik Haug et al.

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2007)

Review Polymer Science

'Click' chemistry in polymer and materials science

Wolfgang H. Binder et al.

MACROMOLECULAR RAPID COMMUNICATIONS (2007)

Article Chemistry, Medicinal

Thyrotropin-releasing hormone (TRH) analogues that exhibit selectivity to TRH receptor subtype 2

N Kaur et al.

JOURNAL OF MEDICINAL CHEMISTRY (2005)

Article Chemistry, Medicinal

Discovery of potent and selective phenylalanine based dipeptidyl peptidase IV inhibitors

JY Xu et al.

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2005)

Article Chemistry, Multidisciplinary

Synthesis of aryl azides and vinyl azides via proline-promoted CuI-catalyzed coupling reactions

W Zhu et al.

CHEMICAL COMMUNICATIONS (2004)

Review Chemistry, Multidisciplinary

The synthesis of peptides and proteins containing non-natural amino acids

DRW Hodgson et al.

CHEMICAL SOCIETY REVIEWS (2004)

Article Chemistry, Medicinal

Antimalarial activities of ring-substituted bioimidazoles

R Jain et al.

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2002)