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Gaspar Pandy-Szekeres et al.
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Denise Wootten et al.
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Rita Santos et al.
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Robert Lutjens et al.
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Viktoriya Syrovatkina et al.
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Yi Zheng et al.
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Intracellular allosteric antagonism of the CCR9 receptor
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Recent updates on GPCR biased agonism
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PHARMACOLOGICAL RESEARCH (2016)
PockDrug-Server: a new web server for predicting pocket druggability on holo and apo proteins
Hiba Abi Hussein et al.
NUCLEIC ACIDS RESEARCH (2015)
Diversity and modularity of G protein-coupled receptor structures
Vsevolod Katritch et al.
TRENDS IN PHARMACOLOGICAL SCIENCES (2012)
Structure-based druggability assessment - identifying suitable targets for small molecule therapeutics
Eric B. Fauman et al.
CURRENT OPINION IN CHEMICAL BIOLOGY (2011)
Allosteric modulators of GPCRs: a novel approach for the treatment of CNS disorders
P. Jeffrey Conn et al.
NATURE REVIEWS DRUG DISCOVERY (2009)
New method for fast and accurate binding-site identification and analysis
Tom Halgren
CHEMICAL BIOLOGY & DRUG DESIGN (2007)
Calcium sensing receptor activators: Calcimimetics
Paul E. Harrington et al.
CURRENT MEDICINAL CHEMISTRY (2007)
Maraviroc (UK-427,857), a potent, orally bioavailable, and selective small-molecule inhibitor of chemokine receptor CCR5 with broad-spectrum anti-human immunodeficiency virus type 1 activity
P Dorr et al.
ANTIMICROBIAL AGENTS AND CHEMOTHERAPY (2005)
International Union of Pharmacology. XLVI. G protein-coupled receptor list
SM Foord et al.
PHARMACOLOGICAL REVIEWS (2005)
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