相关参考文献
注意:仅列出部分参考文献,下载原文获取全部文献信息。Polyphenols and their applications: An approach in food chemistry and innovation potential
Fabio Fernandes de Araujo et al.
FOOD CHEMISTRY (2021)
Synthesis, structure-activity relationships and molecular docking studies of phenyldiazenyl sulfonamides as aromatase inhibitors
Letizia Giampietro et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2021)
Development of new hetero-steroid hybrids with antiproliferative activity against MCF-7 breast cancer cells
Muhamad Mustafa et al.
MONATSHEFTE FUR CHEMIE (2021)
Design, synthesis and biological evaluation of imidazole and triazole-based carbamates as novel aromatase inhibitors
Alessandra Ammazzalorso et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2021)
Synthesis, Cytotoxicity and Anti-Proliferative Activity against AGS Cells of New 3(2H)-Pyridazinone Derivatives Endowed with a Piperazinyl Linker
Mehmet Abdullah Alagoz et al.
PHARMACEUTICALS (2021)
New azolyl-derivatives as multitargeting agents against breast cancer and fungal infections: synthesis, biological evaluation and docking study
Cristina Maccallini et al.
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (2021)
Synthesis, biological evaluation, and docking study of indole aryl sulfonamides as aromatase inhibitors
Marialuigia Fantacuzzi et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2020)
Resveratrol Counteracts Hypoxia-Induced Gastric Cancer Invasion and EMT through Hedgehog Pathway Suppression
Qin-Hong Xu et al.
ANTI-CANCER AGENTS IN MEDICINAL CHEMISTRY (2020)
Aromatase Inhibitors for the Treatment of Breast Cancer: A Journey from the Scratch
Pooja Ratre et al.
ANTI-CANCER AGENTS IN MEDICINAL CHEMISTRY (2020)
Stereoisomer separation of flavanones and flavanone-7-O-glycosides by means of nanoliquid chromatography employing derivatized β-cyclodextrins as mobile-phase additive
Renata Zatopkova et al.
JOURNAL OF SEPARATION SCIENCE (2020)
Antiglioma Activity of Aryl and Amido-Aryl Acetamidine Derivatives Targeting iNOS: Synthesis and Biological Evaluation
Cristina Maccallini et al.
ACS MEDICINAL CHEMISTRY LETTERS (2020)
Synthesis and Biological Evaluation of Halogenated E-Stilbenols as Promising Antiaging Agents
Ester Sara Di Filippo et al.
MOLECULES (2020)
Searching for New Tools to Counteract the Helicobacter pylori Resistance: The Positive Action of Resveratrol Derivatives
Paola Di Fermo et al.
ANTIBIOTICS-BASEL (2020)
Synthesis and evaluation of a large library of nitroxoline derivatives as pancreatic cancer antiproliferative agents
Serena Veschi et al.
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (2020)
Novel Phenyldiazenyl Fibrate Analogues as PPAR α/γ/δ Pan-Agonists for the Amelioration of Metabolic Syndrome
Letizia Giampietro et al.
ACS MEDICINAL CHEMISTRY LETTERS (2019)
Synthesis and cytotoxic effects on pancreatic cancer cells of resveratrol analogs
Barbara De Filippis et al.
MEDICINAL CHEMISTRY RESEARCH (2019)
PPAR-γ agonist GL516 reduces oxidative stress and apoptosis occurrence in a rat astrocyte cell line
Letizia Giampietro et al.
NEUROCHEMISTRY INTERNATIONAL (2019)
Advances in the structural annotation of human carbonic anhydrases and impact on future drug discovery
Alessio Nocentini et al.
EXPERT OPINION ON DRUG DISCOVERY (2019)
Synthesis, molecular docking, and QSAR study of bis-sulfonamide derivatives as potential aromatase inhibitors
Ronnakorn Leechaisit et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2019)
New anticancer drug candidates sulfonamides as selective hCA IX or hCA XII inhibitors
Halise Inci Gul et al.
BIOORGANIC CHEMISTRY (2018)
Sulfonamides as Potential Bioactive Scaffolds
Farhan A. Khan et al.
CURRENT ORGANIC CHEMISTRY (2018)
Potent aromatase inhibitors and molecular mechanism of inhibitory action
Hongjun Kang et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2018)
Synthesis, molecular docking, and QSAR study of sulfonamide-based indoles as aromatase inhibitors
Ratchanok Pingaew et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2018)
Synthesis, Characterization and Evaluation of Gemfibrozil-stilbene Hybrid as Antioxidant
Rosa Amoroso et al.
LETTERS IN DRUG DESIGN & DISCOVERY (2018)
Aromatase inhibitors and apoptotic inducers: Design, synthesis, anticancer activity and molecular modeling studies of novel phenothiazine derivatives carrying sulfonamide moiety as hybrid molecules
Mostafa M. Ghorab et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2017)
Combating breast cancer with non-steroidal aromatase inhibitors (NSAIs): Understanding the chemico-biological interactions through comparative SAR/QSAR study
Nilanjan Adhikari et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2017)
Special Issue: Sulfonamides
Claudiu T. Supuran
MOLECULES (2017)
Genome-wide analysis of the three-way interplay among gene expression, estrogen receptor expression and chemotherapeutic sensitivity in breast cancer
Dong-Xu He et al.
ONCOLOGY REPORTS (2017)
Design, Synthesis, and in vitro and in vivo Evaluations of (Z)-3,4,5-Trimethoxystyrylbenzenesulfonamides/sulfonates as Highly Potent Tubulin Polymerization Inhibitors
Rasala Mahesh et al.
CHEMMEDCHEM (2017)
Anticancer Activity of Stilbene-Based Derivatives
Barbara De Filippis et al.
CHEMMEDCHEM (2017)
Synthesis of Resveratrol Derivatives and In Vitro Screening for Potential Cancer Chemopreventive Activities
Fulvia Orsini et al.
ARCHIV DER PHARMAZIE (2016)
Design, synthesis, and biological evaluation of new arylamide derivatives possessing sulfonate or sulfamate moieties as steroid sulfatase enzyme inhibitors
Mohammed I. El-Gamal et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2016)
Synthesis and biological characterization of 3-(imidazol-1-ylmethyl) piperidine sulfonamides as aromatase inhibitors
Mauro Di Matteo et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2016)
Novel biphenyl bis-sulfonamides as acetyl and butyrylcholinesterase inhibitors: Synthesis, biological evaluation and molecular modeling studies
Sadaf Mutahir et al.
BIOORGANIC CHEMISTRY (2016)
The Use of Stilbene Scaffold in Medicinal Chemistry and Multi-Target Drug Design
Elisa Giacomini et al.
CURRENT MEDICINAL CHEMISTRY (2016)
Rapid determination of nucleotides in infant formula by means of nano-liquid chromatography
Maria Mateos-Vivas et al.
ELECTROPHORESIS (2016)
Aromatase expression and regulation in breast and endometrial cancer
Hong Zhao et al.
JOURNAL OF MOLECULAR ENDOCRINOLOGY (2016)
Resveratrol for breast cancer prevention and therapy: Preclinical evidence and molecular mechanisms
Dona Sinha et al.
SEMINARS IN CANCER BIOLOGY (2016)
Resveratrol and cancer: Challenges for clinical translation
Chandra K. Singh et al.
BIOCHIMICA ET BIOPHYSICA ACTA-MOLECULAR BASIS OF DISEASE (2015)
Pyridine sulfonamide as a small key organic molecule for the potential treatment of type-II diabetes mellitus and Alzheimer's disease: In vitro studies against yeast α-glucosidase, acetylcholinesterase and butyrylcholinesterase
Sadaf Riaz et al.
BIOORGANIC CHEMISTRY (2015)
Recent developments in steroidal and nonsteroidal aromatase inhibitors for the chemoprevention of estrogen-dependent breast cancer
Irshad Ahmad et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2015)
Developing steroidal aromatase inhibitors-an effective armament to win the battle against breast cancer
Mange Ram Yadav et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2015)
PPARα agonists based on stilbene and its bioisosteres: biological evaluation and docking studies
Barbara De Filippis et al.
MEDCHEMCOMM (2015)
Pharmacophore modeling, virtual screening, and 3D-QSAR studies on a series of non-steroidal aromatase inhibitors
Huiding Xie et al.
MEDICINAL CHEMISTRY RESEARCH (2015)
Quinoline- and isoquinoline-sulfonamide analogs of aripiprazole: novel antipsychotic agents?
Pawel Zajdel et al.
FUTURE MEDICINAL CHEMISTRY (2014)
Anti-aromatase effect of resveratrol and melatonin on hormonal positive breast cancer cells co-cultured with breast adipose fibroblasts
Suthat Chottanapund et al.
TOXICOLOGY IN VITRO (2014)
Resveratrol analogs: promising chemopreventive agents
Talysa Ogas et al.
RESVERATROL AND HEALTH (2013)
The development of endocrine therapy for women with breast cancer
Richard Sainsbury
CANCER TREATMENT REVIEWS (2013)
Computational methods for the design of potent aromatase inhibitors
Angelo Danilo Favia et al.
EXPERT OPINION ON DRUG DISCOVERY (2013)
Jaguar: A high-performance quantum chemistry software program with strengths in life and materials sciences
Art D. Bochevarov et al.
INTERNATIONAL JOURNAL OF QUANTUM CHEMISTRY (2013)
Protein and ligand preparation: parameters, protocols, and influence on virtual screening enrichments
G. Madhavi Sastry et al.
JOURNAL OF COMPUTER-AIDED MOLECULAR DESIGN (2013)
Effects of steroidal aromatase inhibitors on sensitive and resistant breast cancer cells: Aromatase inhibition and autophagy
Cristina Amaral et al.
JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY (2013)
Optimization of the aromatase inhibitory activities of pyridylthiazole analogues of resveratrol
Abdelrahman S. Mayhoub et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2012)
Resveratrol in Medicinal Chemistry: A Critical Review of its Pharmacokinetics, Drug-Delivery, and Membrane Interactions
A. R. Neves et al.
CURRENT MEDICINAL CHEMISTRY (2012)
Fibrate-derived N-(methylsulfonyl)amides with antagonistic properties on PPARα
Alessandra Ammazzalorso et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2012)
Design, synthesis and biological evaluation of 5-hydroxy, 5-substituted-pyrimidine-2,4,6-triones as potent inhibitors of gelatinases MMP-2 and MMP-9
Orazio Nicolotti et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2012)
Transport, stability, and biological activity of resveratrol
Dominique Delmas et al.
RESVERATROL AND HEALTH (2011)
Resveratrol derivatives as promising chemopreventive agents with improved potency and selectivity
Tamara P. Kondratyuk et al.
MOLECULAR NUTRITION & FOOD RESEARCH (2011)
Design, synthesis, and biological evaluation of resveratrol analogues as aromatase and quinone reductase 2 inhibitors for chemoprevention of cancer
Bin Sun et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2010)
Selective Synthesis and Biological Evaluation of Sulfate-Conjugated Resveratrol Metabolites
Juma Hoshino et al.
JOURNAL OF MEDICINAL CHEMISTRY (2010)
The potential adverse effects of aromatase inhibitors on wound healing: in vitro and in vivo evidence
Daniel J. Howgate et al.
EXPERT OPINION ON DRUG SAFETY (2009)
Structural basis for androgen specificity and oestrogen synthesis in human aromatase
Debashis Ghosh et al.
NATURE (2009)
In vivo efficacy of STX213, a second-generation steroid sulfatase inhibitor, for hormone-dependent breast cancer therapy
Paul A. Foster et al.
CLINICAL CANCER RESEARCH (2006)
Importance of accurate charges in molecular docking: Quantum mechanical/molecular mechanical (QM/MM) approach
AE Cho et al.
JOURNAL OF COMPUTATIONAL CHEMISTRY (2005)
Bioisosterism: A useful strategy for molecular modification and drug design
LMA Lima et al.
CURRENT MEDICINAL CHEMISTRY (2005)
High absorption but very low bioavailability of oral resveratrol in humans
T Walle et al.
DRUG METABOLISM AND DISPOSITION (2004)
Apoptosis, chemoresistance, and breast cancer: Insights from the MCF-7 cell model system
R Simstein et al.
EXPERIMENTAL BIOLOGY AND MEDICINE (2003)