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AMERICAN JOURNAL OF CHINESE MEDICINE (2013)
Quercetin-3-O-glucuronide induces ABCA1 expression by LXRα activation in murine macrophages
Kazuaki Ohara et al.
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS (2013)
Knock-down of the oxysterol receptor LXRα impairs cholesterol efflux in human primary macrophages: Lack of compensation by LXRβ activation
Minako Ishibashi et al.
BIOCHEMICAL PHARMACOLOGY (2013)
Natural products: A continuing source of novel drug leads
Gordon M. Cragg et al.
BIOCHIMICA ET BIOPHYSICA ACTA-GENERAL SUBJECTS (2013)
Induction of ABCA1 and ABCG1 expression by the liver X receptor modulator cineole in macrophages
Hee-jin Jun et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2013)
Cyanidin, a natural flavonoid, is an agonistic ligand for liver X receptor alpha and beta and reduces cellular lipid accumulation in macrophages and hepatocytes
Yaoyao Jia et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2013)
Resveratrol mediates anti-atherogenic effects on cholesterol flux in human macrophages and endothelium via PPARγ and adenosine
Iryna Voloshyna et al.
EUROPEAN JOURNAL OF PHARMACOLOGY (2013)
Oxysterol receptors and their therapeutic applications in cancer conditions
Hugues De Boussac et al.
EXPERT OPINION ON THERAPEUTIC TARGETS (2013)
Bioactive phenolics and terpenoids from Manglietia insignis
Shan-Zhai Shang et al.
FITOTERAPIA (2013)
Citrange Fruit Extracts Alleviate Obesity-Associated Metabolic Disorder in High-Fat Diet-Induced Obese C57BL/6 Mouse
Yan Lu et al.
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES (2013)
Paeoniflorin acts as a liver X receptor agonist
Hsiang-Ru Lin
JOURNAL OF ASIAN NATURAL PRODUCTS RESEARCH (2013)
Binding Mechanism of the Farnesoid X Receptor Marine Antagonist Suvanine Reveals a Strategy To Forestall Drug Modulation on Nuclear Receptors. Design, Synthesis, and Biological Evaluation of Novel Ligands
Francesco Saverio Di Leva et al.
JOURNAL OF MEDICINAL CHEMISTRY (2013)
Increased effects of ginsenosides on the expression of cholesterol 7α-hydroxylase but not the bile salt export pump are involved in cholesterol metabolism
Atsushi Kawase et al.
JOURNAL OF NATURAL MEDICINES (2013)
Sesame Oil Accelerates Healing of 2,4,6-Trinitrobenzenesulfonic Acid-Induced Acute Colitis by Attenuating Inflammation and Fibrosis
Srinivasan Periasamy et al.
JOURNAL OF PARENTERAL AND ENTERAL NUTRITION (2013)
Identification of liver X receptor and farnesoid X receptor dual agonists from Tithonia diversifolia
Hsiang-Ru Lin
MEDICINAL CHEMISTRY RESEARCH (2013)
Quercetin up-regulates expressions of peroxisome proliferator-activated receptor γ, liver X receptor α, and ATP binding cassette transporter A1 genes and increases cholesterol efflux in human macrophage cell line
Seung-Min Lee et al.
NUTRITION RESEARCH (2013)
Lucidone from Lindera erythrocarpa Makino fruits suppresses adipogenesis in 3T3-L1 cells and attenuates obesity and consequent metabolic disorders in high-fat diet C57BL/6 mice
Yu-Hsin Hsieh et al.
PHYTOMEDICINE (2013)
Regulation of prostaglandin F2α, against β amyloid clearance and its inflammation induction through LXR/RXR heterodimer antagonism in microglia
Jingjing Zhuang et al.
PROSTAGLANDINS & OTHER LIPID MEDIATORS (2013)
Total synthesis of riccardin C and (±)-cavicularin via Pd-catalyzed Ar-Ar cross couplings
Kenichi Harada et al.
TETRAHEDRON (2013)
Saponins, especially platycodin D, from Platycodon grandiflorum modulate hepatic lipogenesis in high-fat diet-fed rats and high glucose-exposed HepG2 cells
Yong Pil Hwang et al.
TOXICOLOGY AND APPLIED PHARMACOLOGY (2013)
Atherosclerosis: lessons from LXR and the intestine
Barbara Bonamassa et al.
TRENDS IN ENDOCRINOLOGY AND METABOLISM (2013)
Investigation of imatinib and other approved drugs as starting points for antidiabetic drug discovery with FXR modulating activity
Ramona Steri et al.
BIOCHEMICAL PHARMACOLOGY (2012)
Liver X receptor and peroxisome proliferator-activated receptor agonist from Cornus alternifolia
Yang-Qing He et al.
BIOCHIMICA ET BIOPHYSICA ACTA-GENERAL SUBJECTS (2012)
Anti-inflammatory and metabolic actions of FXR: Insights into molecular mechanisms
Danielle A. A. Hollman et al.
BIOCHIMICA ET BIOPHYSICA ACTA-MOLECULAR AND CELL BIOLOGY OF LIPIDS (2012)
Ethyl 2,4,6-trihydroxybenzoate is an agonistic ligand for liver X receptor that induces cholesterol efflux from macrophages without affecting lipid accumulation in HepG2 cells
Minh-Hien Hoang et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2012)
Nelumal A, the active principle from Ligularia nelumbifolia, is a novel farnesoid X receptor agonist
Francesco Epifano et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2012)
Triterpenes from Alisma orientalis act as farnesoid X receptor agonists
Hsiang-Ru Lin
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2012)
Sesquiterpenoids from Atractylodes macrocephala act as farnesoid X receptor and progesterone receptor modulators
Chia-Jui Tsai et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2012)
Iristectorigenin B isolated from Belamcanda chinensis is a liver X receptor modulator that increases ABCA1 and ABCG1 expression in macrophage RAW 264.7 cells
Hee-jin Jun et al.
BIOTECHNOLOGY LETTERS (2012)
Development of FXR, PXR and CAR Agonists and Antagonists for Treatment of Liver Disorders
Stefano Fiorucci et al.
CURRENT TOPICS IN MEDICINAL CHEMISTRY (2012)
Soy protein isoflavones differentially regulate liver X receptor isoforms to modulate lipid metabolism and cholesterol transport in the liver and intestine in mice
M. Gonzalez-Granillo et al.
DIABETOLOGIA (2012)
Cycloartane triterpenoids from the stems of Schisandra glaucescens and their bioactivity
Juan Zou et al.
FITOTERAPIA (2012)
Rhein Protects against Obesity and Related Metabolic Disorders through Liver X Receptor-Mediated Uncoupling Protein 1 Upregulation in Brown Adipose Tissue
Xiaoyan Sheng et al.
INTERNATIONAL JOURNAL OF BIOLOGICAL SCIENCES (2012)
Fucosterol Is a Selective Liver X Receptor Modulator That Regulates the Expression of Key Genes in Cholesterol Homeostasis in Macrophages, Hepatocytes, and Intestinal Cells
Minh-Hien Hoang et al.
JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY (2012)
Panax notoginseng saponins attenuate atherosclerosis via reciprocal regulation of lipid metabolism and inflammation by inducing liver X receptor alpha expression
Ji-Shan Fan et al.
JOURNAL OF ETHNOPHARMACOLOGY (2012)
Conicasterol E, a Small Heterodimer Partner Sparing Farnesoid X Receptor Modulator Endowed with a Pregnane X Receptor Agonistic Activity, from the Marine Sponge Theonella swinhoei
Valentina Sepe et al.
JOURNAL OF MEDICINAL CHEMISTRY (2012)
Hesperetin Upregulates ABCA1 Expression and Promotes Cholesterol Efflux from THP-1 Macrophages
Akio Iio et al.
JOURNAL OF NATURAL PRODUCTS (2012)
Taurine is a liver X receptor-α ligand and activates transcription of key genes in the reverse cholesterol transport without inducing hepatic lipogenesis
Minh-Hien Hoang et al.
MOLECULAR NUTRITION & FOOD RESEARCH (2012)
Transcriptional integration of metabolism by the nuclear sterol-activated receptors LXR and FXR
Anna C. Calkin et al.
NATURE REVIEWS MOLECULAR CELL BIOLOGY (2012)
Ethanolic extracts of Brazilian red propolis increase ABCA1 expression and promote cholesterol efflux from THP-1 macrophages
Akio Iio et al.
PHYTOMEDICINE (2012)
Lanostane Triterpenoids from the Stems of Schisandra glaucescens
Juan Zou et al.
PLANTA MEDICA (2012)
Discovery That Theonellasterol a Marine Sponge Sterol Is a Highly Selective FXR Antagonist That Protects against Liver Injury in Cholestasis
Barbara Renga et al.
PLOS ONE (2012)
Sterols from a soft coral, Dendronephthya gigantea as farnesoid X-activated receptor antagonists
Kyoungjin Shin et al.
STEROIDS (2012)
4-Methylenesterols from Theonella swinhoei sponge are natural pregnane-X-receptor agonists and farnesoid-X-receptor antagonists that modulate innate immunity
Simona De Marino et al.
STEROIDS (2012)
A tea catechin, epigallocatechin-3-gallate, is a unique modulator of the farnesoid X receptor
Guodong Li et al.
TOXICOLOGY AND APPLIED PHARMACOLOGY (2012)
Marine sponge steroids as nuclear receptor ligands
Stefano Fiorucci et al.
TRENDS IN PHARMACOLOGICAL SCIENCES (2012)
Liver X receptor biology and pharmacology: new pathways, challenges and opportunities
Tomas Jakobsson et al.
TRENDS IN PHARMACOLOGICAL SCIENCES (2012)
Rhein ameliorates fatty liver disease through negative energy balance, hepatic lipogenic regulation, and immunomodulation in diet-induced obese mice
Xiaoyan Sheng et al.
AMERICAN JOURNAL OF PHYSIOLOGY-ENDOCRINOLOGY AND METABOLISM (2011)
Nuclear bile acid receptor FXR in the hepatic regeneration
Wei-Dong Chen et al.
BIOCHIMICA ET BIOPHYSICA ACTA-MOLECULAR BASIS OF DISEASE (2011)
Pharmacophore-based discovery of FXR-agonists. Part II: Identification of bioactive triterpenes from Ganoderma lucidum
Ulrike Grienke et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2011)
Growth inhibitory activities of oxyprenylated and non-prenylated naturally occurring phenylpropanoids in cancer cell lines
Celine Bruyere et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2011)
Oxepinamides: Novel Liver X Receptor Agonists from Aspergillus puniceus
Xin-Hua Lu et al.
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY (2011)
Theonellasterols and Conicasterols from Theonella swinhoei. Novel Marine Natural Ligands for Human Nuclear Receptors
Simona De Marino et al.
JOURNAL OF MEDICINAL CHEMISTRY (2011)
Discovery of Sulfated Sterols from Marine Invertebrates as a New Class of Marine Natural Antagonists of Farnesoid-X-Receptor
Valentina Sepe et al.
JOURNAL OF MEDICINAL CHEMISTRY (2011)
Tuberatolides, Potent FXR Antagonists from the Korean Marine Tunicate Botryllus tuberatus
Hyukjae Choi et al.
JOURNAL OF NATURAL PRODUCTS (2011)
Diosgenin, the Main Aglycon of Fenugreek, Inhibits LXR alpha Activity in HepG2 Cells and Decreases Plasma and Hepatic Triglycerides in Obese Diabetic Mice
Taku Uemura et al.
JOURNAL OF NUTRITION (2011)
ATP binding cassette transporter G1 (ABCG1) is an intracellular sterol transporter
Elizabeth J. Tarling et al.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2011)
Labdane diterpenes protect against anoxia/reperfusion injury in cardiomyocytes: involvement of AKT activation
I. Cuadrado et al.
CELL DEATH & DISEASE (2011)
Honokiol Increases ABCA1 Expression Level by Activating Retinoid X Receptor Beta
Cha-Gyun Jung et al.
BIOLOGICAL & PHARMACEUTICAL BULLETIN (2010)
Inhibition of liver X receptor-α-dependent hepatic steatosis by isoliquiritigenin, a licorice antioxidant flavonoid, as mediated by JNK1 inhibition
Young Mi Kim et al.
FREE RADICAL BIOLOGY AND MEDICINE (2010)
Inhibition of SREBP-1c-mediated hepatic steatosis and oxidative stress by sauchinone, an AMPK-activating lignan in Saururus chinensis
Young Woo Kim et al.
FREE RADICAL BIOLOGY AND MEDICINE (2010)
Panax notoginseng saponins decrease cholesterol ester via up-regulating ATP-binding cassette transporter Al in foam cells
Yi Jia et al.
JOURNAL OF ETHNOPHARMACOLOGY (2010)
Structure-Activity Relationship Study of Betulinic Acid, A Novel and Selective TGR5 Agonist, and Its Synthetic Derivatives: Potential Impact in Diabetes
Cedric Genet et al.
JOURNAL OF MEDICINAL CHEMISTRY (2010)
X-Ray Structures of the LXRα LBD in Its Homodimeric Form and Implications for Heterodimer Signaling
Xavier Fradera et al.
JOURNAL OF MOLECULAR BIOLOGY (2010)
Dammarane-type saponins from Gynostemma pentaphyllum
Pham Thanh Ky et al.
PHYTOCHEMISTRY (2010)
Oleanolic Acid is a Selective Farnesoid X Receptor Modulator
Wenming Liu et al.
PHYTOTHERAPY RESEARCH (2010)
Transcriptional Regulation of Human and Rat Hepatic Lipid Metabolism by the Grapefruit Flavonoid Naringenin: Role of PPARα, PPARγ and LXRα
Jonathan Goldwasser et al.
PLOS ONE (2010)
Lipid ligand-activated transcription factors regulating lipid storage and release in human macrophages
G. Chinetti-Gbaguidi et al.
BIOCHIMICA ET BIOPHYSICA ACTA-MOLECULAR AND CELL BIOLOGY OF LIPIDS (2009)
Effect of Guggulsterone and Cembranoids of Commiphora mukul on Pancreatic Phospholipase A(2): Role in Hypocholesterolemia
Bao-Zhu Yu et al.
JOURNAL OF NATURAL PRODUCTS (2009)
Minireview: Evolution of NURSA, the Nuclear Receptor Signaling Atlas
Neil J. McKenna et al.
MOLECULAR ENDOCRINOLOGY (2009)
Dietary procyanidins enhance transcriptional activity of bile acid-activated FXR in vitro and reduce triglyceridemia in vivo in a FXR-dependent manner
Josep Maria Del Bas et al.
MOLECULAR NUTRITION & FOOD RESEARCH (2009)
Isorhamnetin Represses Adipogenesis in 3T3-L1 Cells
Jongsung Lee et al.
OBESITY (2009)
Role of Bile Acids and Bile Acid Receptors in Metabolic Regulation
Philippe Lefebvre et al.
PHYSIOLOGICAL REVIEWS (2009)
Effects of coumestrol on lipid and glucose metabolism as a farnesoid X receptor ligand
Miki Takahashi et al.
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS (2008)
Liver X Receptors (LXR) as Therapeutic Targets in Dyslipidemia
Jerzy Beltowski
CARDIOVASCULAR THERAPEUTICS (2008)
Coordination of inflammation and metabolism by PPAR and LXR nuclear receptors
Cynthia Hong et al.
CURRENT OPINION IN GENETICS & DEVELOPMENT (2008)
Recent advances in Liver X Receptor biology and chemistry
Bryan J. Goodwin et al.
CURRENT TOPICS IN MEDICINAL CHEMISTRY (2008)
Brazilian Red PropolisChemical Composition and Botanical Origin
Andreas Daugsch et al.
EVIDENCE-BASED COMPLEMENTARY AND ALTERNATIVE MEDICINE (2008)
Hypolipidemic activity and mechanism of purified herbal extract of Salvia miltiorrhiza in hyperlipidemic rats
W. Ji et al.
JOURNAL OF ETHNOPHARMACOLOGY (2008)
The novel compounds that activate farnesoid X receptor: The diversity of their effects on gene expression
Takuo Suzuki et al.
JOURNAL OF PHARMACOLOGICAL SCIENCES (2008)
Identification of a potent synthetic FXR agonist with an unexpected mode of binding and activation
Stephen M. Soisson et al.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2008)
Scalarane sesterterpenes from a marine sponge of the genus spongia and their FXR antagonistic activity
Sang-Jip Nam et al.
JOURNAL OF NATURAL PRODUCTS (2007)
Nuclear receptor coregulators: Judges, juries, and executioners of cellular regulation
David M. Lonard et al.
MOLECULAR CELL (2007)
Hypolipidemic effects and mechanisms of Panax notoginseng on lipid profile in hyperlipidemic rats
W. Ji et al.
JOURNAL OF ETHNOPHARMACOLOGY (2007)
Stigmasterol, a soy lipid-derived phytosterol, is an antagonist of the bile acid nuclear receptor FXR
Beth A. Carter et al.
PEDIATRIC RESEARCH (2007)
Ligand activation of LXRβ reverses atherosclerosis and cellular cholesterol overload in mice lacking LXRα and apoE
Michelle N. Bradley et al.
JOURNAL OF CLINICAL INVESTIGATION (2007)
Phytochemicals of black bean seed coats: Isolation, structure elucidation, and their antiproliferative and antioxidative activities
Mei Dong et al.
JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY (2007)
The cholesterol-raising factor from coffee beans, cafestol, as an agonist ligand for the farnesoid and pregnane X receptors
Marie-Louise Ricketts et al.
MOLECULAR ENDOCRINOLOGY (2007)
Selective activation of liver X receptors by acanthoic acid-related diterpenes
Paqui G. Traves et al.
MOLECULAR PHARMACOLOGY (2007)
Farnesoid X-activated receptor antagonists from a marine sponge Spongia sp.
Sang-Jip Nam et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2006)
Resveratrol regulates the expression of LXR-α in human macrophages
Marie Sevov et al.
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS (2006)
Lipid efflux by the ATP-binding cassette transporters ABCA1 and ABCG1
Clara Cavelier et al.
BIOCHIMICA ET BIOPHYSICA ACTA-MOLECULAR AND CELL BIOLOGY OF LIPIDS (2006)
Screening of novel nuclear receptor agonists by a convenient reporter gene assay system using green fluorescent protein derivatives
T. Suzuki et al.
PHYTOMEDICINE (2006)
Cholesterol-lowering effect of platycodin D in hypercholesterolemic ICR mice
Hai Lin Zhao et al.
EUROPEAN JOURNAL OF PHARMACOLOGY (2006)
The role of pharmacognosy in modern medicine and pharmacy
WP Jones et al.
CURRENT DRUG TARGETS (2006)
Niemann-Pick C1 like 1 gene expression is down-regulated by LXR activators in the intestine
C Duval et al.
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS (2006)
Xanthohumol, the chalcone from beer hops (Humulus lupulus L.), is the ligand for farnesoid X receptor and ameliorates lipid and glucose metabolism in KK-Ay mice
H Nozawa
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS (2005)
Riccardin C:: A natural product that functions as a liver X receptor (LXR)α agonist and an LXRβ antagonist
N Tamehiro et al.
FEBS LETTERS (2005)
Fibroblast growth factor 15 functions as an enterohepatic signal to regulate bile acid homeostasis
T Inagaki et al.
CELL METABOLISM (2005)
Steroidal and triterpenoidal fungal metabolites as ligands of liver X receptors
JG Ondeyka et al.
JOURNAL OF ANTIBIOTICS (2005)
Anthrabenzoxocinones from Streptomyces sp as liver X receptor ligands and antibacterial agents
KB Herath et al.
JOURNAL OF NATURAL PRODUCTS (2005)
Discovery and development of dimeric podocarpic acid leads as potent agonists of liver X receptor with HDL cholesterol raising activity in mice and hamsters
SB Singh et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2005)
The evolving role of natural products in drug discovery
FE Koehn et al.
NATURE REVIEWS DRUG DISCOVERY (2005)
Genomic analysis of the nuclear receptor family: New insights into structure, regulation, and evolution from the rat genome
ZD Zhang et al.
GENOME RESEARCH (2004)
Polyunsaturated fatty acids are FXR ligands and differentially regulate expression of FXR targets
A Zhao et al.
DNA AND CELL BIOLOGY (2004)
Principles for modulation of the nuclear receptor superfamily
H Gronemeyer et al.
NATURE REVIEWS DRUG DISCOVERY (2004)
A natural product ligand of the oxysterol receptor, liver X receptor
KS Bramlett et al.
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS (2003)
Crystal structure of the heterodimeric complex of LXRα and RXRβ ligand-binding domains in a fully agonistic conformation
S Svensson et al.
EMBO JOURNAL (2003)
Evolution of secondary metabolites from an ecological and molecular phylogenetic perspective
M Wink
PHYTOCHEMISTRY (2003)
X-ray crystal structure of the liver X receptor β ligand binding domain -: Regulation by a histidine-tryptophan switch
S Williams et al.
JOURNAL OF BIOLOGICAL CHEMISTRY (2003)
Stimulation of cholesterol excretion by the liver X receptor agonist requires ATP-binding cassette transporters G5 and G8
LQ Yu et al.
JOURNAL OF BIOLOGICAL CHEMISTRY (2003)
Structural basis for bile acid binding and activation of the nuclear receptor FXR
LZ Mi et al.
MOLECULAR CELL (2003)
Liver X receptor-dependent repression of matrix metalloproteinase-9 expression in macrophages
A Castrillo et al.
JOURNAL OF BIOLOGICAL CHEMISTRY (2003)
The farnesoid X-receptor is an essential regulator of cholesterol homeostasis
G Lambert et al.
JOURNAL OF BIOLOGICAL CHEMISTRY (2003)
Antidiabetic action of a liver X receptor agonist mediated by inhibition of hepatic gluconeogenesis
GQ Cao et al.
JOURNAL OF BIOLOGICAL CHEMISTRY (2003)
A natural product that lowers cholesterol as an antagonist ligand for FXR
NL Urizar et al.
SCIENCE (2002)
Polyunsaturated fatty acids suppress sterol regulatory element-binding protein 1c promoter activity by inhibition of liver X receptor (LXR) binding to LXR response elements
T Yoshikawa et al.
JOURNAL OF BIOLOGICAL CHEMISTRY (2002)
Orphan nuclear receptors as eLiXiRs and FiXeRs of sterol metabolism
TT Lu et al.
JOURNAL OF BIOLOGICAL CHEMISTRY (2001)
The negative effects of bile acids and tumor necrosis factor-α on the transcription of cholesterol 7α-hydroxylase gene (CYP7A1) converge to hepatic nuclear factor-4 -: A novel mechanism of feedback regulation of bile acid synthesis mediated by nuclear receptors
E De Fabiani et al.
JOURNAL OF BIOLOGICAL CHEMISTRY (2001)
Unsaturated fatty acids inhibit transcription of the sterol regulatory element-binding protein-1c (SREBP-1c) gene by antagonizing ligand-dependent activation of the LXR
JF Ou et al.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2001)
The nuclear receptors FXR and LXRα:: Potential targets for the development of drugs affecting lipid metabolism and neoplastic diseases
EJ Niesor et al.
CURRENT PHARMACEUTICAL DESIGN (2001)
Targeted disruption of the nuclear receptor FXR/BAR impairs bile acid and lipid homeostasis
CJ Sinal et al.
CELL (2000)
Oxysterols: Modulators of cholesterol metabolism and other processes
GJ Schroepfer
PHYSIOLOGICAL REVIEWS (2000)
Regulation of absorption and ABC1-mediated efflux of cholesterol by RXR heterodimers
JJ Repa et al.
SCIENCE (2000)