期刊
JOURNAL OF ORGANIC CHEMISTRY
卷 87, 期 2, 页码 1335-1347出版社
AMER CHEMICAL SOC
DOI: 10.1021/acs.joc.1c02644
关键词
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资金
- National Natural Science Foundation of China [22001197]
- Foundation of Guangdong Basic and Applied Basic Research [2019A1515110516, 2019A1515110266]
- Foundation for Young Talents [2019KQNCX159, 2019KQNCX160]
- Foundation of the Department of Education of Guangdong Province [2019KZDXM052, 2021KTSCX140]
- National College Students Innovation and Entrepreneurship Training Program [202111349169]
An efficient anodic C(sp(3))-H acyloxylation protocol has been developed, which enables the direct oxidation of indolin-3-ones to obtain various C2-acyloxy indolin-3-ones without the need for metal catalysts and external oxidants. The practicality of this protocol has been demonstrated through the effective application of several medical drugs and gram-scale experiments.
An efficient anodic C(sp(3))-H acyloxylation protocol has been established via intermolecular cross-dehydrogenative C(sp(3))-O coupling. The protocol provides various C2-acyloxy indolin-3-ones without the addition of metal catalysts and external oxidants because indolin-3-ones can be directly oxidized at the anode. The effective application of several medical drugs and the realization of the gram-scale experiment have proven the practicality of this protocol.
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