4.7 Article

Improving the dissolution behaviors and bioavailability of abiraterone acetate via multicomponent crystal forms

相关参考文献

注意:仅列出部分参考文献,下载原文获取全部文献信息。
Article Pharmacology & Pharmacy

Cocrystals to tune oily vitamin E into crystal vitamin E

Bingqing Zhu et al.

Summary: This study introduces a more effective method to stabilize and solidify d-alpha-tocopherol oil through cocrystallization, increasing its stability and transforming it into solid form.

INTERNATIONAL JOURNAL OF PHARMACEUTICS (2021)

Article Pharmacology & Pharmacy

Understanding solid-state processing of pharmaceutical cocrystals via milling: Role of tablet excipients

Rahamatullah Shaikh et al.

Summary: Research on novel cocrystal systems and their physicochemical properties improvement is prevalent, yet the focus on final product formulation is lacking. This study measured the impact of tablet excipients on pharmaceutical cocrystal formulations, supported by Density Functional Theory calculations of intermolecular binding energies. The presence of certain excipients, such as PEG, HPMC, or lactose, was found to yield purer cocrystals during co-milling.

INTERNATIONAL JOURNAL OF PHARMACEUTICS (2021)

Article Pharmacology & Pharmacy

Crystal structures, dissolution and pharmacokinetic study on a novel phosphodiesterase-4 inhibitor chlorbipram cocrystals

Jianle Zhou et al.

INTERNATIONAL JOURNAL OF PHARMACEUTICS (2020)

Review Pharmacology & Pharmacy

Oral formulation strategies to improve the bioavailability and mitigate the food effect of abiraterone acetate

Hayley B. Schultz et al.

INTERNATIONAL JOURNAL OF PHARMACEUTICS (2020)

Article Medicine, Research & Experimental

Ketoconazole-p-aminobenzoic Acid Cocrystal: Revival of an Old Drug by Crystal Engineering

Flavia Martin et al.

MOLECULAR PHARMACEUTICS (2020)

Article Pharmacology & Pharmacy

Enhancement of abiraterone acetate oral bioavailability by supersaturated-silica lipid hybrids

Hayley B. Schultz et al.

INTERNATIONAL JOURNAL OF PHARMACEUTICS (2020)

Article Chemistry, Multidisciplinary

Improving Solubility of Poorly Soluble Abiraterone Acetate by Cocrystal Design Aided by In Silico Screening

Ramanaiah Chennuru et al.

CRYSTAL GROWTH & DESIGN (2020)

Article Chemistry, Multidisciplinary

Machine-Learning-Guided Cocrystal Prediction Based on Large Data Base

Dingyan Wang et al.

CRYSTAL GROWTH & DESIGN (2020)

Article Pharmacology & Pharmacy

Exploring potential coformers for oxyresveratrol using principal component analysis

Passaporn Ouiyangkul et al.

INTERNATIONAL JOURNAL OF PHARMACEUTICS (2020)

Article Medicine, Research & Experimental

Drug-Drug Binary Solids of Nitrofurantoin and Trimethoprim: Crystal Engineering and Pharmaceutical Properties

Dilip Kumar Maity et al.

MOLECULAR PHARMACEUTICS (2020)

Review Pharmacology & Pharmacy

Food for thought: formulating away the food effect - a PEARRL review

Joseph P. O'Shea et al.

JOURNAL OF PHARMACY AND PHARMACOLOGY (2019)

Article Pharmacology & Pharmacy

Effect of gel formation on the dissolution behavior of clarithromycin tablets

Koki Inukai et al.

INTERNATIONAL JOURNAL OF PHARMACEUTICS (2017)

Article Chemistry, Multidisciplinary

The Plot Thickens: Gelation by Phenylalanine in Water and Dimethyl Sulfoxide

Karol P. Nartowski et al.

CRYSTAL GROWTH & DESIGN (2017)

Article Chemistry, Multidisciplinary

Cocrystals of Baicalein with Higher Solubility and Enhanced Bioavailability

Bingqing Zhu et al.

CRYSTAL GROWTH & DESIGN (2017)

Article Chemistry, Multidisciplinary

Impact of the Dissolution Profile of the Cilostazol Cocrystal with Supersaturation on the Oral Bioavailability

Motoyasu Yoshimura et al.

CRYSTAL GROWTH & DESIGN (2017)

Article Chemistry, Medicinal

The Effect of Food on the Intraluminal Behavior of Abiraterone Acetate in Man

Sophie Geboers et al.

JOURNAL OF PHARMACEUTICAL SCIENCES (2016)

Article Pharmacology & Pharmacy

Aerosil as a novel co-crystal co-former for improving the dissolution rate of hydrochlorothiazide

Sanaa A. El-Gizawy et al.

INTERNATIONAL JOURNAL OF PHARMACEUTICS (2015)

Article Chemistry, Multidisciplinary

Crystal structure refinement with SHELXL

George M. Sheldrick

ACTA CRYSTALLOGRAPHICA SECTION C-STRUCTURAL CHEMISTRY (2015)

Article Chemistry, Multidisciplinary

Polymorphs, Salts, and Cocrystals: What's in a Name?

Srinivasulu Aitipamula et al.

CRYSTAL GROWTH & DESIGN (2012)

Article Chemistry, Multidisciplinary

Solid-state vibrational spectroscopic investigation of cocrystals and salt of indomethacin

Hassan Refat H. Ali et al.

CRYSTENGCOMM (2012)

Article Chemistry, Multidisciplinary

Acid-base crystalline complexes and the pKa rule

Aurora J. Cruz-Cabeza

CRYSTENGCOMM (2012)

Article Chemistry, Multidisciplinary

Vibrational Spectroscopic Studies of Cocrystals and Salts. 2. The Benzylamine-Benzoic Acid System

Harry G. Brittain

CRYSTAL GROWTH & DESIGN (2009)

Article Pharmacology & Pharmacy

Biopharmaceutical classification of drugs using intrinsic dissolution rate (IDR) and rat intestinal permeability

Parvin Zakeri-Milani et al.

EUROPEAN JOURNAL OF PHARMACEUTICS AND BIOPHARMACEUTICS (2009)

Article Chemistry, Multidisciplinary

Mercury CSD 2.0 -: new features for the visualization and investigation of crystal structures

Clare F. Macrae et al.

JOURNAL OF APPLIED CRYSTALLOGRAPHY (2008)

Article Chemistry, Medicinal

Synthesis, biological evaluation, and molecular modeling of abiraterone analogues: Novel CYP17 inhibitors for the treatment of prostate cancer

Mariano A. E. Pinto-Bazurco Mendieta et al.

JOURNAL OF MEDICINAL CHEMISTRY (2008)

Article Medicine, Research & Experimental

Screening for pharmaceutical cocrystal hydrates via neat and liquid-assisted grinding

Shyam Karki et al.

MOLECULAR PHARMACEUTICS (2007)

Article Medicine, Research & Experimental

The salt-cocrystal continuum: The influence of crystal structure on ionization state

Scott L. Childs et al.

MOLECULAR PHARMACEUTICS (2007)