相关参考文献
注意:仅列出部分参考文献,下载原文获取全部文献信息。Protein degradation through covalent inhibitor-based PROTACs
Gang Xue et al.
CHEMICAL COMMUNICATIONS (2020)
Functional rare and low frequency variants in BLK and BANK1 contribute to human lupus
Simon H. Jiang et al.
NATURE COMMUNICATIONS (2019)
A multiprotein supercomplex controlling oncogenic signalling in lymphoma
James D. Phelan et al.
NATURE (2018)
Analysis of KLF4 regulated genes in cancer cells reveals a role of DNA methylation in promoter-enhancer interactions
Olutobi Oyinlade et al.
EPIGENETICS (2018)
Ibrutinib inhibits pre-BCR+ B-cell acute lymphoblastic leukemia progression by targeting BTK and BLK
Ekaterina Kim et al.
BLOOD (2017)
Concordance of Increased B1 Cell Subset and Lupus Phenotypes in Mice and Humans Is Dependent on BLK Expression Levels
Ying-Yu Wu et al.
JOURNAL OF IMMUNOLOGY (2015)
The ins and outs of selective kinase inhibitor development
Susanne Mueller et al.
NATURE CHEMICAL BIOLOGY (2015)
A novel 2,5-diaminopyrimidine-based affinity probe for Bruton's tyrosine kinase
Yingying Zuo et al.
SCIENTIFIC REPORTS (2015)
Autoimmune Disease-Associated Haplotypes of BLK Exhibit Lowered Thresholds for B Cell Activation and Expansion of Ig Class-Switched B Cells
Kim R. Simpfendorfer et al.
ARTHRITIS & RHEUMATOLOGY (2015)
Discovery of a Series of 2,5-Diaminopyrimidine Covalent Irreversible Inhibitors of Bruton's Tyrosine Kinase with in Vivo Antitumor Activity
Xitao Li et al.
JOURNAL OF MEDICINAL CHEMISTRY (2014)
OPEN B-lymphoid tyrosine kinase (Blk) is an oncogene and a potential target for therapy with dasatinib in cutaneous T-cell lymphoma (CTCL)
D. L. Petersen et al.
LEUKEMIA (2014)
Reduced B Lymphoid Kinase (Blk) Expression Enhances Proinflammatory Cytokine Production and Induces Nephrosis in C57BL/6-lpr/lpr Mice
Elizabeth M. Samuelson et al.
PLOS ONE (2014)
Developing Irreversible Inhibitors of the Protein Kinase Cysteinome
Qingsong Liu et al.
CHEMISTRY & BIOLOGY (2013)
Blk haploinsufficiency impairs the development, but enhances the functional responses, of MZ B cells
Elizabeth M. Samuelson et al.
IMMUNOLOGY AND CELL BIOLOGY (2012)
Specific Btk inhibition suppresses B cell- and myeloid cell-mediated arthritis
Julie A. Di Paolo et al.
NATURE CHEMICAL BIOLOGY (2011)
Unexpected Role for the B Cell-Specific Src Family Kinase B Lymphoid Kinase in the Development of IL-17-Producing γδ T Cells
Renee M. Laird et al.
JOURNAL OF IMMUNOLOGY (2010)
Through the Gatekeeper Door: Exploiting the Active Kinase Conformation
Fabio Zuccotto et al.
JOURNAL OF MEDICINAL CHEMISTRY (2010)
Ectopic expression of B-lymphoid kinase in cutaneous T-cell lymphoma
Thorbjorn Krejsgaard et al.
BLOOD (2009)
Discovery of selective irreversible inhibitors for Bruton's tyrosine kinase
Zhengying Pan et al.
CHEMMEDCHEM (2007)
Essential role of Src-family protein tyrosine kinases in NF-κB activation during B cell development
K Saijo et al.
NATURE IMMUNOLOGY (2003)
The B-cell-specific src-family kinase Blk is dispensable for B-cell development and activation
G Texido et al.
MOLECULAR AND CELLULAR BIOLOGY (2000)