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Serena Veschi et al.
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Alexander J. Nielsen et al.
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Alexander J. Nielsen et al.
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Letizia Giampietro et al.
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Barbara De Filippis et al.
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Farhan A. Khan et al.
CURRENT ORGANIC CHEMISTRY (2018)
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Ratchanok Pingaew et al.
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Olivia L. Tseng et al.
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Cardiotoxicity of aromatase inhibitors and tamoxifen in postmenopausal women with breast cancer: a systematic review and meta-analysis of randomized controlled trials
F. Khosrow-Khavar et al.
ANNALS OF ONCOLOGY (2017)
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Mostafa M. Ghorab et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2017)
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Alessandra Ammazzalorso et al.
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Barbara De Filippis et al.
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Edward Harder et al.
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Mauro Di Matteo et al.
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Mostafa M. Ghorab et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2016)
Recent Progress in the Discovery of Next Generation Inhibitors of Aromatase from the Structure-Function Perspective
Debashis Ghosh et al.
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Structural and functional characterization of aromatase, estrogen receptor, and their genes in endocrine-responsive and -resistant breast cancer cells
Hei Jason Chan et al.
JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY (2016)
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Jennifer Blakemore et al.
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Ratchanok Pingaew et al.
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The MM/PBSA and MM/GBSA methods to estimate ligand-binding affinities
Samuel Genheden et al.
EXPERT OPINION ON DRUG DISCOVERY (2015)
Steroidal aromatase inhibitors inhibit growth of hormone-dependent breast cancer cells by inducing cell cycle arrest and apoptosis
Cristina Amaral et al.
APOPTOSIS (2013)
Protein and ligand preparation: parameters, protocols, and influence on virtual screening enrichments
G. Madhavi Sastry et al.
JOURNAL OF COMPUTER-AIDED MOLECULAR DESIGN (2013)
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Fabiana Caporuscio et al.
JOURNAL OF MEDICINAL CHEMISTRY (2011)
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Tamara P. Kondratyuk et al.
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The VSGB 2.0 model: A next generation energy model for high resolution protein structure modeling
Jianing Li et al.
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Bin Sun et al.
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Debashis Ghosh et al.
NATURE (2009)
Novel procedure for modeling ligand/receptor induced fit effects
W Sherman et al.
JOURNAL OF MEDICINAL CHEMISTRY (2006)
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RW Brueggemeier et al.
ENDOCRINE REVIEWS (2005)
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LMA Lima et al.
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RA Friesner et al.
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Apoptosis, chemoresistance, and breast cancer: Insights from the MCF-7 cell model system
R Simstein et al.
EXPERIMENTAL BIOLOGY AND MEDICINE (2003)
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