4.5 Article

Cyclic Tetrapeptide HDAC Inhibitors with Improved Plasmodium falciparum Selectivity and Killing Profile

相关参考文献

注意:仅列出部分参考文献,下载原文获取全部文献信息。
Article Chemistry, Medicinal

Antiplasmodial Compounds from Deep-Water Marine Invertebrates

Amy E. Wright et al.

Summary: Novel diterpene bebrycin A and known terpene nitenin showed potent antiplasmodial effects against chloroquine-resistant Plasmodium falciparum strain Dd2, with different mechanisms of action at different stages of the intraerythrocytic life cycle of the parasite.

MARINE DRUGS (2021)

Article Multidisciplinary Sciences

Epigenetic inhibitors target multiple stages of Plasmodium falciparum parasites

Nanika Coetzee et al.

SCIENTIFIC REPORTS (2020)

Article Biochemistry & Molecular Biology

Immunofluorescence staining protocol for STED nanoscopy of Plasmodium-infected red blood cells

Ann-Kathrin Mehnert et al.

MOLECULAR AND BIOCHEMICAL PARASITOLOGY (2019)

Article Parasitology

Effect of clinically approved HDAC inhibitors on Plasmodium, Leishmania and Schistosoma parasite growth

Ming Jang Chua et al.

INTERNATIONAL JOURNAL FOR PARASITOLOGY-DRUGS AND DRUG RESISTANCE (2017)

Article Biochemistry & Molecular Biology

Binding of the Microbial Cyclic Tetrapeptide Trapoxin A to the Class I Histone Deacetylase HDAC8

Nicholas J. Porter et al.

ACS CHEMICAL BIOLOGY (2017)

Article Microbiology

Metabolomic Profiling of the Malaria Box Reveals Antimalarial Target Pathways

Erik L. Allman et al.

ANTIMICROBIAL AGENTS AND CHEMOTHERAPY (2016)

Article Biochemistry & Molecular Biology

Histone deacetylase 6 structure and molecular basis of catalysis and inhibition

Yang Hai et al.

NATURE CHEMICAL BIOLOGY (2016)

Article Chemistry, Medicinal

Hydroxamic acid based histone deacetylase inhibitors with confirmed activity against the malaria parasite

Giuseppe Giannini et al.

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2015)

Article Biochemical Research Methods

Homology modeling of parasite histone deacetylases to guide the structure-based design of selective inhibitors

Jelena Melesina et al.

JOURNAL OF MOLECULAR GRAPHICS & MODELLING (2015)

Review Chemistry, Medicinal

An Overview of Naturally Occurring Histone Deacetylase Inhibitors

Bumki Kim et al.

CURRENT TOPICS IN MEDICINAL CHEMISTRY (2014)

Article Biotechnology & Applied Microbiology

Epigenetic regulation of the Plasmodium falciparum genome

Michael F. Duffy et al.

BRIEFINGS IN FUNCTIONAL GENOMICS (2014)

Article Chemistry, Medicinal

Discovery of HDAC inhibitors with potent activity against multiple malaria parasite life cycle stages

Finn K. Hansen et al.

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2014)

Article Biochemistry & Molecular Biology

Protein and ligand preparation: parameters, protocols, and influence on virtual screening enrichments

G. Madhavi Sastry et al.

JOURNAL OF COMPUTER-AIDED MOLECULAR DESIGN (2013)

Article Chemistry, Medicinal

Discovery of HDAC Inhibitors That Lack an Active Site Zn2+-Binding Functional Group

Chris J. Vickers et al.

ACS MEDICINAL CHEMISTRY LETTERS (2012)

Article Biotechnology & Applied Microbiology

Chemoproteomics profiling of HDAC inhibitors reveals selective targeting of HDAC complexes

Marcus Bantscheff et al.

NATURE BIOTECHNOLOGY (2011)

Article Biotechnology & Applied Microbiology

AS1387392, a novel immunosuppressive cyclic tetrapeptide compound with inhibitory activity against mammalian histone deacetylase

Satoshi Sasamura et al.

JOURNAL OF ANTIBIOTICS (2010)

Article Multidisciplinary Sciences

A Moonlighting Function of Plasmodium falciparum Histone 3, Mono-Methylated at Lysine 9?

Yen-Hoon Luah et al.

PLOS ONE (2010)

Article Immunology

Drug inhibition of HDAC3 and epigenetic control of differentiation in Apicomplexa parasites

Alexandre Bougdour et al.

JOURNAL OF EXPERIMENTAL MEDICINE (2009)

Article Cell Biology

Active genes at the nuclear pore complex

Angela Taddei

CURRENT OPINION IN CELL BIOLOGY (2007)

Article Parasitology

Anti-malarial effect of histone deacetylation inhibitors and mammalian tumour cytodifferentiating agents

KT Andrews et al.

INTERNATIONAL JOURNAL FOR PARASITOLOGY (2000)