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PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2013)
Multiple Modes of α7 nAChR Noncompetitive Antagonism of Control Agonist-Evoked and Allosterically Enhanced Currents
Can Peng et al.
MOLECULAR PHARMACOLOGY (2013)
Short-Term Tropisetron Treatment and Cognitive and P50 Auditory Gating Deficits in Schizophrenia
Xiang Yang Zhang et al.
AMERICAN JOURNAL OF PSYCHIATRY (2012)
The discovery of 2-fluoro-N-(3-fluoro-4-(5-((4-morpholinobutyl)amino)-1,3,4-oxadiazol-2-yl)phenyl)benzamide, a full agonist of the alpha-7 nicotinic acetylcholine receptor showing efficacy in the novel object recognition model of cognition enhancement
John Skidmore et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2012)
Consequences of linker length alteration of the α7 nicotinic acetylcholine receptor (nAChR) agonist, SEN12333
Corinne Beinat et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2012)
A New Era for the α7-nAChR
Patrizia Russo et al.
CURRENT DRUG TARGETS (2012)
N-[5-(5-Fluoropyridin-3-yl)-1H-pyrazol-3-yl]-4-piperidin-1-ylbutyramide (SEN78702, WYE-308775): A Medicinal Chemistry Effort toward an α7 Nicotinic Acetylcholine Receptor Agonist Preclinical Candidate
Riccardo Zanaletti et al.
JOURNAL OF MEDICINAL CHEMISTRY (2012)
Discovery of a Novel Alpha-7 Nicotinic Acetylcholine Receptor Agonist Series and Characterization of the Potent, Selective, and Orally Efficacious Agonist 5-(4-Acetyl[1,4]diazepan-1-yl)pentanoic Acid [5-(4-Methoxyphenyl)-1H-pyrazol-3-yl] Amide (SEN15924, WAY-361789)
Riccardo Zanaletti et al.
JOURNAL OF MEDICINAL CHEMISTRY (2012)
Type I and II positive allosteric modulators differentially modulate agonist-induced up-regulation of a7 nicotinic acetylcholine receptors
Morten S. Thomsen et al.
JOURNAL OF NEUROCHEMISTRY (2012)
EVP-6124, a novel and selective α7 nicotinic acetylcholine receptor partial agonist, improves memory performance by potentiating the acetylcholine response of α7 nicotinic acetylcholine receptors
Jos Prickaerts et al.
NEUROPHARMACOLOGY (2012)
Treatment of Tobacco Dependence in People With Mental Health and Addictive Disorders
Kristen M. Mackowick et al.
CURRENT PSYCHIATRY REPORTS (2012)
The expression of nicotinic receptor alpha7 during cochlear development
Scott W. Rogers et al.
BRAIN AND BEHAVIOR (2012)
Synthesis of Selective Agonists for the α7 Nicotinic Acetylcholine Receptor with In Situ Click-Chemistry on Acetylcholine-Binding Protein Templates
John G. Yamauchi et al.
MOLECULAR PHARMACOLOGY (2012)
Activation of α7 Nicotinic Receptors by Orthosteric and Allosteric Agonists: Influence on Single-Channel Kinetics and Conductance
Magda M. Palczynska et al.
MOLECULAR PHARMACOLOGY (2012)
Intrinsically Low Open Probability of α7 Nicotinic Acetylcholine Receptors Can Be Overcome by Positive Allosteric Modulation and Serum Factors Leading to the Generation of Excitotoxic Currents at Physiological Temperatures
Dustin K. Williams et al.
MOLECULAR PHARMACOLOGY (2012)
A Series of α7 Nicotinic Acetylcholine Receptor Allosteric Modulators with Close Chemical Similarity but Diverse Pharmacological Properties
JasKiran K. Gill et al.
MOLECULAR PHARMACOLOGY (2012)
Functional Impact of Allosteric Agonist Activity of Selective Positive Allosteric Modulators of Metabotropic Glutamate Receptor Subtype 5 in Regulating Central Nervous System Function
Meredith J. Noetzel et al.
MOLECULAR PHARMACOLOGY (2012)
Positive allosteric modulators as an approach to nicotinic acetylcholine receptor-targeted therapeutics: Advantages and limitations
Dustin K. Williams et al.
BIOCHEMICAL PHARMACOLOGY (2011)
α7 Nicotinic acetylcholine receptor agonist GTS-21 attenuates ventilator-induced tumour necrosis factor-α production and lung injury
M. Kox et al.
BRITISH JOURNAL OF ANAESTHESIA (2011)
Design, Synthesis, and Pharmacological Characterization of Novel Spirocyclic Quinuclidinyl-Δ2-Isoxazoline Derivatives as Potent and Selective Agonists of α7 Nicotinic Acetylcholine Receptors
Clelia Dallanoce et al.
CHEMMEDCHEM (2011)
A transgenic mouse model reveals fast nicotinic transmission in hippocampal pyramidal neurons
Michael J. Grybko et al.
EUROPEAN JOURNAL OF NEUROSCIENCE (2011)
The effective opening of nicotinic acetylcholine receptors with single agonist binding sites
Dustin K. Williams et al.
JOURNAL OF GENERAL PHYSIOLOGY (2011)
Characterization of 2-[[4-Fluoro-3-(trifluoromethyl)phenyl]amino]-4-(4-pyridinyl)-5-thiazolemethanol (JNJ-1930942), a Novel Positive Allosteric Modulator of the α7 Nicotinic Acetylcholine Receptor
Theo Dinklo et al.
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS (2011)
Electrophysiological Perspectives on the Therapeutic Use of Nicotinic Acetylcholine Receptor Partial Agonists
Roger L. Papke et al.
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS (2011)
Urinary N-methylpyridinium and trigonelline as candidate dietary biomarkers of coffee consumption
Roman Lang et al.
MOLECULAR NUTRITION & FOOD RESEARCH (2011)
Investigation of the Molecular Mechanism of the α7 Nicotinic Acetylcholine Receptor Positive Allosteric Modulator PNU-120596 Provides Evidence for Two Distinct Desensitized States
Dustin K. Williams et al.
MOLECULAR PHARMACOLOGY (2011)
Agonist activation of α7 nicotinic acetylcholine receptors via an allosteric transmembrane site
JasKiran K. Gill et al.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2011)
Voltage- and temperature-dependent allosteric modulation of alpha 7 nicotinic receptors by PNU120596
Fabrio Sitzia et al.
FRONTIERS IN PHARMACOLOGY (2011)
Discovery of novel α7 nicotinic receptor antagonists
Youyi Peng et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2010)
Discovery of 4-(5-Methyloxazolo[4,5-b]pyridin-2-yl)-1,4-diazabicyclo[3.2.2]nonane (CP-810,123), a Novel α7 Nicotinic Acetylcholine Receptor Agonist for the Treatment of Cognitive Disorders in Schizophrenia: Synthesis, SAR Development, and in Vivo Efficacy in Cognition Models
Christopher J. O'Donnell et al.
JOURNAL OF MEDICINAL CHEMISTRY (2010)
Tricks of Perspective: Insights and Limitations to the Study of Macroscopic Currents for the Analysis of nAChR Activation and Desensitization
Roger L. Papke
JOURNAL OF MOLECULAR NEUROSCIENCE (2010)
An alpha 7 Nicotinic Acetylcholine Receptor-Selective Agonist Reduces Weight Gain and Metabolic Changes in a Mouse Model of Diabetes
Mario B. Marrero et al.
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS (2010)
In Vitro Pharmacological Characterization of a Novel Selective α7 Neuronal Nicotinic Acetylcholine Receptor Agonist ABT-107
John Malysz et al.
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS (2010)
Nicotinic Acetylcholine Receptor Transmembrane Mutations Convert Ivermectin from a Positive to a Negative Allosteric Modulator
Toby Collins et al.
MOLECULAR PHARMACOLOGY (2010)
Working with OpusXpress: Methods for high volume oocyte experiments
Roger L. Papke et al.
METHODS (2010)
Glutamate Receptor Ion Channels: Structure, Regulation, and Function
Stephen F. Traynelis et al.
PHARMACOLOGICAL REVIEWS (2010)
Rat neuronal nicotinic acetylcholine receptors containing alpha 7 subunit: pharmacological properties of ligand binding and function
Yingxian Xiao et al.
ACTA PHARMACOLOGICA SINICA (2009)
Cholinergic agonists regulate JAK2/STAT3 signaling to suppress endothelial cell activation
Prodyot K. Chatterjee et al.
AMERICAN JOURNAL OF PHYSIOLOGY-CELL PHYSIOLOGY (2009)
Selective α7 nicotinic receptor activation by AZD0328 enhances cortical dopamine release and improves learning and attentional processes
Simon Sydserff et al.
BIOCHEMICAL PHARMACOLOGY (2009)
SAR and biological evaluation of SEN12333/WAY-317538: Novel alpha 7 nicotinic acetylcholine receptor agonist
Simon N. Haydar et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2009)
Investigating the role of protein folding and assembly in cell-type dependent expression of α7 nicotinic receptors using a green fluorescent protein chimera
H. K. Lee et al.
BRAIN RESEARCH (2009)
Convergence of alpha 7 nicotinic acetylcholine receptor-activated pathways for anti-apoptosis and anti-inflammation: Central role for JAK2 activation of STAT3 and NF-κB
Mario B. Marrero et al.
BRAIN RESEARCH (2009)
Positive allosteric modulation of α7 neuronal nicotinic acetylcholine receptors: lack of cytotoxicity in PC12 cells and rat primary cortical neurons
Min Hu et al.
BRITISH JOURNAL OF PHARMACOLOGY (2009)
Role of channel activation in cognitive enhancement mediated by α7 nicotinic acetylcholine receptors
Clark A. Briggs et al.
BRITISH JOURNAL OF PHARMACOLOGY (2009)
Structural determinants for interaction of partial agonists with acetylcholine binding protein and neuronal α7 nicotinic acetylcholine receptor
Ryan E. Hibbs et al.
EMBO JOURNAL (2009)
Cholinergic control of inflammation
M. Rosas-Ballina et al.
JOURNAL OF INTERNAL MEDICINE (2009)
Discovery of 4-(5-(4-Chlorophenyl)-2-methyl-3-propionyl-1H-pyrrol-1-yl)benzenesulfonamide (A-867744) as a Novel Positive Allosteric Modulator of the α7 Nicotinic Acetylcholine Receptor
Ramin Faghih et al.
JOURNAL OF MEDICINAL CHEMISTRY (2009)
Old and New Pharmacology: Positive Allosteric Modulation of the α7 Nicotinic Acetylcholine Receptor by the 5-Hydroxytryptamine2B/C Receptor Antagonist SB-206553 (3,5-Dihydro-5-methyl-N-3-pyridinylbenzo[1,2-b:4,5-b′]di pyrrole-1(2H)-carboxamide)
John Dunlop et al.
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS (2009)
Activation and Desensitization of Nicotinic α7-type Acetylcholine Receptors by Benzylidene Anabaseines and Nicotine
Roger L. Papke et al.
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS (2009)
Procognitive and Neuroprotective Activity of a Novel α7 Nicotinic Acetylcholine Receptor Agonist for Treatment of Neurodegenerative and Cognitive Disorders
Renza Roncarati et al.
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS (2009)
Proteomic Analysis of an α7 Nicotinic Acetylcholine Receptor Interactome
Joao A. Paulo et al.
JOURNAL OF PROTEOME RESEARCH (2009)
Antidepressant-like effects of nicotinic acetylcholine receptor antagonists, but not agonists, in the mouse forced swim and mouse tail suspension tests
J. T. Andreasen et al.
JOURNAL OF PSYCHOPHARMACOLOGY (2009)
The Selective α7 Agonist GTS-21 Attenuates Cytokine Production in Human Whole Blood and Human Monocytes Activated by Ligands for TLR2, TLR3, TLR4, TLR9, and RAGE
Mauricio Rosas-Ballina et al.
MOLECULAR MEDICINE (2009)
Selective Inhibition of Acetylcholine-Evoked Responses of α7 Neuronal Nicotinic Acetylcholine Receptors by Novel tris- and tetrakis-Azaaromatic Quaternary Ammonium Antagonists
Gretchen Y. Lopez-Hernandez et al.
MOLECULAR PHARMACOLOGY (2009)
Discovery of N-[(3R,5R)-1-azabicyclo[3.2.1]oct-3-yl]furo[2,3-c]pyridine-5-carboxamide as an agonist of the α7 nicotinic acetylcholine receptor:: In vitro and in vivo activity
Brad A. Acker et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2008)
α7 nicotinic acetylcholine receptor agonist properties of tilorone and related tricyclic analogues
C. A. Briggs et al.
BRITISH JOURNAL OF PHARMACOLOGY (2008)
Preclinical Characterization of A-582941: A Novel α7 Neuronal Nicotinic Receptor Agonist with Broad Spectrum Cognition-Enhancing Properties
Karin R. Tietje et al.
CNS Neuroscience & Therapeutics (2008)
αConotoxin Arenatus IB[V11I,V16D] Is a Potent and Selective Antagonist at Rat and Human Native α7 Nicotinic Acetylcholine Receptors
Neal Innocent et al.
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS (2008)
Sazetidine-A is a potent and selective agonist at native and recombinant alpha 4 beta 2 nicotinic acetylcholine receptors
Ruud Zwart et al.
MOLECULAR PHARMACOLOGY (2008)
Positive Allosteric Modulation of the α7 Nicotinic Acetylcholine Receptor: Ligand Interactions with Distinct Binding Sites and Evidence for a Prominent Role of the M2-M3 Segment
Daniel Bertrand et al.
MOLECULAR PHARMACOLOGY (2008)
Multiple Pharmacophores for the Selective Activation of Nicotinic α7-Type Acetylcholine Receptors
Nicole A. Horenstein et al.
MOLECULAR PHARMACOLOGY (2008)
On the nature of partial agonism in the nicotinic receptor superfamily
Remigijus Lape et al.
NATURE (2008)
Potentiation of α7 nicotinic acetylcholine receptors via an allosteric transmembrane site
Gareth T. Young et al.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2008)
Improvement of contextual memory by S 24795 in aged mice: comparison with memantine
Daniel Beracochea et al.
PSYCHOPHARMACOLOGY (2008)
In vitro screening strategies for nicotinic receptor ligands
John Dunlop et al.
BIOCHEMICAL PHARMACOLOGY (2007)
An allosteric modulator of the α7 nicotinic acetylcholine receptor possessing cognition-enhancing properties in vivo
Daniel B. Timmermann et al.
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS (2007)
Identification of domains influencing assembly and ion channel properties in α7 nicotinic receptor and 5-HT3 receptor subunit chimaeras
V. J. Gee et al.
BRITISH JOURNAL OF PHARMACOLOGY (2007)
Distinct profiles of α7 nAChR positive allosteric modulation revealed by structurally diverse chemotypes
Jens Halvard Gronlien et al.
MOLECULAR PHARMACOLOGY (2007)
Partial agonist and neuromodulatory activity of S 24795 for alpha7 nAChR responses of hippocampal interneurons
Gretchen Lopez-Hernandez et al.
NEUROPHARMACOLOGY (2007)
Nootropic α7 nicotinic receptor allosteric modulator derived from GABAA receptor modulators
Herman J. Ng et al.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2007)
The novel α7 nicotinic acetylcholine receptor agonist N-[(3R)-1-azabicyclo[2.2.2]oct-3-yl]-7-[2-(methoxy)phenyl]-1-benzofuran-2-carboxamide improves working and recognition memory in rodents
Frank G. Boess et al.
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS (2007)
JN403, in vitro characterization of a novel nicotinic acetylcholine receptor α7 selective agonist
Dominik Feuerbach et al.
NEUROSCIENCE LETTERS (2007)
Selective α7-nicotinic acetylcholine receptor agonist GTS-21 improves survival in murine endotoxemia and severe sepsis
Valentin A. Pavlov et al.
CRITICAL CARE MEDICINE (2007)
The pharmacological activity of nicotine and nornicotine on nAChRs subtypes: relevance to nicotine dependence and drug discovery
Roger L. Papke et al.
JOURNAL OF NEUROCHEMISTRY (2007)
α7 Nicotinic receptor gene delivery into mouse hippocampal neurons leads to functional receptor expression, improved spatial memory-related performance, and tau hyperphosphorylation
K. Ren et al.
NEUROSCIENCE (2007)
SSR180711, a novel selective α7 nicotinic receptor partial agonist:: (I) binding and functional profile
Bruno Biton et al.
NEUROPSYCHOPHARMACOLOGY (2007)
Sazetidine-a, a novel ligand that desensitizes α4β2 nicotinic acetylcholine receptors without activating them
Yingxian Xiao et al.
MOLECULAR PHARMACOLOGY (2006)
An autoradiographic analysis of [125I] α-bungarotoxin binding in rat brain after chronic nicotine exposure
Bruce A. Rasmussen et al.
NEUROSCIENCE LETTERS (2006)
Selective nicotinic acetylcholine receptor subunit deficits identified in Alzheimer's disease, Parkinson's disease and dementia with Lewy bodies by immunoprecipitation
Cecilia Gotti et al.
NEUROBIOLOGY OF DISEASE (2006)
α-selenoconotoxins, a new class of potent α7 neuronal nicotinic receptor antagonists
Christopher J. Armishaw et al.
JOURNAL OF BIOLOGICAL CHEMISTRY (2006)
The vagus nerve and nicotinic receptors modulate experimental pancreatitis severity in mice
David J. Van Westerloo et al.
GASTROENTEROLOGY (2006)
Desensitization characteristics of the human alpha 7nAChR/5HT3A chimera receptor
Theo Dinklo et al.
JOURNAL OF MOLECULAR NEUROSCIENCE (2006)
Structures of Aplysia AChBP complexes with nicotinic agonists and antagonists reveal distinctive binding interfaces and conformations
SB Hansen et al.
EMBO JOURNAL (2005)
The characterization of a novel rigid nicotine analog with α7-selective nAChR agonist activity and modulation of agonist properties by boron inclusion
RL Papke et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2005)
Stimulation of the vagus nerve attenuates macrophage activation by activating the Jak2-STAT3 signaling pathway
WJ de Jonge et al.
NATURE IMMUNOLOGY (2005)
Tropisetron improves deficits in auditory P50 suppression in schizophrenia
K Koike et al.
SCHIZOPHRENIA RESEARCH (2005)
A novel positive allosteric modulator of the α7 neuronal nicotinic acetylcholine receptor:: In vitro and in vivo characterization
RS Hurst et al.
JOURNAL OF NEUROSCIENCE (2005)
Molecular dissection of tropisetron, an α7 nicotinic acetylcholine receptor-selective partial agonist
RL Papke et al.
NEUROSCIENCE LETTERS (2005)
Refined structure of the nicotinic acetylcholine receptor at 4 Å resolution
N Unwin
JOURNAL OF MOLECULAR BIOLOGY (2005)
Discovery and structure -: Activity relationship of quinuclidine benzamides as agonists of α7 nicotinic acetylcholine receptors
AL Bodnar et al.
JOURNAL OF MEDICINAL CHEMISTRY (2005)
Ric-3 promotes functional expression of the nicotinic acetylcholine receptor α7 subunit in mammalian cells
ME Williams et al.
JOURNAL OF BIOLOGICAL CHEMISTRY (2005)
Activity of α7-selective agonists at nicotinic and serotonin 5HT3 receptors expressed in Xenopus oocytes
RL Papke et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2004)
The neuroprotective effect of 2-(3-pyridyl)-1-azabicyclo[3.2.2]nonane (TC-1698), a novel α7 ligand, is prevented through angiotensin II activation of a tyrosine phosphatase
MB Marrero et al.
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS (2004)
(+)-3-[2-(benzo[b]thiophen-2-yl)-2-oxoethyl]-1-azabicyclo[2.2.2]octane, as potent agonists for the α7 nicotinic acetylcholine receptor
R Tatsumi et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2004)
Alpha-7 nicotinic receptor agonists: potential new candidates for the treatment of schizophrenia
LF Martin et al.
PSYCHOPHARMACOLOGY (2004)
Stable expression and characterisation of a human α7 nicotinic subunit chimera:: a tool for functional high-throughput screening
PJ Craig et al.
EUROPEAN JOURNAL OF PHARMACOLOGY (2004)
Conservation within the RIC-3 gene family - Effectors of mammalian nicotinic acetylcholine receptor expression
S Halevi et al.
JOURNAL OF BIOLOGICAL CHEMISTRY (2003)
Galantamine is an allosterically potentiating ligand of neuronal nicotinic but not of muscarinic acetylcholine receptors
M Samochocki et al.
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS (2003)
Nicotinic acetylcholine receptor α7 subunit is an essential regulator of inflammation
H Wang et al.
NATURE (2003)
α-conotoxins ImI and ImII -: Similar α7 nicotinic receptor antagonists act at different sites
M Ellison et al.
JOURNAL OF BIOLOGICAL CHEMISTRY (2003)
The role of neuronal nicotinic acetylcholine receptor subunits in autonomic ganglia: lessons from knockout mice
NS Wang et al.
PROGRESS IN NEUROBIOLOGY (2002)
PSAB-OFP, a selective α7 nicotinic receptor agonist, is also a potent agonist of the 5-HT3 receptor
LM Broad et al.
EUROPEAN JOURNAL OF PHARMACOLOGY (2002)
Activation and inhibition of native neuronal alpha-bungarotoxin-sensitive nicotinic ACh receptors
VV Uteshev et al.
BRAIN RESEARCH (2002)
5-hydroxyindole potentiates human α7 nicotinic receptor-mediated responses and enhances acetylcholine-induced glutamate release in cerebellar slices
R Zwart et al.
NEUROPHARMACOLOGY (2002)
Comparative pharmacology of rat and human α7 nAChR conducted with net charge analysis
RL Papke et al.
BRITISH JOURNAL OF PHARMACOLOGY (2002)
Pharmacological properties of rat α7 nicotinic receptors expressed in native and recombinant cell systems
C Virginio et al.
EUROPEAN JOURNAL OF PHARMACOLOGY (2002)
Some properties of human neuronal α7 nicotinic acetylcholine receptors fused to the green fluorescent protein
E Palma et al.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2002)
Hippocampal alpha 7 and alpha 4 beta 2 nicotinic receptors and working memory
ED Levin et al.
NEUROSCIENCE (2002)
Specific activation pf the α7 nicotinic acetylcholine receptor by a quaternary analog of cocaine
MM Francis et al.
MOLECULAR PHARMACOLOGY (2001)
Crystal structure of an ACh-binding protein reveals the ligand-binding domain of nicotinic receptors
K Brejc et al.
NATURE (2001)
α10:: A determinant of nicotinic cholinergic receptor function in mammalian vestibular and cochlear mechanosensory hair cells
AB Elgoyhen et al.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2001)
Molecular and physiological diversity of nicotinic acetylcholine receptors in the midbrain dopaminergic nuclei
R Klink et al.
JOURNAL OF NEUROSCIENCE (2001)
The 5-HT3 antagonist tropisetron (ICS 205-930) is a potent and selective α7 nicotinic receptor partial agonist
JE Macor et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2001)
Overview of nicotinic receptors and their roles in the central nervous system
JA Dani
BIOLOGICAL PSYCHIATRY (2001)
(-)-spiro[1-azabicyclo[2.2.2]octane-3,5′-oxazolidin-2′-one], a conformationally restricted analogue of acetylcholine, is a highly selective full agonist at the α7 nicotinic acetylcholine receptor
G Mullen et al.
JOURNAL OF MEDICINAL CHEMISTRY (2000)
α-Bungarotoxin-sensitive nicotinic receptors indirectly modulate [3H]dopamine release in rat striatal slices via glutamate release
S Kaiser et al.
MOLECULAR PHARMACOLOGY (2000)
Vagus nerve stimulation attenuates the systemic inflammatory response to endotoxin
LV Borovikova et al.
NATURE (2000)
Neuronal alpha-bungarotoxin receptors are alpha 7 subunit homomers
RC Drisdel et al.
JOURNAL OF NEUROSCIENCE (2000)
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