相关参考文献
注意:仅列出部分参考文献,下载原文获取全部文献信息。Synthesis, Characterization, Antimicrobial Evaluation, and Computational Investigation of Substituted Imidazo[2,1-b][1,3,4]Thiadiazole Derivatives
Meltem Dagli et al.
CHEMISTRYSELECT (2020)
Synthesis, characterization, molecular docking and biological activity of 5,6-bis-(4-fluoro-phenyl)-3,4,7,8-tetraaza-bicyclo[8.3.1]tetradeca-1(13),4,6,10(14),11-pentaene-2,9-dione and its transition metal complexes
Preeti Jain et al.
JOURNAL OF SAUDI CHEMICAL SOCIETY (2018)
Quantitative structure-activity relationship of substituted imidazothiadiazoles for their binding against the ecdysone receptor of Sf-9 cells
Taiyo Yokoi et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2017)
Benzenesulfonamide bearing imidazothiadiazole and thiazolotriazole scaffolds as potent tumor associated human carbonic anhydrase IX and XII inhibitors
Rajiv Kumar et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2017)
SAR Exploration Guided by LE and Fsp(3): Discovery of a Selective and Orally Efficacious ROR gamma Inhibitor
Kazuyuki Hirata et al.
ACS MEDICINAL CHEMISTRY LETTERS (2016)
A novel inhibitor of BCL2, Disarib abrogates tumor growth while sparing platelets, by activating intrinsic pathway of apoptosis
Supriya V. Vartak et al.
BIOCHEMICAL PHARMACOLOGY (2016)
Identification of a novel BCL2-specific inhibitor that binds predominantly to the BH1 domain
Divyaanka Iyer et al.
FEBS JOURNAL (2016)
Imidazothiazole and related heterocyclic systems. Synthesis, chemical and biological properties
Mirta L. Fascio et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2015)
Novel imidazo[2,1-b]-1,3,4-thiadiazoles as promising antifungal agents against clinical isolate of Cryptococcus neoformans
Wesam S. Alwan et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2015)
Synthesis and Regioselective Reaction of Some Unsymmetrical Heterocyclic Chalcone Derivatives and Spiro Heterocyclic Compounds as Antibacterial Agents
Maher A. El-Hashash et al.
MOLECULES (2015)
Synthesis and antiproliferative activity of imidazo[2,1-b][1,3,4]thiadiazole derivatives
Sujeet Kumar et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2014)
2-(4-Chlorobenzyl)-6-arylimidazo[2,1-b][1,3,4]thiadiazoles: Synthesis, cytotoxic activity and mechanism of action
Sujeet Kumar et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2014)
Novel imidazo[2,1-b][1,3,4]thiadiazole carrying rhodanine-3-acetic acid as potential antitubercular agents
Shankar G. Alegaon et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2012)
2,6-Disubstituted imidazo[2,1-b][1,3,4]thiadiazoles: Search for anticancer agents
Malleshappa N. Noolvi et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2012)
Microwave-assisted synthesis and antimicrobial activity of some imidazo[2,1-b][1,3,4]thiadiazole derivatives
Sharad Dhepe et al.
MEDICINAL CHEMISTRY RESEARCH (2012)
Novel Levamisole Derivative Induces Extrinsic Pathway of Apoptosis in Cancer Cells and Inhibits Tumor Progression in Mice
Mahesh Hegde et al.
PLOS ONE (2012)
Synthesis and biological evaluation of novel 2-aralkyl-5-substituted-6-(4′-fluorophenyl)-imidazo[2,1-b][1,3,4]thiadiazole derivatives as potent anticancer agents
Subhas S. Karki et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2011)
Epidermal growth factor receptor in relation to tumor development: EGFR gene and cancer
Tetsuya Mitsudomi et al.
FEBS JOURNAL (2010)
Software News and Update AutoDock Vina: Improving the Speed and Accuracy of Docking with a New Scoring Function, Efficient Optimization, and Multithreading
Oleg Trott et al.
JOURNAL OF COMPUTATIONAL CHEMISTRY (2010)
Escape from Flatland: Increasing Saturation as an Approach to Improving Clinical Success
Frank Lovering et al.
JOURNAL OF MEDICINAL CHEMISTRY (2009)
Synthesis and biological evaluation of 2-trifluoromethyl/sulfonamido-5,6-diaryl substituted imidazo[2,1-b]-1,3,4-thiadiazoles: A novel class of cyclooxygenase-2 inhibitors
Andanappa K. Gadad et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2008)
Synthesis and anti-inflammatory evaluation of methylene bridged benzofuranyl imidazo[2,1-b][1,3,4]thiadiazoles
V. B. Jadhav et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2008)
Regiospecific and highly flexible synthesis of 1,4,5-trisubstituted 2-sulfanylimidazoles from structurally diverse ethanone precursors
Stefan A. Laufer et al.
SYNTHESIS-STUTTGART (2008)
Epidermal growth factor receptor biology in head and neck cancer
Shailaja Kalyankrishna et al.
JOURNAL OF CLINICAL ONCOLOGY (2006)
Synthesis and anti-tubercular activity of a series of 2-sulfonamido/trifluoromethyl-6-substituted imidazo[2,1-b]-1,3,4-thiadiazole derivatives
AK Gadad et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2004)
Design, synthesis, and biological evaluation of hybrid molecules containing α-methylene-γ-butyrolactones and polypyrrole minor groove binders
PG Baraldi et al.
JOURNAL OF MEDICINAL CHEMISTRY (2004)
Derivatized amino acids relevant to native peptide synthesis by chemical ligation and acyl transfer
DLJ Clive et al.
JOURNAL OF ORGANIC CHEMISTRY (2003)
Molecular properties that influence the oral bioavailability of drug candidates
DF Veber et al.
JOURNAL OF MEDICINAL CHEMISTRY (2002)
Synthesis and antibacterial activity of some 5-guanylhydrazone/thiocyanato-6-arylimidazo[2,1-b]-1,3,4-thiadiazole-2-sulfonamide derivatives
AK Gadad et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2000)