相关参考文献
注意：仅列出部分参考文献，下载原文获取全部文献信息。Design, synthesis and evaluation of novel thienopyrimidine-based agents bearing diaryl urea functionality as potential inhibitors of angiogenesis
Aram Faraji et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2021)
A facile method for preparation and evaluation of the antimicrobial efficiency of various heterocycles containing thieno[2,3-d]pyrimidine
Ahmed F. Saber et al.
SYNTHETIC COMMUNICATIONS (2021)
Novel thienopyrimidine analogues as potential metabotropic glutamate receptors inhibitors and anticancer activity: Synthesis, In-vitro, In-silico, and SAR approaches
Mohammed A. Khedr et al.
BIOORGANIC CHEMISTRY (2021)
Design, synthesis, biological evaluation and molecular modeling study of new thieno[2,3-d]pyrimidines with anti-proliferative activity on pancreatic cancer cell lines
Mohamed S. H. Salem et al.
BIOORGANIC CHEMISTRY (2020)
Thiazole-containing compounds as therapeutic targets for cancer therapy
Prabodh Chander Sharma et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2020)
Design, synthesis and molecular modeling study of certain VEGFR-2 inhibitors based on thienopyrimidne scaffold as cancer targeting agents
Amna Ghith et al.
BIOORGANIC CHEMISTRY (2019)
Thieno[2,3-d] pyrimidine as a promising scaffold in medicinal chemistry: Recent advances
Eslam M. H. Ali et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2019)
Phytochemicals Targeting VEGF and VEGF-Related Multifactors as Anticancer Therapy
Amna Parveen et al.
JOURNAL OF CLINICAL MEDICINE (2019)
Synthesis, reactions, and biological study of some new thienopyrimidine derivatives as antimicrobial and anti-inflammatory agents
Mahmoud S. Tolba et al.
JOURNAL OF THE CHINESE CHEMICAL SOCIETY (2019)
Synthesis and Antioxidant Evaluation of a New Class of Thienopyrimidine-rhodanine Hybrids
Kerru Nagaraju et al.
LETTERS IN DRUG DESIGN & DISCOVERY (2018)
Design and synthesis of thienopyrimidine urea derivatives with potential cytotoxic and pro-apoptotic activity against breast cancer cell line MCF-7
Eman F. Abdelhaleem et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2018)
Anti-Angiogenics: Their Value in Lung Cancer Therapy
Melanie Janning et al.
ONCOLOGY RESEARCH AND TREATMENT (2018)
Anti-Angiogenics: Current Situation and Future Perspectives
Katja Zirlik et al.
ONCOLOGY RESEARCH AND TREATMENT (2018)
Anti-Angiogenics: Their Value in Colorectal Cancer Therapy
Andreas Seeber et al.
ONCOLOGY RESEARCH AND TREATMENT (2018)
Serum levels of VEGF and MCSF in HER2+/HER2- breast cancer patients with metronomic neoadjuvant chemotherapy
Roberto J. Arai et al.
BIOMARKER RESEARCH (2018)
2-Substituted-thio-N-(4-substituted-thiazo1/1H-imidazol-2-yl) acetamides as BACE1 inhibitors: Synthesis, biological evaluation and docking studies
Gang Yan et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2017)
Design, synthesis and biological evaluations of N-Hydroxy thienopyrimidine-2,4-diones as inhibitors of HIV reverse transcriptase-associated RNase H
Jayakanth Kankanala et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2017)
RTN1-C mediates cerebral ischemia/reperfusion injury via ER stress and mitochondria-associated apoptosis pathways
Lingli Gong et al.
CELL DEATH & DISEASE (2017)
Computer-aided identification, synthesis and evaluation of substituted thienopyrimidines as novel inhibitors of HCV replication
Marcella Bassetto et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2016)
Discovery of Potent VEGFR-2 Inhibitors based on Furopyrimidine and Thienopyrimidne Scaffolds as Cancer Targeting Agents
Marwa A. Aziz et al.
SCIENTIFIC REPORTS (2016)
Synthesis, antiangiogenesis evaluation and molecular docking studies of 1-aryl-3-[(thieno[3,2-b]pyridin-7-ylthio)phenyl]ureas: Discovery of a new substitution pattern for type II VEGFR-2 Tyr kinase inhibitors
Vera A. Machado et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2015)
Evolution of a thienopyrimidine antitubercular relying on medicinal chemistry and metabolomics insights
Shao-Gang Li et al.
TETRAHEDRON LETTERS (2015)
FDA-approved small-molecule kinase inhibitors
Peng Wu et al.
TRENDS IN PHARMACOLOGICAL SCIENCES (2015)
Thieno[2,3-d]pyrimidine-2-carboxamides bearing a carboxybenzene group at 5-position: Highly potent, selective, and orally available MMP-13 inhibitors interacting with the S1 binding site
Hiroshi Nara et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2014)
Molecular Modeling Studies and Synthesis of Novel Methyl 2-(2-(4-Oxo-3-aryl-3,4-dihydroquinazolin-2-ylthio)acetamido)alkanoates with Potential Anti-cancer Activity as Inhibitors for Methionine Synthase
Ismail Mahmoud Elfekki et al.
CHEMICAL & PHARMACEUTICAL BULLETIN (2014)
Synthesis and Biological Evaluation of Chromenylurea and Chromanylurea Derivatives as Anti-TNF-α agents that Target the p38 MAPK Pathway
Xingzhou Li et al.
MOLECULES (2014)
Caffeic acid phenethyl ester synergistically enhances docetaxel and paclitaxel cytotoxicity in prostate cancer cells
Mai F. Tolba et al.
IUBMB LIFE (2013)
Vascular Endothelial Growth Factor (VEGF) Receptors: Drugs and New Inhibitors
Francesca Musumeci et al.
JOURNAL OF MEDICINAL CHEMISTRY (2012)
Molecular conformations, interactions, and properties associated with drug efficiency and clinical performance among VEGFR TK inhibitors
Michele McTigue et al.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2012)
Impact of aryloxy-linked quinazolines: A novel series of selective VEGFR-2 receptor tyrosine kinase inhibitors
Antonio Garofalo et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2011)
The design, synthesis, and evaluation of 8 hybrid DFG-out allosteric kinase inhibitors: A structural analysis of the binding interactions of Gleevec®, Nexavar®, and BIRB-796
Justin Dietrich et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2010)
Design, synthesis and biological evaluation of novel quinazoline derivatives as potential antitumor agents: Molecular docking study
Adel S. El-Azab et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2010)
Synthesis, Characterization and Biological Studies of Some Novel Thieno[2,3-d]pyrimidines
Khulud M. Al-Taisan et al.
MOLECULES (2010)
Analogs of a 4-aminothieno[2,3-d]pyrimidine lead (QB13) as modulators of P-glycoprotein substrate specificity
Hans-Georg Haecker et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2009)
Synthesis and antitumor activity of 6-and 2-(1-substituted-thio-4-methylpent-3-enyl)-5,8-dimethoxynaphthalene-1,4-diones
Li-Ming Zhao et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2009)
Synthesis and Biological Evaluation of 17β-Hydroxysteroid Dehydrogenase Type 1 (17β-HSD1) Inhibitors Based on a Thieno[2,3-d]pyrimidin-4(3H)-one Core
Annamaria Lilienkampf et al.
JOURNAL OF MEDICINAL CHEMISTRY (2009)
Pharmacophore modeling studies of type I and type II kinase inhibitors of Tie2
Qing-Qing Xie et al.
JOURNAL OF MOLECULAR GRAPHICS & MODELLING (2009)
Angiogenesis in brain tumours
Rakesh K. Jain et al.
NATURE REVIEWS NEUROSCIENCE (2007)
The NCI60 human tumour cell line anticancer drug screen
Robert H. Shoemaker
NATURE REVIEWS CANCER (2006)
Parallel synthesis and biological evaluation of 5,6,7,8-tetrahydrobenzothieno[2,3-d]pyrimidin-4(3H)-one cytotoxic agents selective for p21-deficient cells
LD Jennings et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2005)
Well diffusion for antifungal susceptibility testing
S Magaldi et al.
INTERNATIONAL JOURNAL OF INFECTIOUS DISEASES (2004)
分享论文
