相关参考文献
注意:仅列出部分参考文献,下载原文获取全部文献信息。Front Cover: Antibody Conjugation of a Chimeric BET Degrader Enables in vivo Activity (ChemMedChem 1/2020)
Thomas H. Pillow et al.
ChemMedChem (2020)
Pyrrolo[1,2-a]quinoxalines: Insulin Mimetics that Exhibit Potent and Selective Inhibition against Protein Tyrosine Phosphatase 1B
Javier Garcia-Marin et al.
CHEMMEDCHEM (2020)
Discovery of 4-[(5-arylidene-4-oxothiazolidin-3-yl)methyl]benzoic acid derivatives active as novel potent allosteric inhibitors of protein tyrosine phosphatase 1B: In silico studies and in vitro evaluation as insulinomimetic and anti-inflammatory agents
Rosaria Ottana et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2017)
Peripheral insulin resistance in ILK-depleted mice by reduction of GLUT4 expression
Marco Hatem-Vaquero et al.
JOURNAL OF ENDOCRINOLOGY (2017)
Metformin ameliorates high uric acid-induced insulin resistance in skeletal muscle cells
Huier Yuan et al.
MOLECULAR AND CELLULAR ENDOCRINOLOGY (2017)
Cyclocarya paliurus extract activates insulin signaling via Sirtuin1 in C2C12 myotubes and decreases blood glucose level in mice with impaired insulin secretion
Hisae Yoshitomi et al.
PLOS ONE (2017)
Novel Non-carboxylate Benzoylsulfonamide-Based Protein Tyrosine Phosphatase 1B Inhibitors with Non-competitive Actions
Ko Morishita et al.
CHEMICAL & PHARMACEUTICAL BULLETIN (2017)
Covalent Allosteric Inactivation of Protein Tyrosine Phosphatase 1B (PTP1B) by an Inhibitor-Electrophile Conjugate
Puminan Punthasee et al.
BIOCHEMISTRY (2017)
Selective Inhibition of PTP1B by Vitalboside A from Syzygium cumini Enhances Insulin Sensitivity and Attenuates Lipid Accumulation Via Partial Agonism to PPARγ: In Vitro and In Silico Investigation
Gopal Thiyagarajan et al.
CHEMICAL BIOLOGY & DRUG DESIGN (2016)
Targeting the disordered C terminus of PTP1B with an allosteric inhibitor
Navasona Krishnan et al.
NATURE CHEMICAL BIOLOGY (2014)
Design, synthesis and insulin-sensitising effects of novel PTP1B inhibitors
Yan-Bo Tang et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2013)
PTP1B: A simple enzyme for a complex world
Matthew Feldhammer et al.
CRITICAL REVIEWS IN BIOCHEMISTRY AND MOLECULAR BIOLOGY (2013)
Binding and discerning interactions of PTP1B allosteric inhibitors: Novel insights from molecular dynamics simulations
Ranajit Nivrutti Shinde et al.
JOURNAL OF MOLECULAR GRAPHICS & MODELLING (2013)
Reduction of heart failure by pharmacological inhibition or gene deletion of protein tyrosine phosphatase 1B
Elodie Gomez et al.
JOURNAL OF MOLECULAR AND CELLULAR CARDIOLOGY (2012)
Docking Study of Biflavonoids, Allosteric Inhibitors of Protein Tyrosine Phosphatase 1B
BULLETIN OF THE KOREAN CHEMICAL SOCIETY (2010)
Protein Tyrosine Phosphatase 1B, a Major Regulator of Leptin-Mediated Control of Cardiovascular Function
Eric J. Belin de Chantemele et al.
CIRCULATION (2009)
Deletion of Protein Tyrosine Phosphatase 1b Improves Peripheral Insulin Resistance and Vascular Function in Obese, Leptin-Resistant Mice via Reduced Oxidant Tone
M. Irfan Ali et al.
CIRCULATION RESEARCH (2009)
Structural insights into the design of nonpeptidic isothiazolidinone-containing inhibitors of protein-tyrosine phosphatase 1B
Paul J. Ala et al.
JOURNAL OF BIOLOGICAL CHEMISTRY (2006)
Allosteric inhibition of PTP1B activity by selective modification of a non-active site cysteine residue
SK Hansen et al.
BIOCHEMISTRY (2005)
Allosteric inhibition of protein tyrosine phosphatase 1B
C Wiesmann et al.
NATURE STRUCTURAL & MOLECULAR BIOLOGY (2004)
PTP1B regulates leptin signal transduction in vivo
JM Zabolotny et al.
DEVELOPMENTAL CELL (2002)
Attenuation of leptin action and regulation of obesity by protein tyrosine phosphatase 1B
A Cheng et al.
DEVELOPMENTAL CELL (2002)
Molecular basis for the dephosphorylation of the activation segment of the insulin receptor by protein tyrosine phosphatase 1B
A Salmeen et al.
MOLECULAR CELL (2000)