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EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2009)
Synthesis of Functionalized Spiroaziridine-oxindoles from 3-Ylideneoxindoles: An Easy Route to 3-(Aminoalkyl)oxindoles
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EUROPEAN JOURNAL OF ORGANIC CHEMISTRY (2009)
Catalytic Enantioselective Aza-Henry Reactions
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EUROPEAN JOURNAL OF ORGANIC CHEMISTRY (2009)
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FUTURE MEDICINAL CHEMISTRY (2009)
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FUTURE MEDICINAL CHEMISTRY (2009)
A New Strategy for the Synthesis of Optically Pure β-Fluoroalkyl β-Amino Acid Derivatives
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ORGANIC LETTERS (2009)
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SYNLETT (2009)
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R Ballini et al.
TETRAHEDRON (2004)
Virtually complete control of simple and face diastereoselectivity in the Michael addition reactions between achiral equivalents of a nucleophilic glycine and (S)- or (R)-3-(E-Enoyl)-4-phenyl-1,3-oxazolidin-2-ones:: Practical method for preparation of β-substituted pyroglutamic acids and prolines
VA Soloshonok et al.
JOURNAL OF ORGANIC CHEMISTRY (2004)
Mimicking enzymatic transaminations: attempts to understand and develop a catalytic asymmetric approach to chiral alpha-amino acids
S Bachmann et al.
ORGANIC & BIOMOLECULAR CHEMISTRY (2004)
Convenient asymmetric synthesis off β-substituted α,α-difluoro-β-amino acids via Reformatsky reaction between Davis' N-sulfinylimines and ethyl bromodifluoroacetate
A Sorochinsky et al.
JOURNAL OF ORGANIC CHEMISTRY (2003)
Efficient synthesis of sterically constrained symmetrically α,α-disubstituted α-amino acids under operationally convenient conditions
TK Ellis et al.
JOURNAL OF ORGANIC CHEMISTRY (2003)
Simple and highly diastereoselective synthesis of trifluoromethyl-containing myosmines via reaction between 2-(aminomethyl)pyridine and 1,1,1,5,5,5-hexafluoro-2,4-pentanedione
H Ohkura et al.
TETRAHEDRON LETTERS (2003)
Chemo- and regioselectivity in the reactions between highly electrophilic fluorine containing dicarbonyl compounds and amines. Improved synthesis of the corresponding imines/enamines
H Ohkura et al.
TETRAHEDRON (2003)
Efficient, practical synthesis of symmetrically α,α-disubstituted α-amino acids
TK Ellis et al.
TETRAHEDRON LETTERS (2003)
N-tert-Butanesulfinyl imines:: Versatile intermediates for the asymmetric synthesis of amines
JA Ellman et al.
ACCOUNTS OF CHEMICAL RESEARCH (2002)
Convenient, large-scale asymmetric synthesis of β-aryl-substituted α,α-difluoro-β-amino acids
VA Soloshonok et al.
TETRAHEDRON LETTERS (2002)
Efficient enantioselective additions of terminal alkynes and aldehydes under operationally convenient conditions
D Boyall et al.
ORGANIC LETTERS (2002)
New strategy for the stereoselective synthesis of fluorinated β-amino acids
S Fustero et al.
JOURNAL OF ORGANIC CHEMISTRY (2002)
New approach to biomimetic transamination using bifunctional [1,3]-proton transfer catalysis in thioxanthenyl dioxide imines
A Hjelmencrantz et al.
JOURNAL OF ORGANIC CHEMISTRY (2002)
Asymmetric synthesis of diarylmethylamines by diastereoselective addition of organometallic reagents to chiral N-tert-butanesulfinimines:: switchover of diastereofacial selectivity
N Plobeck et al.
TETRAHEDRON-ASYMMETRY (2002)
Simple access to novel β-hydroxy-β-trifluoromethyl imines
JA Barten et al.
JOURNAL OF FLUORINE CHEMISTRY (2002)
iso-propyl phenylacetate:: formation of a single enolate with tBuP4 as base
A Solladié-Cavallo et al.
TETRAHEDRON LETTERS (2002)
Large-scale asymmetric synthesis of novel sterically constrained 2′,6′-dimethyl- and α,2′,6′-trimethyltyrosine and -phenylalanine derivatives via alkylation of chiral equivalents of nucleophilic glycine and alanine
VA Soloshonok et al.
TETRAHEDRON (2001)
Asymmetric synthesis of α,β-dialkyl-α-phenylalanines via direct alkylation of a chiral alanine derivative with racemic α-alkylbenzyl bromides.: A case of high enantiomer differentiation at room temperature
VA Soloshonok et al.
ORGANIC LETTERS (2001)
A unique case of face diastereoselectivity in the Michael addition reactions between Ni(II)-complexes of glycine and chiral 3-(E-enoyl)-1,3-oxazolidin-2-ones
VA Soloshonok et al.
TETRAHEDRON LETTERS (2000)
Convenient, asymmetric synthesis of enantiomerically pure 2′,6′-dimethyltyrosine (DMT) via alkylation of chiral equivalent of nucleophilic glycine
XJ Tang et al.
TETRAHEDRON-ASYMMETRY (2000)
Convenient, large-scale asymmetric synthesis of enantiomerically pure trans-cinnamylglycine and -α-alanine
W Qiu et al.
TETRAHEDRON (2000)
(S)- or (R)-3-(E-enoyl)-4-phenyl-1,3-oxazolidin-2-ones:: Ideal Michael accepters to afford a virtually complete control of simple and face diastereoselectivity in addition reactions with glycine derivatives
VA Soloshonok et al.
ORGANIC LETTERS (2000)