期刊
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY
卷 2016, 期 14, 页码 2398-2403出版社
WILEY-V C H VERLAG GMBH
DOI: 10.1002/ejoc.201600384
关键词
Alkylation; Cyclization; Fused-ring systems; Nitrogen heterocycles; Oxidation
资金
- Department of Science and Technology (DST), New Delhi
- Council of Scientific and Industrial Research (CSIR), New Delhi
- CSIR
- DST (New Delhi)
- University Grants Commission (UGC), New Delhi
- UGC
- DST
A convenient one-pot protocol for the synthesis of benzo-fused and indole-fused indolizines from Baylis-Hillman acetates was developed. This strategy involves CuBr/tert-butyl hydroperoxide promoted oxidation, intramolecular cyclization, and aromatization as key steps. The efficacy of this methodology was demonstrated by the formal synthesis of (+/-)-crispine A, a biologically active molecule.
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