4.8 Article

Sulfopin is a covalent inhibitor of Pin1 that blocks Myc-driven tumors in vivo

相关参考文献

注意:仅列出部分参考文献,下载原文获取全部文献信息。
Article Biochemistry & Molecular Biology

Identification of a potent and selective covalent Pin1 inhibitor

Benika J. Pinch et al.

NATURE CHEMICAL BIOLOGY (2020)

Article Biochemistry & Molecular Biology

Synaptic Protein Degradation Controls Sexually Dimorphic Circuits through Regulation of DCC/UNC-40

Yehuda Salzberg et al.

CURRENT BIOLOGY (2020)

Article Chemistry, Multidisciplinary

Rapid Covalent-Probe Discovery by Electrophile-Fragment Screening

Efrat Resnick et al.

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2019)

Article Chemistry, Multidisciplinary

A Chemoproteomic Strategy for Direct and Proteome-Wide Covalent Inhibitor Target-Site Identification

Christopher M. Browne et al.

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2019)

Article Chemistry, Analytical

A Dimethyl-Labeling-Based Strategy for Site-Specifically Quantitative Chemical Proteomics

Fan Yang et al.

ANALYTICAL CHEMISTRY (2018)

Article Biochemistry & Molecular Biology

Targeting KRAS Mutant Cancers with a Covalent G12C-Specific Inhibitor

Matthew R. Janes et al.

Review Cell Biology

Prolyl isomerase Pin1: a promoter of cancer and a target for therapy

Yang Chen et al.

CELL DEATH & DISEASE (2018)

Article Multidisciplinary Sciences

A covalent PIN1 inhibitor selectively targets cancer cells by a dual mechanism of action

Elena Campaner et al.

NATURE COMMUNICATIONS (2017)

Article Biochemistry & Molecular Biology

Defining a Cancer Dependency Map

Aviad Tsherniak et al.

Article Multidisciplinary Sciences

Proteome-wide covalent ligand discovery in native biological systems

Keriann M. Backus et al.

NATURE (2016)

Article Biotechnology & Applied Microbiology

High-throughput identification of genotype-specific cancer vulnerabilities in mixtures of barcoded tumor cell lines

Channing Yu et al.

NATURE BIOTECHNOLOGY (2016)

Article Biochemistry & Molecular Biology

Enrichr: a comprehensive gene set enrichment analysis web server 2016 update

Maxim V. Kuleshov et al.

NUCLEIC ACIDS RESEARCH (2016)

Article Biochemical Research Methods

ProLuCID: An improved SEQUEST-like algorithm with enhanced sensitivity and specificity

T. Xu et al.

JOURNAL OF PROTEOMICS (2015)

Article Chemistry, Medicinal

Structure-based design of novel human Pin1 inhibitors (III): Optimizing affinity beyond the phosphate recognition pocket

Chuangxing Guo et al.

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2014)

Article Medicine, Research & Experimental

Prolyl-isomerase Pin1 controls normal and cancer stem cells of the breast

Alessandra Rustighi et al.

EMBO MOLECULAR MEDICINE (2014)

Article Biochemistry & Molecular Biology

Covalent docking of large libraries for the discovery of chemical probes

Nir London et al.

NATURE CHEMICAL BIOLOGY (2014)

Article Biotechnology & Applied Microbiology

Moderated estimation of fold change and dispersion for RNA-seq data with DESeq2

Michael I. Love et al.

GENOME BIOLOGY (2014)

Article Biochemical Research Methods

STAR: ultrafast universal RNA-seq aligner

Alexander Dobin et al.

BIOINFORMATICS (2013)

Article Chemistry, Medicinal

Pin1 inhibitors: Pitfalls, progress and cellular pharmacology

Jonathan D. Moore et al.

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2013)

Article Biochemistry & Molecular Biology

Pin1 Regulates the Dynamics of c-Myc DNA Binding To Facilitate Target Gene Regulation and Oncogenesis

Amy S. Farrell et al.

MOLECULAR AND CELLULAR BIOLOGY (2013)

Article Oncology

A Pin1/Mutant p53 Axis Promotes Aggressiveness in Breast Cancer

Javier E. Girardini et al.

CANCER CELL (2011)

Article Biochemical Research Methods

XDS

Wolfgang Kabsch

ACTA CRYSTALLOGRAPHICA SECTION D-BIOLOGICAL CRYSTALLOGRAPHY (2010)

Article Biochemical Research Methods

PHENIX: a comprehensive Python-based system for macromolecular structure solution

Paul D. Adams et al.

ACTA CRYSTALLOGRAPHICA SECTION D-STRUCTURAL BIOLOGY (2010)

Article Chemistry, Medicinal

Structure-based design of novel human Pin1 inhibitors (II)

Liming Dong et al.

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2010)

Article Oncology

Pin1 expression contributes to lung cancer Prognosis and carcinogenesis

Xiaogang Tan et al.

CANCER BIOLOGY & THERAPY (2010)

Article Chemistry, Medicinal

Structure-based design of novel human Pin1 inhibitors (I)

Chuangxing Guo et al.

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2009)

Article Biochemistry & Molecular Biology

Juglone inactivates cysteine-rich proteins required for progression through mitosis

Claudia Fila et al.

JOURNAL OF BIOLOGICAL CHEMISTRY (2008)

Article Biochemistry & Molecular Biology

Prolyl isomerase Pin1 is highly expressed in Her2-positive breast cancer and regulates erbB2 protein stability

Prudence B. Lam et al.

MOLECULAR CANCER (2008)

Review Cell Biology

The prolyl isomerase PIN 1: a pivotal new twist in phosphorylation signalling and disease

Kun Ping Lu et al.

NATURE REVIEWS MOLECULAR CELL BIOLOGY (2007)

Article Chemistry, Multidisciplinary

Phaser crystallographic software

Airlie J. McCoy et al.

JOURNAL OF APPLIED CRYSTALLOGRAPHY (2007)

Article Biochemistry & Molecular Biology

Structural basis for high-affinity peptide inhibition of human Pin1

Yan Zhang et al.

ACS CHEMICAL BIOLOGY (2007)

Article Biochemistry & Molecular Biology

Modeling breast cancer in vivo and ex vivo reveals an essential role of Pin1 in tumorigenesis

G Wulf et al.

EMBO JOURNAL (2004)

Article Biochemical Research Methods

Coot:: model-building tools for molecular graphics

P Emsley et al.

ACTA CRYSTALLOGRAPHICA SECTION D-STRUCTURAL BIOLOGY (2004)

Article Pathology

Prevalent overexpression of prolyl isomerase Pin1 in human cancers

L Bao et al.

AMERICAN JOURNAL OF PATHOLOGY (2004)

Review Oncology

c-MYC: More than just a matter of life and death

S Pelengaris et al.

NATURE REVIEWS CANCER (2002)

Article Biochemistry & Molecular Biology

Juglone, an inhibitor of the peptidyl-prolyl isomerase Pin1, also directly blocks transcription

SH Chao et al.

NUCLEIC ACIDS RESEARCH (2001)