4.6 Article

Chemical Degradation of Androgen Receptor (AR) Using Bicalutamide Analog-Thalidomide PROTACs

相关参考文献

注意:仅列出部分参考文献,下载原文获取全部文献信息。
Article Medicine, Research & Experimental

Androgen receptor splice variant-7 expression emerges with castration resistance in prostate cancer

Adam Sharp et al.

JOURNAL OF CLINICAL INVESTIGATION (2019)

Meeting Abstract Oncology

ARV-110: An androgen receptor PROTAC degrader for prostate cancer

Taavi Neklesa et al.

CANCER RESEARCH (2018)

Review Chemistry, Multidisciplinary

Small-Molecule Modulation of Protein Homeostasis

George M. Burslem et al.

CHEMICAL REVIEWS (2017)

Article Multidisciplinary Sciences

Phthalimide conjugation as a strategy for in vivo target protein degradation

Georg E. Winter et al.

SCIENCE (2015)

Review Oncology

Androgen receptor antagonists for prostate cancer therapy

Christine Helsen et al.

ENDOCRINE-RELATED CANCER (2014)

Article Chemistry, Medicinal

Isosteric analogs of lenalidomide and pomalidomide: Synthesis and biological activity

Alexander L. Ruchelman et al.

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2013)

Article Chemistry, Multidisciplinary

Synthesis of aryl nitriles using the stable aryl diazonium silica sulfates

Davood Habibi et al.

JOURNAL OF CHEMICAL RESEARCH (2012)

Article Biochemistry & Molecular Biology

Targeting steroid hormone receptors for ubiquitination and degradation in breast and prostate cancer

A. Rodriguez-Gonzalez et al.

ONCOGENE (2008)

Article Multidisciplinary Sciences

Structural basis for antagonism and resistance of bicalutamide in prostate cancer

CE Bohl et al.

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2005)

Review Endocrinology & Metabolism

Androgen receptor in prostate cancer

CA Heinlein et al.

ENDOCRINE REVIEWS (2004)

Review Pharmacology & Pharmacy

Androgen replacement therapy - Present and future

LJG Gooren et al.

Article Chemistry, Organic

Facile synthesis of an azido-labeled thalidomide analogue

SM Capitosti et al.

ORGANIC LETTERS (2003)

Article Biochemistry & Molecular Biology

Bicalutamide functions as an androgen receptor antagonist by assembly of a transcriptionally inactive receptor

D Masiello et al.

JOURNAL OF BIOLOGICAL CHEMISTRY (2002)

Article Multidisciplinary Sciences

Protacs: Chimeric molecules that target proteins to the Skp1-Cullin-F box complex for ubiquitination and degradation

KM Sakamoto et al.

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2001)